Abstract
We have developed a simple one‐step synthesis of 2‐chloromethyl‐1,3,4‐oxadiazoles from commercially available acylhydrazides using 1‐chloro‐2,2,2‐trimethoxyethane as a solvent under microwave irradiation.
Acknowledgments
We would like to thank Dr. David Lustig and Mr. Irving Fong for their help with liquid chromatography and mass‐spectrometry, and Dr. Brent Blackburn for helpful discussions.
Notes
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