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Research Article

A 100K well screen for a muscarinic receptor using the Epic® label-free system – a reflection on the benefits of the label-free approach to screening seven-transmembrane receptors

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Pages 163-172 | Published online: 23 Jul 2009

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Reena Halai & Matthew A Cooper. (2012) Using label-free screening technology to improve efficiency in drug discovery. Expert Opinion on Drug Discovery 7:2, pages 123-131.
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Wayne Stallaert, Arthur Christopoulos & Michel Bouvier. (2011) Ligand functional selectivity and quantitative pharmacology at G protein-coupled receptors. Expert Opinion on Drug Discovery 6:8, pages 811-825.
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Sheraz Gul & Philip Gribbon. (2010) Exemplification of the challenges associated with utilising fluorescence intensity based assays in discovery. Expert Opinion on Drug Discovery 5:7, pages 681-690.
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