Barbara Saxty & Peter J. Coombs. 2023. The Handbook of Medicinal Chemistry. The Handbook of Medicinal Chemistry
359
401
.
Nicole B. Servant, Mark E. Williams, Paul F. Brust, Huixian Tang, Melissa S. Wong, Qing Chen, Marketa Lebl-Rinnova, Sara L. Adamski-Werner, Catherine Tachdjian & Guy Servant. (2022) A Dynamic Mass Redistribution Assay for the Human Sweet Taste Receptor Uncovers G-Protein Dependent Biased Ligands. Frontiers in Pharmacology 13.
Crossref
Lala Qu, Xiuli Zhang, Jixia Wang, Han Zhou, Tao Hou, Lai Wei, Fangfang Xu & Xinmiao Liang. (2019) Phenotypic assessment and ligand screening of ETA/ETB receptors with label-free dynamic mass redistribution assay. Naunyn-Schmiedeberg's Archives of Pharmacology 393:6, pages 937-950.
Crossref
Lala Qu, Jixia Wang, Tao Hou, Han Zhou, Zhiwei Wang, Xiuli Zhang & Xinmiao Liang. (2020) Systematic characterization of AT1 receptor antagonists with label-free dynamic mass redistribution assays. Journal of Pharmacological and Toxicological Methods 102, pages 106682.
Crossref
Sean S. So, Tony Ngo, Peter Keov, Nicola J. Smith & Irina Kufareva. 2020. GPCRs. GPCRs
295
334
.
László Kiss, Attila Cselenyák & András Visegrády. (2019) Label-free drug screening assay multiplexed with an orthogonal time-resolved fluorescence labeled assay. Analytical Biochemistry 566, pages 126-132.
Crossref
Weijia Zhou, Jixia Wang, Yaopeng Zhao, Long Yu, Ye Fang, Hongli Jin, Han Zhou, Pengyu Zhang, Yanfang Liu, Xiuli Zhang & Xinmiao Liang. (2018) Discovery of β2- adrenoceptor agonists in Curcuma zedoaria Rosc using label-free cell phenotypic assay combined with two-dimensional liquid chromatography. Journal of Chromatography A 1577, pages 59-65.
Crossref
Arjun Saha, Teena Varghese, Annie Liu, Samantha J. Allen, Taraneh Mirzadegan & Michael D. Hack. (2018) An Analysis of Different Components of a High-Throughput Screening Library. Journal of Chemical Information and Modeling 58:10, pages 2057-2068.
Crossref
Y. Fang. 2019. Label-Free Monitoring of Cells in vitro. Label-Free Monitoring of Cells in vitro
189
217
.
Hanna B. Christensen, David E. Gloriam, Daniel Sejer Pedersen, Jack B. Cowland, Niels Borregaard & Hans Bräuner-Osborne. (2017) Applying label-free dynamic mass redistribution assay for studying endogenous FPR1 receptor signalling in human neutrophils. Journal of Pharmacological and Toxicological Methods 88, pages 72-78.
Crossref
Y. Fang. 2017. Comprehensive Medicinal Chemistry III. Comprehensive Medicinal Chemistry III
416
433
.
Ye Fang. (2015) Are label-free investigations the best approach to drug discovery?. Future Medicinal Chemistry 7:12, pages 1561-1564.
Crossref
Kyle C. Wilcox, Matthew R. Marunde, Aditi Das, Pauline T. Velasco, Benjamin D. Kuhns, Michael T. Marty, Haoming Jiang, Chi-Hao Luan, Stephen G. Sligar & William L. Klein. (2015) Nanoscale Synaptic Membrane Mimetic Allows Unbiased High Throughput Screen That Targets Binding Sites for Alzheimer?s-Associated A? Oligomers. PLOS ONE 10:4, pages e0125263.
Crossref
Ye Fang. (2015) Total Internal Reflection Fluorescence Quantification of Receptor Pharmacology. Biosensors 5:2, pages 223-240.
Crossref
Linda Zander Balderud, David Murray, Niklas Larsson, Uma Vempati, Stephan C. Schürer, Marcus Bjäreland & Ola Engkvist. (2015) Using the BioAssay Ontology for Analyzing High-Throughput Screening Data. SLAS Discovery 20:3, pages 402-415.
Crossref
Ye Fang. 2015. Label-Free Biosensor Methods in Drug Discovery. Label-Free Biosensor Methods in Drug Discovery
17
33
.
Xinmiao Liang, Jixia Wang, Xiuli Zhang & Ye Fang. 2015. Label-Free Biosensor Methods in Drug Discovery. Label-Free Biosensor Methods in Drug Discovery
233
252
.
Ann M. Ferrie, Vasiliy Goral, Chaoming Wang & Ye Fang. 2015. G Protein-Coupled Receptor Screening Assays. G Protein-Coupled Receptor Screening Assays
227
246
.
Manuel Grundmann & Evi Kostenis. 2015. G Protein-Coupled Receptor Screening Assays. G Protein-Coupled Receptor Screening Assays
199
213
.
Ye Fang. (2014) Label-free drug discovery. Frontiers in Pharmacology 5.
Crossref
Hannah J. Gitschier, Audrey B. Bergeron & David H. Randle. (2014) Label‐Free Cell‐Based Dynamic Mass Redistribution Assays. Current Protocols in Chemical Biology 6:1, pages 39-51.
Crossref
Xiuli Zhang, Huayun Deng, Yuansheng Xiao, Xingya Xue, Ann M. Ferrie, Elizabeth Tran, Xinmiao Liang & Ye Fang. (2014) Label-free cell phenotypic profiling identifies pharmacologically active compounds in two traditional Chinese medicinal plants. RSC Adv. 4:50, pages 26368-26377.
Crossref
Régis Méjard, Hans J. Griesser & Benjamin Thierry. (2014) Optical biosensing for label-free cellular studies. TrAC Trends in Analytical Chemistry 53, pages 178-186.
Crossref
Sang Hun Lee, Seung-min Park & Luke P. Lee. 2014. Bioelectronic Nose. Bioelectronic Nose
191
220
.
Zhan-Guo Gao & Kenneth A. Jacobson. (2013) Allosteric modulation and functional selectivity of G protein-coupled receptors. Drug Discovery Today: Technologies 10:2, pages e237-e243.
Crossref
Kenneth Lundstrom. (2013) Present and future approaches to screening of G-protein-coupled receptors. Future Medicinal Chemistry 5:5, pages 523-538.
Crossref
Andy Barker, Jason G. Kettle, Thorsten Nowak & J. Elizabeth Pease. (2013) Expanding medicinal chemistry space. Drug Discovery Today 18:5-6, pages 298-304.
Crossref
Magalie Rocheville, Julio Martin, Jeff Jerman & Evi Kostenis. 2013. Oligomerization and Allosteric Modulation in G-Protein Coupled Receptors. Oligomerization and Allosteric Modulation in G-Protein Coupled Receptors
123
142
.
Michael T. Klein, Paige N. Vinson & Colleen M. Niswender. 2013. Oligomerization and Allosteric Modulation in G-Protein Coupled Receptors. Oligomerization and Allosteric Modulation in G-Protein Coupled Receptors
1
59
.
Geoffrey Holdgate, Stefan Geschwindner, Alex Breeze, Gareth Davies, Nicola Colclough, David Temesi & Lara Ward. 2013. Protein-Ligand Interactions. Protein-Ligand Interactions
327
355
.
Reena Halai, Daniel E. Croker, Jacky Y. Suen, David P. Fairlie & Matthew A. Cooper. (2012) A Comparative Study of Impedance versus Optical Label-Free Systems Relative to Labelled Assays in a Predominantly Gi Coupled GPCR (C5aR) Signalling. Biosensors 2:3, pages 273-290.
Crossref
Stefan Geschwindner, Johan F. Carlsson & Wolfgang Knecht. (2012) Application of Optical Biosensors in Small-Molecule Screening Activities. Sensors 12:4, pages 4311-4323.
Crossref
Ru Zhang & Xin Xie. (2012) Tools for GPCR drug discovery. Acta Pharmacologica Sinica 33:3, pages 372-384.
Crossref
Yuhong Du, Jie Xu, Haian Fu & Arron S. Xu. 2012. Chemical Genomics. Chemical Genomics
245
258
.
Wayne Stallaert, Jonas F. Dorn, Emma van der Westhuizen, Martin Audet & Michel Bouvier. (2012) Impedance Responses Reveal β2-Adrenergic Receptor Signaling Pluridimensionality and Allow Classification of Ligands with Distinct Signaling Profiles. PLoS ONE 7:1, pages e29420.
Crossref
Megan Morse, Elizabeth Tran, Haiyan Sun, Robert Levenson & Ye Fang. (2011) Ligand-Directed Functional Selectivity at the Mu Opioid Receptor Revealed by Label-Free Integrative Pharmacology On-Target. PLoS ONE 6:10, pages e25643.
Crossref
Charles A Lunn. (2011) A new look at membrane protein binding. Nature Biotechnology 29:4, pages 328-329.
Crossref
Sung-Hou Lee. (2011) Platform Technologies for Research on the G Protein Coupled Receptor: Applications to Drug Discovery Research. Biomolecules and Therapeutics 19:1, pages 1-8.
Crossref
Ye Fang. (2011) Label-Free Biosensors for Cell Biology. International Journal of Electrochemistry 2011, pages 1-16.
Crossref
Charles A Lunn. (2010) Label-free screening assays: a strategy for finding better drug candidates. Future Medicinal Chemistry 2:11, pages 1703-1716.
Crossref
Geoff A. Holdgate, Malcolm Anderson, Fredrik Edfeldt & Stefan Geschwindner. (2010) Affinity-based, biophysical methods to detect and analyze ligand binding to recombinant proteins: Matching high information content with high throughput. Journal of Structural Biology 172:1, pages 142-157.
Crossref
Ralf Schröder, Nicole Janssen, Johannes Schmidt, Anna Kebig, Nicole Merten, Stephanie Hennen, Anke Müller, Stefanie Blättermann, Marion Mohr-Andrä, Sabine Zahn, Jörg Wenzel, Nicola J Smith, Jesús Gomeza, Christel Drewke, Graeme Milligan, Klaus Mohr & Evi Kostenis. (2010) Deconvolution of complex G protein–coupled receptor signaling in live cells using dynamic mass redistribution measurements. Nature Biotechnology 28:9, pages 943-949.
Crossref
Julio Martin. (2010) Label‐Free Imaging and Temporal Signature in Phenotypic Cellular Assays: A New Approach to High‐Content Screening. Current Protocols in Pharmacology 50:1.
Crossref
Oliver Nayler, Magdalena Birker‐Robaczewska & John Gatfield. 2010. GPCR Molecular Pharmacology and Drug Targeting. GPCR Molecular Pharmacology and Drug Targeting
252
275
.
William Kisaalita. 2010. 3D Cell-Based Biosensors in Drug Discovery Programs. 3D Cell-Based Biosensors in Drug Discovery Programs
221
251
.