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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 38, 2023 - Issue 1
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Research Paper

Design and statistical optimisation of emulsomal nanoparticles for improved anti-SARS-CoV-2 activity of N-(5-nitrothiazol-2-yl)-carboxamido candidates: in vitro and in silico studies

Ahmed A. Al-Karmalawya Pharmaceutical Chemistry Department, Faculty of Pharmacy, Ahram Canadian University, Giza, EgyptCorrespondence[email protected]
ORCID Iconhttps://orcid.org/0000-0002-8173-6073View further author information
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Dalia S. El-Gamila Pharmaceutical Chemistry Department, Faculty of Pharmacy, Ahram Canadian University, Giza, EgyptView further author information
,
Rabeh El-Sheshenyb Water Pollution Research Department, The Center of Scientific Excellence for Influenza Viruses, Environmental Research Institute, National Research Centre, Giza, EgyptView further author information
,
Marwa Sharakyc Cancer Biology Department, Pharmacology Unit, National Cancer Institute (NCI), Cairo University, Cairo, EgyptView further author information
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Radwan Alnajjard Department of Chemistry, Faculty of Science, University of Benghazi, Benghazi, Libya;e Faculty of Pharmacy, Libyan International Medical University, Benghazi, Libya;f Department of Chemistry, University of Cape Town, Rondebosch, South AfricaView further author information
,
Omnia Kutkatb Water Pollution Research Department, The Center of Scientific Excellence for Influenza Viruses, Environmental Research Institute, National Research Centre, Giza, EgyptView further author information
,
Yassmin Moatasimb Water Pollution Research Department, The Center of Scientific Excellence for Influenza Viruses, Environmental Research Institute, National Research Centre, Giza, EgyptView further author information
,
Mohamed Elagawanyg Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Damanhour University, Damanhour, EgyptView further author information
,
Sara T. Al-Rashoodh Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh, Saudi ArabiaView further author information
,
Faizah A. Binjubairh Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh, Saudi ArabiaView further author information
,
Wagdy M. Eldehnai Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, Egypt;j School of Biotechnology, Badr University in Cairo, Badr City, EgyptORCID Iconhttps://orcid.org/0000-0001-6996-4017View further author information
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Ayman M. Noreddink Department of Internal Medicine, School of Medicine, University of California Irvine, Irvine, CA, USA;l Department of Clinical Pharmacy, Faculty of Pharmacy, Ahram Canadian University, Giza, EgyptView further author information
&
Mohamed Y. Zakariam Department of Pharmaceutics and Industrial Pharmacy, Faculty of Pharmacy, Port Said University, Port Said, EgyptView further author information
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Article: 2202357 | Received 03 Feb 2023, Accepted 07 Apr 2023, Published online: 24 Apr 2023

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Mai H. ElNaggar, Abdullah A. Elgazar, Ghada Gamal, Shimaa M. Hamed, Zainab M. Elsayed, Mohamed K. El-Ashrey, Amira Abood, Mahmoud A. El Hassab, Ahmed M. Soliman, Ramadan A. El-Domany, Farid A. Badria, Claudiu T. Supuran & Wagdy M. Eldehna. (2023) Identification of sulphonamide-tethered N-((triazol-4-yl)methyl)isatin derivatives as inhibitors of SARS-CoV-2 main protease. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Baohui Zhu, Ryota Ouda, Paul de Figueiredo & Koichi S Kobayashi. (2023) ORF6, a repressor of the MHC class I pathway: new molecular target for SARS-CoV-2 drug discovery?. Expert Opinion on Therapeutic Targets 27:8, pages 639-644.
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Articles from other publishers (2)

Ahmed A. Al-Karmalawy, Mai H. A. Mousa, Marwa Sharaky, Mai A. E. Mourad, Ahmed M. El-Dessouki, Amir O. Hamouda, Radwan Alnajjar, Abdelmoneim A. Ayed, Moataz A. Shaldam & Haytham O. Tawfik. (2023) Lead Optimization of BIBR1591 To Improve Its Telomerase Inhibitory Activity: Design and Synthesis of Novel Four Chemical Series with In Silico, In Vitro, and In Vivo Preclinical Assessments. Journal of Medicinal Chemistry 67:1, pages 492-512.
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Saad Shaaban, Ahmed A. Al-Karmalawy, Abdulrahman G. Alhamzani, Mortaga M. Abou–Krisha, Mahmoud A. Al–Qudah & Tarek A. Yousef. (2023) Synthesis and Molecular Docking Analysis of New Thiazo-isoindolinedione Hybrids as Potential Inhibitors of the SARS-CoV-2 Main Protease. Oriental Journal Of Chemistry 39:4, pages 913-918.
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