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Review

Trk kinase inhibitors as new treatments for cancer and pain

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Pages 305-319 | Published online: 27 Mar 2009

Keep up to date with the latest research on this topic with citation updates for this article.

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Xiaoyun Wu, Qinlan Li, Shanhe Wan & Jiajie Zhang. (2021) Molecular dynamics simulation and free energy calculation studies of the binding mechanism of allosteric inhibitors with TrkA kinase. Journal of Biomolecular Structure and Dynamics 39:1, pages 202-208.
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Justin J. Bailey, Ralf Schirrmacher, Kristen Farrell & Vadim Bernard-Gauthier. (2017) Tropomyosin receptor kinase inhibitors: an updated patent review for 2010-2016 – Part II. Expert Opinion on Therapeutic Patents 27:7, pages 831-849.
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Vadim Bernard-Gauthier & Ralf Schirrmacher. (2016) Evaluation of WO2015042088 A1 - a novel urea-based scaffold for TrkA inhibition. Expert Opinion on Therapeutic Patents 26:2, pages 291-295.
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Clive McCarthy & Edward Walker. (2014) Tropomyosin receptor kinase inhibitors: a patent update 2009 – 2013. Expert Opinion on Therapeutic Patents 24:7, pages 731-744.
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Servane Tauszig-Delamasure & Jimena Bouzas-Rodriguez. (2011) Targeting neurotrophin-3 and its dependence receptor tyrosine kinase receptor C: a new antitumoral strategy. Expert Opinion on Therapeutic Targets 15:7, pages 847-858.
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Yasuhiro Indo. (2010) Nerve growth factor, pain, itch and inflammation: lessons from congenital insensitivity to pain with anhidrosis. Expert Review of Neurotherapeutics 10:11, pages 1707-1724.
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