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Review

Estrogen receptor modulator review

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Pages 559-572 | Published online: 25 Apr 2006

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Ilaria Paterni, Simone Bertini, Carlotta Granchi, Marco Macchia & Filippo Minutolo. (2013) Estrogen receptor ligands: a patent review update. Expert Opinion on Therapeutic Patents 23:10, pages 1247-1271.
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A. Chandrasekaran, S. Ahmad, L. Shen, W. DeMaio, T. Hultin & J. Scatina. (2010) Disposition of bazedoxifene in rats. Xenobiotica 40:8, pages 578-585.
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Michael L Mohler, Ramesh Narayanan, Christopher C Coss, Kejiang Hu, Yali He, Zhongzhi Wu, Seoung-Soo Hong, Dong Jin Hwang, Duane D Miller & James T Dalton. (2010) Estrogen receptor β selective nonsteroidal estrogens: seeking clinical indications. Expert Opinion on Therapeutic Patents 20:4, pages 507-534.
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Articles from other publishers (16)

Kassrin Tangdenpaisal, Kanokpish Chuayboonsong, Patchaya Sukjarean, Varisa Katesampao, Nok Noiphrom, Somsak Ruchirawat & Poonsakdi Ploypradith. (2015) Synthesis of C4C5 Cycloalkyl-Fused and C6-Modified Chromans via ortho -Quinone Methides . Chemistry - An Asian Journal 10:4, pages 1050-1064.
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Amarjit Luniwal, Rachael Jetson & Paul Erhardt. 2012. Analogue‐Based Drug Discovery III. Analogue‐Based Drug Discovery III 165 185 .
Suttipol Radomkit, Pakornwit Sarnpitak, Jumreang Tummatorn, Paratchata Batsomboon, Somsak Ruchirawat & Poonsakdi Ploypradith. (2011) Pt(IV)-catalyzed generation and [4+2]-cycloaddition reactions of o-quinone methides. Tetrahedron 67:21, pages 3904-3914.
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Filippo Minutolo, Marco Macchia, Benita S. Katzenellenbogen & John A. Katzenellenbogen. (2011) Estrogen receptor β ligands: Recent advances and biomedical applications. Medicinal Research Reviews 31:3, pages 364-442.
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Li Shen, Syed Ahmad, SeongHee Park, William DeMaio, Aram Oganesian, Theresa Hultin, JoAnn Scatina, Peter Bungay & Appavu Chandrasekaran. (2010) In Vitro Metabolism, Permeability, and Efflux of Bazedoxifene in Humans. Drug Metabolism and Disposition 38:9, pages 1471-1479.
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Jumreang Tummatorn, Somsak Ruchirawat & Poonsakdi Ploypradith. (2010) A Convergent General Strategy for the Functionalized 2‐Aryl Cycloalkyl‐Fused Chromans: Intramolecular Hetero‐Diels–Alder Reactions of ortho ‐Quinone Methides . Chemistry – A European Journal 16:5, pages 1445-1448.
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Paratchata Batsomboon, Wong Phakhodee, Somsak Ruchirawat & Poonsakdi Ploypradith. (2009) Generation of ortho -Quinone Methides by p -TsOH on Silica and Their Hetero-Diels−Alder Reactions with Styrenes . The Journal of Organic Chemistry 74:10, pages 4009-4012.
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Hugh S. Taylor. (2009) Designing the ideal selective estrogen receptor modulator-an achievable goal?. Menopause 16:3, pages 609-615.
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Yogendra Kharode, Peter V. N. Bodine, Christopher P. Miller, C. Richard Lyttle & Barry S. Komm. (2008) The Pairing of a Selective Estrogen Receptor Modulator, Bazedoxifene, with Conjugated Estrogens as a New Paradigm for the Treatment of Menopausal Symptoms and Osteoporosis Prevention. Endocrinology 149:12, pages 6084-6091.
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Gerrit H. Veeneman. 2008. Nuclear Receptors as Drug Targets. Nuclear Receptors as Drug Targets 65 126 .
Timothy I. Richardson, Jeffrey A. Dodge, Yong Wang, Jim D. Durbin, Venkatesh Krishnan & Bryan H. Norman. (2007) Benzopyrans as selective estrogen receptor β agonists (SERBAs). Part 5: Combined A- and C-ring structure–activity relationship studies. Bioorganic & Medicinal Chemistry Letters 17:20, pages 5563-5566.
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Bryan H. Norman, Timothy I. Richardson, Jeffrey A. Dodge, Lance A. Pfeifer, Gregory L. Durst, Yong Wang, Jim D. Durbin, Venkatesh Krishnan, Sean R. Dinn, Shengquan Liu, John E. Reilly & Kendal T. Ryter. (2007) Benzopyrans as selective estrogen receptor β agonists (SERBAs). Part 4: Functionalization of the benzopyran A-ring. Bioorganic & Medicinal Chemistry Letters 17:18, pages 5082-5085.
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Timothy I. Richardson, Jeffrey A. Dodge, Gregory L. Durst, Lance A. Pfeifer, Jikesh Shah, Yong Wang, Jim D. Durbin, Venkatesh Krishnan & Bryan H. Norman. (2007) Benzopyrans as selective estrogen receptor β agonists (SERBAs). Part 3: Synthesis of cyclopentanone and cyclohexanone intermediates for C-ring modification. Bioorganic & Medicinal Chemistry Letters 17:17, pages 4824-4828.
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An T. Vu, Alison N. Campbell, Heather A. Harris, Rayomand J. Unwalla, Eric S. Manas & Richard E. Mewshaw. (2007) ERβ ligands. Part 6: 6H-Chromeno[4,3-b]quinolines as a new series of estrogen receptor β-selective ligands. Bioorganic & Medicinal Chemistry Letters 17:14, pages 4053-4056.
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Timothy I. Richardson, Bryan H. Norman, Charles W. Lugar, Scott A. Jones, Yong Wang, Jim D. Durbin, Venkatesh Krishnan & Jeffrey A. Dodge. (2007) Benzopyrans as selective estrogen receptor β agonists (SERBAs). Part 2: Structure–activity relationship studies on the benzopyran scaffold. Bioorganic & Medicinal Chemistry Letters 17:13, pages 3570-3574.
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John W. Ullrich, Rayomand J. Unwalla, Robert R. SinghausJr.Jr., Heather A. Harris & Richard E. Mewshaw. (2007) Estrogen receptor β ligands: Design and synthesis of new 2-phenyl-isoindole-1,3-diones. Bioorganic & Medicinal Chemistry Letters 17:1, pages 118-122.
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