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Developments around the bioactive diketopiperazines: a patent review

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Pages 1415-1433 | Published online: 21 Aug 2013

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Sangluo Chen, Di Zhang, Mengxuan Chen, Zhizhen Zhang & Xiao-Yuan Lian. (2020) A rare diketopiperazine glycoside from marine-sourced Streptomyces sp. ZZ446. Natural Product Research 34:7, pages 1046-1050.
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Xuewei Ye, Weiyun Chai, Xiao-Yuan Lian & Zhizhen Zhang. (2017) Novel propanamide analogue and antiproliferative diketopiperazines from mangrove Streptomyces sp. Q24. Natural Product Research 31:12, pages 1390-1396.
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Xue-Song Yin, Wei-Yi Qi & Bing-Feng Shi. (2021) Synthesis of tryptophan-containing 2,5-diketopiperazines via sequential C–H activation: total syntheses of tryprostatin A, maremycins A and B . Chemical Science 12:39, pages 13137-13143.
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Dan-dan Li, Ying Wang, Eun La Kim, Jongki Hong & Jee H. Jung. (2021) Neuroprotective Effect of Cyclo-(L-Pro-L-Phe) Isolated from the Jellyfish-Derived Fungus Aspergillus flavus. Marine Drugs 19:8, pages 417.
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Heegyu Kim, Ji-Yeon Hwang, Jongheon Shin & Ki-Bong Oh. (2019) Inhibitory Effects of Diketopiperazines from Marine-Derived Streptomyces puniceus on the Isocitrate Lyase of Candida albicans. Molecules 24:11, pages 2111.
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Hyejin Kang, Sae-Kwang Ku, Hyukjae Choi & Jong-Sup Bae. (2016) Three diketopiperazines from marine-derived bacteria inhibit LPS-induced endothelial inflammatory responses. Bioorganic & Medicinal Chemistry Letters 26:8, pages 1873-1876.
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Shigeki Sano & Michiyasu Nakao. (2015) Chemistry of 2,5-Diketopiperazine and Its Bis-Lactim Ether: A Brief Review. HETEROCYCLES 91:7, pages 1349.
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Shengrong Liao, Ying Xu, Yong Tang, Junfeng Wang, Xuefeng Zhou, Liang Xu & Yonghong Liu. (2015) Design, synthesis and biological evaluation of soluble 2,5-diketopiperazines derivatives as potential antifouling agents. RSC Advances 5:63, pages 51020-51026.
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