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Drug Evaluations

Lixivaptan: a novel vasopressin receptor antagonist

, MD, & , MD
Pages 657-662 | Published online: 21 Apr 2009

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Brendan T Bowman & Mitchell H Rosner. (2013) Lixivaptan – an evidence-based review of its clinical potential in the treatment of hyponatremia. Core Evidence 8, pages 47-56.
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Haitham Alrabiah, Mohammed Abunassif, Sabry Attia & Gamal Abdel-Hafiz Mostafa. (2018) A new selective, and sensitive method for the determination of lixivaptan, a vasopressin 2 (V2)-receptor antagonist, in mouse plasma and its application in a pharmacokinetic study. Open Chemistry 16:1, pages 614-620.
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Adnan A. Kadi, Haitham Alrabiah, Mohamed W. Attwa, Sabry Attia & Gamal A. E. Mostafa. (2017) Development and validation of HPLC-MS/MS method for the determination of lixivaptan in mouse plasma and its application in a pharmacokinetic study. Biomedical Chromatography 31:11, pages e4007.
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Hidetsugu Tabata, Jun Nakagomi, Daisuke Morizono, Tetsuta Oshitari, Hideyo Takahashi & Hideaki Natsugari. (2011) Atropisomerism in the Vaptan Class of Vasopressin Receptor Ligands: The Active Conformation Recognized by the Receptor. Angewandte Chemie International Edition 50:13, pages 3075-3079.
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Alexander Geppert. (2010) Gleiche Therapien bei kardiogenem und septischem Schock?. Wiener klinisches Magazin 13:2, pages 24-29.
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A. Geppert. (2009) Einsatz von inotropen und vasopressorischen Substanzen bei der akut dekompensierten HerzinsuffizienzUse of inotropic and vasopressor substances in acute decompensated heart failure. Intensivmedizin und Notfallmedizin 46:6, pages 407-414.
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