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Sachin B. Pandya, Bhavesh N. Socha, Kaushik P. Chaudhary, Rahul P. Dubey, Bhavin R. Chavda, Urmila H. Patel, Maheshkumar K. Patel, Nikita J. Patel & Bhupesh S. Bhatt. (2021) Combined experimental and computational studies on molecular structure of nickel complex of 4-amino-N-(1, 3-thiazol-2-yl) benzenesulfonamide with coordinated pyridine. Inorganic and Nano-Metal Chemistry 51:9, pages 1280-1290.
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Nadya Jammal, Caitlin R. Rausch, Tapan M. Kadia & Naveen Pemmaraju. (2020) Cell cycle inhibitors for the treatment of acute myeloid leukemia: a review of phase 2 & 3 clinical trials. Expert Opinion on Emerging Drugs 25:4, pages 491-499.
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Kirna Devi & Pamita Awasthi. (2020) Sulfonamide phenylalanine (SPA) series of analogues as an antibacterial, antifungal, anticancer agents along with p53 tumor suppressor-DNA complex inhibitor – part 1. Journal of Biomolecular Structure and Dynamics 38:14, pages 4081-4097.
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Claudiu T. Supuran. (2018) Carbonic anhydrase inhibitors as emerging agents for the treatment and imaging of hypoxic tumors. Expert Opinion on Investigational Drugs 27:12, pages 963-970.
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Rahul P. Dubey, Urmila H. Patel & Bharatkumar D. Patel. (2018) Study on molecular structure, Spectral investigations, NBO, NLO, Hirshfeld surface analysis and Homo-Lumo energy of silver complex of 4-Amino-N-(2,6-dimethoxypyrimidin-4-yl)benzenesulfonamide. Inorganic and Nano-Metal Chemistry 48:2, pages 110-119.
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Thurpu Raghavender Reddy, Suresh Kumar Battina & Sudhir Kashyap. (2015) Zn(II) Triflate-Catalyzed N-Glycosylation: Synthesis of Sulfonamide and Amide Functionalized 2,3-Unsaturated Glycosides. Journal of Carbohydrate Chemistry 34:3, pages 133-144.
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Sonia Del Prete, Viviana De Luca, Daniela Vullo, Andrea Scozzafava, Vincenzo Carginale, Claudiu T. Supuran & Clemente Capasso. (2014) Biochemical characterization of the γ-carbonic anhydrase from the oral pathogen Porphyromonas gingivalis, PgiCA. Journal of Enzyme Inhibition and Medicinal Chemistry 29:4, pages 532-537.
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Clemente Capasso & Claudiu T. Supuran. (2014) Sulfa and trimethoprim-like drugs – antimetabolites acting as carbonic anhydrase, dihydropteroate synthase and dihydrofolate reductase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 29:3, pages 379-387.
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Jinhe Pan, Joseph Lau, Felix Mesak, Navjit Hundal, Maral Pourghiasian, Zhibo Liu, François Bénard, Shoukat Dedhar, Claudiu T. Supuran & Kuo-Shyan Lin. (2014) Synthesis and evaluation of 18F-labeled carbonic anhydrase IX inhibitors for imaging with positron emission tomography. Journal of Enzyme Inhibition and Medicinal Chemistry 29:2, pages 249-255.
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Asif Husain & Diwakar Madhesia. (2012) Heterocyclic compounds as carbonic anhydrase inhibitor. Journal of Enzyme Inhibition and Medicinal Chemistry 27:6, pages 773-783.
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Claudiu T Supuran. (2012) Amide derivatives of benzene-sulfonanilide, pharmaceutical composition thereof and method for cancer treatment using the same (US20120095092). Expert Opinion on Therapeutic Patents 22:10, pages 1251-1255.
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Fabrizio Carta, Andrea Scozzafava & Claudiu T Supuran. (2012) Sulfonamides: a patent review (2008 – 2012). Expert Opinion on Therapeutic Patents 22:7, pages 747-758.
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Mohammed K. Abdel-Hamid, Atef A. Abdel-Hafez, Nawal A. El-Koussi & Nadia M. Mahfouz. (2009) Quantitative structure–activity relationship (QSAR) studies on a series of 1,3,4-thiadiazole-2-thione derivatives as tumor-associated carbonic anhydrase IX inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 24:3, pages 722-729.
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Pedro
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D. Bravo. (2008) Sulfonamidoglycosylation of Methyl Glycosides Employing Perchloric Acid Supported on Silica Gel. Journal of Carbohydrate Chemistry 27:3, pages 141-147.
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Neeraj Mahindroo, Jing-Ping Liou, Jang-Yang Chang & Hsing-Pang Hsieh. (2006) Antitubulin agents for the treatment of cancer – a medicinal chemistry update. Expert Opinion on Therapeutic Patents 16:5, pages 647-691.
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Brian W Clare & Claudiu T Supuran. (2006) A perspective on quantitative structure–activity relationships and carbonic anhydrase inhibitors. Expert Opinion on Drug Metabolism & Toxicology 2:1, pages 113-137.
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Silvia Pastorekova, Daniela Vullo, Angela Casini, Andrea Scozzafava, Jaromir Pastorek, Isao Nishimori & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors: Inhibition of the tumor-associated isozymes IX and XII with polyfluorinated aromatic/heterocyclic sulfonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 20:3, pages 211-217.
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Peter M Fischer & Athos Gianella-Borradori. (2005) Recent progress in the discovery and development of cyclin-dependent kinase inhibitors. Expert Opinion on Investigational Drugs 14:4, pages 457-477.
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Olcay Hİsar, Şükrü Beydemİr, İlhami Gülçİn, Ö. İrfan Küfrevİoğlu & Claudiu T. Supuran. (2005) Effects of low molecular weight plasma inhibitors of rainbow trout (Oncorhynchus mykiss) on human erythrocyte carbonic anhydrase-II isozyme activity in vitro and rat erythrocytes in vivo. Journal of Enzyme Inhibition and Medicinal Chemistry 20:1, pages 35-39.
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Özen Özensoy, Semra Isik, Oktay Arslan, Mikail Arslan, Andrea Scozzafava & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors. Inhibition of red blood cell ostrich (Struthio camelus) carbonic anhydrase with a series of aromatic and heterocyclic sulfonamides. Journal of Enzyme Inhibition and Medicinal Chemistry 20:4, pages 383-387.
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Jean-Yves Winum, Andrea Scozzafava, Jean-Louis Montero & Claudiu T Supuran. (2004) Therapeutic applications of sulfamates. Expert Opinion on Therapeutic Patents 14:9, pages 1273-1308.
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Andrea Scozzafava, Antonio Mastrolorenzo & Claudiu T Supuran. (2004) Modulation of carbonic anhydrase activity and its applications in therapy. Expert Opinion on Therapeutic Patents 14:5, pages 667-702.
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Peter M Fischer & Athos Gianella-Borradori. (2003) CDK inhibitors in clinical development for the treatment of cancer. Expert Opinion on Investigational Drugs 12:6, pages 955-970.
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Jean-Yves Winum, Alfonso Maresca, Fabrizio Carta, Andrea Scozzafava & Claudiu T. Supuran. (2012) Polypharmacology of sulfonamides: pazopanib, a multitargeted receptor tyrosine kinase inhibitor in clinical use, potently inhibits several mammalian carbonic anhydrases. Chemical Communications 48:66, pages 8177.
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Fatemeh Bootorabi, Joonas Haapasalo, Elona Smith, Hannu Haapasalo & Seppo Parkkila. (2011) Carbonic anhydrase VII–a potential prognostic marker in gliomas. Health 03:01, pages 6-12.
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Anthony Bertucci, Alessio Innocenti, Andrea Scozzafava, Sylvie Tambutté, Didier Zoccola & Claudiu T. Supuran. (2011) Carbonic anhydrase inhibitors. Inhibition studies with anions and sulfonamides of a new cytosolic enzyme from the scleractinian coral Stylophora pistillata. Bioorganic & Medicinal Chemistry Letters 21:2, pages 710-714.
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Kristiina Nordfors, Joonas Haapasalo, Miikka Korja, Anssi Niemelä, Jukka Laine, Anna-Kaisa Parkkila, Silvia Pastorekova, Jaromir Pastorek, Abdul Waheed, William S Sly, Seppo Parkkila & Hannu Haapasalo. (2010) The tumour-associated carbonic anhydrases CA II, CA IX and CA XII in a group of medulloblastomas and supratentorial primitive neuroectodermal tumours: an association of CA IX with poor prognosis. BMC Cancer 10:1.
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Carlos A. Témpera, Pedro A. Colinas & Rodolfo D. Bravo. (2010) Efficient synthesis of 2,3-unsaturated sulfonamidoglycosides by Amberlyst 15. Tetrahedron Letters 51:41, pages 5372-5374.
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Deniz Ekinci, Hüseyin Çavdar, Oktay Talaz, Murat Şentürk & Claudiu T. Supuran. (2010) NO-releasing esters show carbonic anhydrase inhibitory action against human isoforms I and II. Bioorganic & Medicinal Chemistry 18:10, pages 3559-3563.
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Daniel A. Tennant, Raúl V. Durán & Eyal Gottlieb. (2010) Targeting metabolic transformation for cancer therapy. Nature Reviews Cancer 10:4, pages 267-277.
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Alessio Innocenti, S. Beyza Öztürk Sarıkaya, İlhami Gülçin & Claudiu T. Supuran. (2010) Carbonic anhydrase inhibitors. Inhibition of mammalian isoforms I–XIV with a series of natural product polyphenols and phenolic acids. Bioorganic & Medicinal Chemistry 18:6, pages 2159-2164.
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Laura Ciani, Alessandro Cecchi, Claudia Temperini, Claudiu T. Supuran & Sandra Ristori. (2009) Dissecting the Inhibition Mechanism of Cytosolic versus Transmembrane Carbonic Anhydrases by ESR. The Journal of Physical Chemistry B 113:42, pages 13998-14005.
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Anthony Bertucci, Alessio Innocenti, Didier Zoccola, Andrea Scozzafava, Sylvie Tambutté & Claudiu T. Supuran. (2009) Carbonic anhydrase inhibitors. Inhibition studies of a coral secretory isoform by sulfonamides. Bioorganic & Medicinal Chemistry 17:14, pages 5054-5058.
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Saori Morishita, Isao Nishimori, Tomoko Minakuchi, Saburo Onishi, Hiroaki Takeuchi, Tetsuro Sugiura, Daniela Vullo, Andrea Scozzafava & Claudiu T. Supuran. (2008) Cloning, polymorphism, and inhibition of β-carbonic anhydrase of Helicobacter pylori. Journal of Gastroenterology 43:11, pages 849-857.
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Esra Bayram, Murat Senturk, O. Irfan Kufrevioglu & Claudiu T. Supuran. (2008) In vitro inhibition of salicylic acid derivatives on human cytosolic carbonic anhydrase isozymes I and II. Bioorganic & Medicinal Chemistry 16:20, pages 9101-9105.
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Claudiu T. Supuran. (2008) Carbonic anhydrase inhibitors: possible anticancer drugs with a novel mechanism of action. Drug Development Research 69:6, pages 297-303.
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Alessio Innocenti, Daniela Vullo, Andrea Scozzafava & Claudiu T. Supuran. (2008) Carbonic anhydrase inhibitors: Inhibition of mammalian isoforms I–XIV with a series of substituted phenols including paracetamol and salicylic acid. Bioorganic & Medicinal Chemistry 16:15, pages 7424-7428.
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Alessio Innocenti, Alfonso Maresca, Andrea Scozzafava & Claudiu T. Supuran. (2008) Carbonic anhydrase inhibitors: Thioxolone versus sulfonamides for obtaining isozyme-selective inhibitors?. Bioorganic & Medicinal Chemistry Letters 18:14, pages 3938-3941.
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Anne Thiry, Claudiu T. Supuran, Bernard Masereel & Jean-Michel Dogné. (2008) Recent Developments of Carbonic Anhydrase Inhibitors as Potential Anticancer Drugs. Journal of Medicinal Chemistry 51:11, pages 3051-3056.
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Alessandro Cecchi, Laura Ciani, Jean-Yves Winum, Jean-Louis Montero, Andrea Scozzafava, Sandra Ristori & Claudiu T. Supuran. (2008) Carbonic anhydrase inhibitors: Design of spin-labeled sulfonamides incorporating TEMPO moieties as probes for cytosolic or transmembrane isozymes. Bioorganic & Medicinal Chemistry Letters 18:12, pages 3475-3480.
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Jean‐Yves Winum, Marouan Rami, Andrea Scozzafava, Jean‐Louis Montero & Claudiu Supuran. (2007) Carbonic anhydrase IX: A new druggable target for the design of antitumor agents. Medicinal Research Reviews 28:3, pages 445-463.
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Claudia Temperini, Alessandro Cecchi, Andrea Scozzafava & Claudiu T. Supuran. (2008) Carbonic anhydrase inhibitors. Interaction of indapamide and related diuretics with 12 mammalian isozymes and X-ray crystallographic studies for the indapamide–isozyme II adduct. Bioorganic & Medicinal Chemistry Letters 18:8, pages 2567-2573.
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Vijay M. Krishnamurthy, George K. Kaufman, Adam R. Urbach, Irina Gitlin, Katherine L. Gudiksen, Douglas B. Weibel & George M. Whitesides. (2008) Carbonic Anhydrase as a Model for Biophysical and Physical-Organic Studies of Proteins and Protein−Ligand Binding. Chemical Reviews 108:3, pages 946-1051.
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Carmen Avendaño & J. Carlos Menéndez. 2008. Medicinal Chemistry of Anticancer Drugs. Medicinal Chemistry of Anticancer Drugs
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Lyudmila A. Vereshchagina, Orit Scharf & A. Dimitrios Colevas. 2008. The Role of Microtubules in Cell Biology, Neurobiology, and Oncology. The Role of Microtubules in Cell Biology, Neurobiology, and Oncology
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Michaela Pojarová, Doris Kaufmann, Robert Gastpar, Tsuyuki Nishino, Przemyslaw Reszka, Patrick J. Bednarski & Erwin von Angerer. (2007) [(2-Phenylindol-3-yl)methylene]propanedinitriles inhibit the growth of breast cancer cells by cell cycle arrest in G2/M phase and apoptosis. Bioorganic & Medicinal Chemistry 15:23, pages 7368-7379.
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Erol Eroglu & Hasan Türkmen. (2007) A DFT-based quantum theoretic QSAR study of aromatic and heterocyclic sulfonamides as carbonic anhydrase inhibitors against isozyme, CA-II. Journal of Molecular Graphics and Modelling 26:4, pages 701-708.
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Pedro A. Colinas & Rodolfo D. Bravo. (2007) Ferrier sulfonamidoglycosylation of d-glycals. Carbohydrate Research 342:15, pages 2297-2302.
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Mohammed K. Abdel-Hamid, Atef A. Abdel-Hafez, Nawal A. El-Koussi, Nadia M. Mahfouz, Alessio Innocenti & Claudiu T. Supuran. (2007) Design, synthesis, and docking studies of new 1,3,4-thiadiazole-2-thione derivatives with carbonic anhydrase inhibitory activity. Bioorganic & Medicinal Chemistry 15:22, pages 6975-6984.
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Rhoda Molife, Ian Collins, Paul Workman & Stan B. Kaye. 2005. The Cancer Handbook. The Cancer Handbook.
Joonas Haapasalo, Kristiina Nordfors, Sally Järvelä, Helena Bragge, Immo Rantala, Anna-Kaisa Parkkila, Hannu Haapasalo & Seppo Parkkila. (2007) Carbonic anhydrase II in the endothelium of glial tumors: A potential target for therapy. Neuro-Oncology 9:3, pages 308-313.
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Jean-Yves Winum, Claudia Temperini, Khaled El Cheikh, Alessio Innocenti, Daniela Vullo, Samuele Ciattini, Jean-Louis Montero, Andrea Scozzafava & Claudiu T. Supuran. (2006) Carbonic Anhydrase Inhibitors: Clash with Ala65 as a Means for Designing Inhibitors with Low Affinity for the Ubiquitous Isozyme II, Exemplified by the Crystal Structure of the Topiramate Sulfamide Analogue. Journal of Medicinal Chemistry 49:24, pages 7024-7031.
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Alexander Weber, Markus Böhm, Claudiu T. Supuran, Andrea Scozzafava, Christoph A. Sotriffer & Gerhard Klebe. (2006) 3D QSAR Selectivity Analyses of Carbonic Anhydrase Inhibitors: Insights for the Design of Isozyme Selective Inhibitors. Journal of Chemical Information and Modeling 46:6, pages 2737-2760.
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Jean-Yves Winum, Andrea Scozzafava, Jean-Louis Montero & Claudiu T. Supuran. (2006) Therapeutic potential of sulfamides as enzyme inhibitors. Medicinal Research Reviews 26:6, pages 767-792.
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Claudia Temperini, Andrea Scozzafava, Daniela Vullo & Claudiu T. Supuran. (2006)
Carbonic Anhydrase Activators. Activation of Isozymes I, II, IV, VA, VII, and XIV with
L
‐ and
D
‐Histidine and Crystallographic Analysis of Their Adducts with Isoform II: Engineering Proton‐Transfer Processes within the Active Site of an Enzyme
. Chemistry – A European Journal 12:27, pages 7057-7066.
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Franciszek Sączewski, Jarosław Sławiński, Anita Kornicka, Zdzisław Brzozowski, Elżbieta Pomarnacka, Alessio Innocenti, Andrea Scozzafava & Claudiu T. Supuran. (2006) Carbonic anhydrase inhibitors. Inhibition of the cytosolic human isozymes I and II, and the transmembrane, tumor-associated isozymes IX and XII with substituted aromatic sulfonamides activatable in hypoxic tumors. Bioorganic & Medicinal Chemistry Letters 16:18, pages 4846-4851.
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Claudia Temperini, Andrea Scozzafava, Daniela Vullo & Claudiu T. Supuran. (2006)
Carbonic Anhydrase Activators. Activation of Isoforms I, II, IV, VA, VII, and XIV with
l
- and
d
-Phenylalanine and Crystallographic Analysis of Their Adducts with Isozyme II: Stereospecific Recognition within the Active Site of an Enzyme and Its Consequences for the Drug Design
. Journal of Medicinal Chemistry 49:10, pages 3019-3027.
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Sally-Ann Poulsen & Laurent F. Bornaghi. (2006) Fragment-based drug discovery of carbonic anhydrase II inhibitors by dynamic combinatorial chemistry utilizing alkene cross metathesis. Bioorganic & Medicinal Chemistry 14:10, pages 3275-3284.
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Daniel Edmund Bryan Swinson & Kenneth John O'Byrne. (2006) Interactions Between Hypoxia and Epidermal Growth Factor Receptor in Non–Small-Cell Lung Cancer. Clinical Lung Cancer 7:4, pages 250-256.
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Sally-Ann Poulsen, Laurent F. Bornaghi & Peter C. Healy. (2005) Synthesis and structure–activity relationships of novel benzene sulfonamides with potent binding affinity for bovine carbonic anhydrase II. Bioorganic & Medicinal Chemistry Letters 15:24, pages 5429-5433.
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Özen Özensoy, Luca Puccetti, Giuseppe Fasolis, Oktay Arslan, Andrea Scozzafava & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors: Inhibition of the tumor-associated isozymes IX and XII with a library of aromatic and heteroaromatic sulfonamides. Bioorganic & Medicinal Chemistry Letters 15:21, pages 4862-4866.
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Alessio Innocenti, Raquel Villar, Victor Martinez-Merino, María J. Gil, Andrea Scozzafava, Daniela Vullo & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors: Inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with benzo[b]thiophene 1,1-dioxide sulfonamides. Bioorganic & Medicinal Chemistry Letters 15:21, pages 4872-4876.
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Jan-Hendrik Beumer, Michel J. X. Hillebrand, Dick Pluim, Hilde Rosing, Karen Foley, S. Murray Yule, Jan H. M. Schellens & Jos H. Beijnen. (2005) Human metabolism of [14C]indisulam following i.v. infusion in cancer patients. Investigational New Drugs 23:4, pages 317-330.
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Vladimir Garaj, Luca Puccetti, Giuseppe Fasolis, Jean-Yves Winum, Jean-Louis Montero, Andrea Scozzafava, Daniela Vullo, Alessio Innocenti & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors: Novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II and IX. Bioorganic & Medicinal Chemistry Letters 15:12, pages 3102-3108.
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Luca Puccetti, Giuseppe Fasolis, Daniela Vullo, Zahid H. Chohan, Andrea Scozzafava & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors. Inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with Schiff’s bases incorporating chromone and aromatic sulfonamide moieties, and their zinc complexes. Bioorganic & Medicinal Chemistry Letters 15:12, pages 3096-3101.
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Gabriela Laura Almajan, Alessio Innocenti, Luca Puccetti, Gheorghe Manole, Stefania Barbuceanu, Ioana Saramet, Andrea Scozzafava & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors. Inhibition of the cytosolic and tumor-associated carbonic anhydrase isozymes I, II, and IX with a series of 1,3,4-thiadiazole- and 1,2,4-triazole-thiols. Bioorganic & Medicinal Chemistry Letters 15:9, pages 2347-2352.
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Luca Puccetti, Giuseppe Fasolis, Alessandro Cecchi, Jean-Yves Winum, Alessandro Gamberi, Jean-Louis Montero, Andrea Scozzafava & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating thioureido-sulfanilyl scaffolds. Bioorganic & Medicinal Chemistry Letters 15:9, pages 2359-2364.
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Anna Di Fiore, Giuseppina De Simone, Valeria Menchise, Carlo Pedone, Angela Casini, Andrea Scozzafava & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II. Bioorganic & Medicinal Chemistry Letters 15:7, pages 1937-1942.
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Jean-Yves WinumJean-Michel DognéAngela CasiniXavier de LevalJean-Louis MonteroAndrea ScozzafavaDaniela VulloAlessio InnocentiClaudiu T. Supuran. (2004) Carbonic Anhydrase Inhibitors: Synthesis and Inhibition of Cytosolic/Membrane-Associated Carbonic Anhydrase Isozymes I, II, and IX with Sulfonamides Incorporating Hydrazino Moieties. Journal of Medicinal Chemistry 48:6, pages 2121-2125.
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Pedro A. Colinas & Rodolfo D. Bravo. (2005) Sulfonamidoglycosylation of methyl ribofuranosides: a novel approach to furanosylsulfonamides. Tetrahedron Letters 46:10, pages 1687-1689.
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Jean‐Yves Winum, Andrea Scozzafava, Jean‐Louis Montero & Claudiu T. Supuran. (2004) Sulfamates and their therapeutic potential. Medicinal Research Reviews 25:2, pages 186-228.
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Daniela Vullo, Alessio Innocenti, Isao Nishimori, Jaromı́r Pastorek, Andrea Scozzafava, Silvia Pastoreková & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors. Inhibition of the transmembrane isozyme XII with sulfonamides—a new target for the design of antitumor and antiglaucoma drugs?. Bioorganic & Medicinal Chemistry Letters 15:4, pages 963-969.
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Hasan Turkmen, Mustafa Durgun, Serpil Yilmaztekin, Mahmut Emul, Alessio Innocenti, Daniela Vullo, Andrea Scozzafava & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors. Novel sulfanilamide/acetazolamide derivatives obtained by the tail approach and their interaction with the cytosolic isozymes I and II, and the tumor-associated isozyme IX. Bioorganic & Medicinal Chemistry Letters 15:2, pages 367-372.
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Jerapan Krungkrai, Andrea Scozzafava, Sutarnthip Reungprapavut, Sudaratana R. Krungkrai, Roonglawan Rattanajak, Sumalee Kamchonwongpaisan & Claudiu T. Supuran. (2005) Carbonic anhydrase inhibitors. Inhibition of Plasmodium falciparum carbonic anhydrase with aromatic sulfonamides: towards antimalarials with a novel mechanism of action?. Bioorganic & Medicinal Chemistry 13:2, pages 483-489.
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Peter M. Fischer, David M. Glover & David P. Lane. (2004) Targeting the cell cycle. Drug Discovery Today: Therapeutic Strategies 1:4, pages 417-423.
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Sabrina Zimmerman, Alessio Innocenti, Angela Casini, James G. Ferry, Andrea Scozzafava & Claudiu T. Supuran. (2004) Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides. Bioorganic & Medicinal Chemistry Letters 14:24, pages 6001-6006.
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Alessandro Cecchi, Jean-Yves Winum, Alessio Innocenti, Daniela Vullo, Jean-Louis Montero, Andrea Scozzafava & Claudiu T. Supuran. (2004) Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides derived from 4-isothiocyanato-benzolamide. Bioorganic & Medicinal Chemistry Letters 14:23, pages 5775-5780.
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Vladimir Garaj, Luca Puccetti, Giuseppe Fasolis, Jean-Yves Winum, Jean-Louis Montero, Andrea Scozzafava, Daniela Vullo, Alessio Innocenti & Claudiu T. Supuran. (2004) Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties. Bioorganic & Medicinal Chemistry Letters 14:21, pages 5427-5433.
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Alessio Innocenti, Jochen Antel, Michael Wurl, Andrea Scozzafava & Claudiu T. Supuran. (2004) Carbonic anhydrase inhibitors: inhibition of human cytosolic isozyme II and mitochondrial isozyme V with a series of benzene sulfonamide derivatives. Bioorganic & Medicinal Chemistry Letters 14:22, pages 5703-5707.
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C R Ireson, S K Chander, A Purohit, D C Parish, L W L Woo, B V L Potter & M J Reed. (2004) Pharmacokinetics of the nonsteroidal steroid sulphatase inhibitor 667 COUMATE and its sequestration into red blood cells in rats. British Journal of Cancer 91:7, pages 1399-1404.
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Alessio Innocenti, Angela Casini, Maria C. Alcaro, Anna M. Papini, Andrea Scozzafava & Claudiu T. Supuran. (2004) Carbonic Anhydrase Inhibitors: The First On-Resin Screening of a 4-Sulfamoylphenylthiourea Library. Journal of Medicinal Chemistry 47:21, pages 5224-5229.
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Abir L. Banerjee, Michael Swanson, Sanku Mallik & D.K. Srivastava. (2004) Purification of recombinant human carbonic anhydrase-II by metal affinity chromatography without incorporating histidine tags. Protein Expression and Purification 37:2, pages 450-454.
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Abir L. Banerjee, Michael Swanson, Bidhan C. Roy, Xiao Jia, Manas K. Haldar, Sanku Mallik & D. K. Srivastava. (2004) Protein Surface-Assisted Enhancement in the Binding Affinity of an Inhibitor for Recombinant Human Carbonic Anhydrase-II. Journal of the American Chemical Society 126:35, pages 10875-10883.
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Mona Jaiswal, Padmakar V. Khadikar, Andrea Scozzafava & Claudiu T. Supuran. (2004) Carbonic anhydrase inhibitors: the first QSAR study on inhibition of tumor-associated isoenzyme IX with aromatic and heterocyclic sulfonamides. Bioorganic & Medicinal Chemistry Letters 14:12, pages 3283-3290.
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Mark Gray & J. Jonathan Harburn. 2004. Encyclopedia of Supramolecular Chemistry. Encyclopedia of Supramolecular Chemistry
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Daniela Vullo, Andrea Scozzafava, Silvia Pastorekova, Jaromir Pastorek & Claudiu T Supuran. (2004) Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with fluorine-containing sulfonamides. The first subnanomolar CA IX inhibitor discovered. Bioorganic & Medicinal Chemistry Letters 14:9, pages 2351-2356.
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Joseph. R. Casey, Patricio E. Morgan, Daniela Vullo, Andrea Scozzafava, Antonio Mastrolorenzo & Claudiu T. Supuran. (2004) Carbonic Anhydrase Inhibitors. Design of Selective, Membrane-Impermeant Inhibitors Targeting the Human Tumor-Associated Isozyme IX. Journal of Medicinal Chemistry 47:9, pages 2337-2347.
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Silvia Pastorekova, Angela Casini, Andrea Scozzafava, Daniela Vullo, Jaromir Pastorek & Claudiu T. Supuran. (2004) Carbonic anhydrase inhibitors: The first selective, membrane-impermeant inhibitors targeting the tumor-associated isozyme IX. Bioorganic & Medicinal Chemistry Letters 14:4, pages 869-873.
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Francesco Abbate, Anita Coetzee, Angela Casini, Samuele Ciattini, Andrea Scozzafava & Claudiu T. Supuran. (2004) Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with the antipsychotic drug sulpiride. Bioorganic & Medicinal Chemistry Letters 14:2, pages 337-341.
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Francesco Abbate, Jean-Yves Winum, Barry V.L. Potter, Angela Casini, Jean-Louis Montero, Andrea Scozzafava & Claudiu T. Supuran. (2004) Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with EMATE, a dual inhibitor of carbonic anhydrases and steroid sulfatase. Bioorganic & Medicinal Chemistry Letters 14:1, pages 231-234.
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Francesco Abbate, Angela Casini, Takashi Owa, Andrea Scozzafava & Claudiu T. Supuran. (2004) Carbonic anhydrase inhibitors: E7070, a sulfonamide anticancer agent, potently inhibits cytosolic isozymes I and II, and transmembrane, tumor-associated isozyme IX. Bioorganic & Medicinal Chemistry Letters 14:1, pages 217-223.
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Ahmed Kamal, P Ramulu, O Srinivas & G Ramesh. (2003) Synthesis of C-8 methanesulphonate substituted pyrrolobenzodiazepines as potential antitumour agents. Bioorganic & Medicinal Chemistry Letters 13:20, pages 3517-3519.
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Y.T. Ho, A. Purohit, N. Vicker, S.P. Newman, J.J. Robinson, M.P. Leese, D. Ganeshapillai, L.W.L. Woo, B.V.L. Potter & M.J. Reed. (2003) Inhibition of carbonic anhydrase II by steroidal and non-steroidal sulphamates. Biochemical and Biophysical Research Communications 305:4, pages 909-914.
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