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The therapeutic potential of CRF1 antagonists for anxiety

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Pages 799-828 | Published online: 24 Feb 2005

Keep up to date with the latest research on this topic with citation updates for this article.

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Mishra Shashank Shekhar, T. Venkatachalam, Chandra Shekhar Sharma, Hemendra Pratap Singh, Sourav Kalra & Neeraj Kumar. (2019) Computational investigation of binding mechanism of substituted pyrazinones targeting corticotropin releasing factor-1 receptor deliberated for anti-depressant drug design. Journal of Biomolecular Structure and Dynamics 37:12, pages 3226-3244.
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Neeraj Kumar, Shashank Shekhar Mishra, Chandra Shekhar Sharma, Hamendra Pratap Singh & Sourav Kalra. (2018) In silico binding mechanism prediction of benzimidazole based corticotropin releasing factor-1 receptor antagonists by quantitative structure activity relationship, molecular docking and pharmacokinetic parameters calculation. Journal of Biomolecular Structure and Dynamics 36:7, pages 1691-1712.
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Rowan A. Stringer, Eckhard Weber, Andrew Culshaw, Jeff McKenna, Gareth Williams, Jonathan Rose & Bindi Sohal. (2014) Preclinical metabolism and pharmacokinetics of NVS-CRF38, a potent and orally bioavailable corticotropin-releasing factor receptor 1 antagonist. Xenobiotica 44:10, pages 902-912.
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Marcelo Paez-Pereda, Felix Hausch & Florian Holsboer. (2011) Corticotropin releasing factor receptor antagonists for major depressive disorder. Expert Opinion on Investigational Drugs 20:4, pages 519-535.
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Susan K Wood & James H Woods. (2007) Corticotropin-releasing factor receptor-1: a therapeutic target for cardiac autonomic disturbances. Expert Opinion on Therapeutic Targets 11:11, pages 1401-1413.
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Dimitri E Grigoriadis. (2005) The corticotropin-releasing factor receptor: a novel target for the treatment of depression and anxiety-related disorders. Expert Opinion on Therapeutic Targets 9:4, pages 651-684.
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Raye Z Litten, Joanne Fertig, Margaret Mattson & Mark Egli. (2005) Development of medications for alcohol use disorders: recent advances and ongoing challenges. Expert Opinion on Emerging Drugs 10:2, pages 323-343.
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