1,039
Views
196
CrossRef citations to date
0
Altmetric
Reviews

A potential therapeutic role for P2X7 receptor (P2X7R) antagonists in the treatment of inflammatory diseases

, MRCP, &
Pages 897-915 | Published online: 21 Apr 2011

Keep up to date with the latest research on this topic with citation updates for this article.

Read on this site (7)

Malek Zarei, Navideh Sahebi Vaighan & Seyed Ali Ziai. (2021) Purinergic receptor ligands: the cytokine storm attenuators, potential therapeutic agents for the treatment of COVID-19. Immunopharmacology and Immunotoxicology 43:6, pages 633-643.
Read now
Seyed Ahmad Rasoulinejad, Ahmad Karkhah, Alireza Paniri, Kiarash Saleki, Marzieh Pirzadeh & Hamid Reza Nouri. (2020) Contribution of inflammasome complex in inflammatory-related eye disorders and its implications for anti-inflammasome therapy. Immunopharmacology and Immunotoxicology 42:5, pages 400-407.
Read now
You Sheng Chong, Chun Wai Mai, Chee Onn Leong & Lai Chun Wong. (2018) Lutein improves cell viability and reduces Alu RNA accumulation in hydrogen peroxide challenged retinal pigment epithelial cells. Cutaneous and Ocular Toxicology 37:1, pages 52-60.
Read now
Ema Ozaki, Matthew Campbell & Sarah L Doyle. (2015) Targeting the NLRP3 inflammasome in chronic inflammatory diseases: current perspectives. Journal of Inflammation Research 8, pages 15-27.
Read now
Christopher NJ Young, Anthony Sinadinos, Alexis Lefebvre, Philippe Chan, Stephen Arkle, David Vaudry & Dariusz C Gorecki. (2015) A novel mechanism of autophagic cell death in dystrophic muscle regulated by P2RX7 receptor large-pore formation and HSP90. Autophagy 11:1, pages 113-130.
Read now
Ceren Sahin & Feyza Aricioglu. (2013) Future Directions of Cytokine Hypothesis in Depression: ‘NLRP3 inflamazomu’. Klinik Psikofarmakoloji Bülteni-Bulletin of Clinical Psychopharmacology 23:3, pages 280-288.
Read now
Gloria López-Castejón & Pablo Pelegrín. (2012) Current status of inflammasome blockers as anti-inflammatory drugs. Expert Opinion on Investigational Drugs 21:7, pages 995-1007.
Read now

Articles from other publishers (189)

Juan-min Li, Hai-shan Deng, Yun-da Yao, Wei-ting Wang, Jia-qin Hu, Yan Dong, Pei-xun Wang, Liang Liu, Zhong-qiu Liu, Ying Xie, Lin-lin Lu & Hua Zhou. (2023) Sinomenine ameliorates collagen-induced arthritis in mice by targeting GBP5 and regulating the P2X7 receptor to suppress NLRP3-related signaling pathways. Acta Pharmacologica Sinica 44:12, pages 2504-2524.
Crossref
Cecilia Napodano, Valeria Carnazzo, Valerio Basile, Krizia Pocino, Annunziata Stefanile, Stefania Gallucci, Patrizia Natali, Umberto Basile & Mariapaola Marino. (2023) NLRP3 Inflammasome Involvement in Heart, Liver, and Lung Diseases—A Lesson from Cytokine Storm Syndrome. International Journal of Molecular Sciences 24:23, pages 16556.
Crossref
Yanling Ai, Hengyi Wang, Lu Liu, Yulin Qi, Shiyun Tang, Jianyuan Tang & Nianzhi Chen. (2023) Purine and purinergic receptors in health and disease. MedComm 4:5.
Crossref
Yunyun Zou, Aziz Ghaderpour, Bolormaa Munkhbileg, Sang-Uk Seo & Seung-Yong Seong. (2023) Taurodeoxycholate ameliorates DSS-induced colitis in mice. International Immunopharmacology 122, pages 110628.
Crossref
Francesco Di Virgilio, Valentina Vultaggio-Poma, Simonetta Falzoni & Anna Lisa Giuliani. (2023) The Coming of Age of the P2X7 Receptor in Diagnostic Medicine. International Journal of Molecular Sciences 24:11, pages 9465.
Crossref
Fabio Grassi & Rebecca Marino. (2023) The P2X7 receptor in mucosal adaptive immunity. Purinergic Signalling.
Crossref
Deidiane Elisa Ribeiro, Lyvia Lintzmaier Petiz, Talita Glaser, Ágatha Oliveira-Giacomelli, Roberta Andrejew, Fernando de Azevedo Ribeiro Saab, Milena da Silva Milanis, Henrique Correia Campos, Vanessa Fernandes Arnaud Sampaio, Sophia La Banca, Beatriz Monteiro Longo, Claudiana Lameu, Yong Tang, Rodrigo Ribeiro Resende, Sergio T. Ferreira & Henning Ulrich. (2023) Purinergic signaling in cognitive impairment and neuropsychiatric symptoms of Alzheimer's disease. Neuropharmacology 226, pages 109371.
Crossref
Cristina Eusébio Mendes, Kelly Palombit, Thaira Thalita Alves Pereira, Henrique Inhauser Riceti Magalhães, Marcos Antônio Ferreira Caetano & Patricia Castelucci. (2023) Effects of probenecid and brilliant blue G on rat enteric glial cells following intestinal ischemia and reperfusion. Acta Histochemica 125:1, pages 151985.
Crossref
Waldemar Schäfer, Tobias Stähler, Carolina Pinto Espinoza, Welbeck Danquah, Jan Hendrik Knop, Björn Rissiek, Friedrich Haag & Friedrich Koch-Nolte. (2022) Origin, distribution, and function of three frequent coding polymorphisms in the gene for the human P2X7 ion channel. Frontiers in Pharmacology 13.
Crossref
Omaima A. Ahmedy, Dalia M. El-Tanbouly, Asmaa K. Al-Mokaddem & Yasmin A.M. El-Said. (2022) Insights into the role of P2X7R/DUSP6/ERK1/2 and SIRT2/MDM2 signaling in the nephroprotective effect of berberine against cisplatin-induced renal fibrosis in rats. Life Sciences 309, pages 121040.
Crossref
Daria Andreeva, Lada Murashova, Nikita Burzak & Vyacheslav Dyachuk. (2022) Satellite Glial Cells: Morphology, functional heterogeneity, and role in pain. Frontiers in Cellular Neuroscience 16.
Crossref
Peng Yan, Ben Ke & Xiangdong Fang. (2022) Ion channels as a therapeutic target for renal fibrosis. Frontiers in Physiology 13.
Crossref
Lidia de Tapia, Belén García-Fojeda, Nina Kronqvist, Jan Johansson & Cristina Casals. (2022) The collectin SP-A and its trimeric recombinant fragment protect alveolar epithelial cells from the cytotoxic and proinflammatory effects of human cathelicidin in vitro. Frontiers in Immunology 13.
Crossref
Valentina Vultaggio-Poma & Francesco Di Virgilio. (2022) P2 Receptors: Novel Disease Markers and Metabolic Checkpoints in Immune Cells. Biomolecules 12:7, pages 983.
Crossref
Federica Gasparri, Debayan Sarkar, Sarune Bielickaite, Mette Homann Poulsen, Alexander Sebastian Hauser & Stephan Alexander Pless. (2022) P2X2 receptor subunit interfaces are missense variant hotspots, where mutations tend to increase apparent ATP affinity. British Journal of Pharmacology 179:14, pages 3859-3874.
Crossref
Julie Sarrand, Laurie Baglione, Dorian Parisis & Muhammad Soyfoo. (2022) The Involvement of Alarmins in the Pathogenesis of Sjögren’s Syndrome. International Journal of Molecular Sciences 23:10, pages 5671.
Crossref
Valentina Vultaggio-Poma, Simonetta Falzoni, Giada Salvi, Anna Lisa Giuliani & Francesco Di Virgilio. (2022) Signalling by extracellular nucleotides in health and disease. Biochimica et Biophysica Acta (BBA) - Molecular Cell Research 1869:5, pages 119237.
Crossref
Ying Deng, Mengting Zhou, Xingtao Zhao, Xinyan Xue, Li Liao, Jing Wang & Yunxia Li. (2022) Immune Response Studies Based on P2X7 Receptors: A Mini-Review. Current Pharmaceutical Design 28:12, pages 993-999.
Crossref
Hongjuan Guo, Lili Wang, Wei Zhu, Xiaofei Qi, Qi Zhang, Yang Jiao & Jianping Cao. (2022) Respiratory flora: The potential biomarker of radiation-induced pulmonary injury. Radiation Medicine and Protection 3:1, pages 43-46.
Crossref
Weiye Li. 2022. Age-Related Macular Degeneration. Age-Related Macular Degeneration 129 163 .
Mariá Munhoz Evangelinellis, Roberta Figueiroa Souza, Cristina Eusébio Mendes & Patricia Castelucci. (2021) Effects of a P2X7 receptor antagonist on myenteric neurons in the distal colon of an experimental rat model of ulcerative colitis. Histochemistry and Cell Biology 157:1, pages 65-81.
Crossref
Komal Thapa, Nitin Verma, Thakur Gurjeet Singh, Amarjot Kaur Grewal, Neha Kanojia & Lata Rani. (2021) COVID-19-Associated acute respiratory distress syndrome (CARDS): Mechanistic insights on therapeutic intervention and emerging trends. International Immunopharmacology 101, pages 108328.
Crossref
Avik Shome, Odunayo O. Mugisho, Rachael L. Niederer & Ilva D. Rupenthal. (2021) Blocking the inflammasome: A novel approach to treat uveitis. Drug Discovery Today 26:12, pages 2839-2857.
Crossref
J.C.C. Arruda, N.C. Rocha, E.G. Santos, L.G.B. Ferreira, M.L. Bello, C. Penido, T.E.M.M. Costa, J.A.A. Santos, I.M. Ribeiro, T.C.B. Tomassini & R.X. Faria. (2021) Physalin pool from Physalis angulata L. leaves and physalin D inhibit P2X7 receptor function in vitro and acute lung injury in vivo. Biomedicine & Pharmacotherapy 142, pages 112006.
Crossref
Robert J. Unwin. (2021) Purinergic signalling in the kidney – A beginning with Geoffrey Burnstock. Autonomic Neuroscience 234, pages 102833.
Crossref
Maria Luiza Mukai Franciosi, Millena Daher Medeiros Lima, Maria Rosa Chitolina Schetinger & Andréia Machado Cardoso. (2021) Possible role of purinergic signaling in COVID-19. Molecular and Cellular Biochemistry 476:8, pages 2891-2898.
Crossref
Gholamreza Bahari, Farhad Tabasi, Mohammad Hashemi, Zahra Zakeri & Mohsen Taheri. (2021) Association of P2X7 receptor genetic polymorphisms and expression with rheumatoid arthritis susceptibility in a sample of the Iranian population: a case-control study. Clinical Rheumatology 40:8, pages 3115-3126.
Crossref
Stefania Merighi, Tino Emanuele Poloni, Anna Terrazzan, Eva Moretti, Stefania Gessi & Davide Ferrari. (2021) Alzheimer and Purinergic Signaling: Just a Matter of Inflammation?. Cells 10:5, pages 1267.
Crossref
Jing Wang, Naoki Takemura & Tatsuya Saitoh. (2021) Macrophage Response Driven by Extracellular ATP. Biological and Pharmaceutical Bulletin 44:5, pages 599-604.
Crossref
Francesco Di Virgilio, Valentina Vultaggio-Poma & Alba Clara Sarti. (2021) P2X receptors in cancer growth and progression. Biochemical Pharmacology 187, pages 114350.
Crossref
Junteng Zhou, Zhichao Zhou, Xiaojing Liu, Hai-Yan Yin, Yong Tang & Xin Cao. (2021) P2X7 Receptor–Mediated Inflammation in Cardiovascular Disease. Frontiers in Pharmacology 12.
Crossref
Patrizia Marchese, Maria Lombardi, Maria Elena Mantione, Domenico Baccellieri, David Ferrara, Roberto Chiesa, Ottavio Alfieri & Chiara Foglieni. (2021) Confocal Blood Flow Videomicroscopy of Thrombus Formation over Human Arteries and Local Targeting of P2X7. International Journal of Molecular Sciences 22:8, pages 4066.
Crossref
Zihao Li, Ziyu Huang & Lunhao Bai. (2021) The P2X7 Receptor in Osteoarthritis. Frontiers in Cell and Developmental Biology 9.
Crossref
Marco Manfredini, Anna Lisa Giuliani, Giulia Ruina, Roberta Gafà, Cristina Bosi, Elisabetta Zoppas, Francesco Di Virgilio & Vincenzo Bettoli. (2021) The P2X7 Receptor Is Overexpressed in the Lesional Skin of Subjects Affected by Hidradenitis Suppurativa: A Preliminary Study. Dermatology 237:1, pages 111-118.
Crossref
Claudia Giuseppina Fresta, Giuseppe Caruso, Annamaria Fidilio, Chiara Bianca Maria Platania, Nicolò Musso, Filippo Caraci, Filippo Drago & Claudio Bucolo. (2020) Dihydrotanshinone, a Natural Diterpenoid, Preserves Blood-Retinal Barrier Integrity via P2X7 Receptor. International Journal of Molecular Sciences 21:23, pages 9305.
Crossref
Mirco Govoni, Michele Bassi, Stefano Vezzoli, Germano Lucci, Aida Emirova, Marie Anna Nandeuil, Stefano Petruzzelli, Gera L. Jellema, Ebenezer K. Afolabi, Brendan Colgan, Brian Leaker, Oliver Kornmann, Kai Michael Beeh, Henrik Watz & Dave Singh. (2020) Sputum and blood transcriptomics characterisation of the inhaled PDE4 inhibitor CHF6001 on top of triple therapy in patients with chronic bronchitis. Respiratory Research 21:1.
Crossref
Francesco Di Virgilio, Yong Tang, Alba Clara Sarti & Marco Rossato. (2020) A rationale for targeting the P2X7 receptor in Coronavirus disease 19. British Journal of Pharmacology 177:21, pages 4990-4994.
Crossref
Mélanie Demeules, Allan Scarpitta, Catalina Abad, Henri Gondé, Romain Hardet, Carolina Pinto-Espinoza, Anna Marei Eichhoff, Waldemar Schäfer, Friedrich Haag, Friedrich Koch-Nolte & Sahil Adriouch. (2020) Evaluation of P2X7 Receptor Function in Tumor Contexts Using rAAV Vector and Nanobodies (AAVnano). Frontiers in Oncology 10.
Crossref
Eldio G. dos Santos, Robson X. Faria, Carlos R. Rodrigues & Murilo L. Bello. (2020) Molecular dynamic simulations of full-length human purinergic receptor subtype P2X7 bonded to potent inhibitors. European Journal of Pharmaceutical Sciences 152, pages 105454.
Crossref
Xiaoling Hu, Yiming Liu, Junting Wu, Yu Liu, Wenjie Liu, Ji Chen & Fengrui Yang. (2020) Inhibition of P2X7R in the amygdala ameliorates symptoms of neuropathic pain after spared nerve injury in rats. Brain, Behavior, and Immunity 88, pages 507-514.
Crossref
Romain Lara, Elena Adinolfi, Catherine A. Harwood, Mike Philpott, Julian A. Barden, Francesco Di Virgilio & Shaun McNulty. (2020) P2X7 in Cancer: From Molecular Mechanisms to Therapeutics. Frontiers in Pharmacology 11.
Crossref
Bernat Baeza-Raja, Andrew Goodyear, Xiao Liu, Kevin Lam, Lynn Yamamoto, Yingwu Li, G. Steven Dodson, Toshi Takeuchi, Tatiana Kisseleva, David A. Brenner & Karim Dabbagh. (2020) Pharmacological inhibition of P2RX7 ameliorates liver injury by reducing inflammation and fibrosis. PLOS ONE 15:6, pages e0234038.
Crossref
Qi-Huang Zheng. (2020) Radioligands targeting purinergic P2X7 receptor. Bioorganic & Medicinal Chemistry Letters 30:12, pages 127169.
Crossref
Amanda Ferreira Neves, Felipe Hertzing Farias, Silviane Fernandes de Magalhães, Dionéia Araldi, Marco PagliusiJr.Jr., Claudia Herrera Tambeli, Cesar Renato Sartori, Celina Monteiro da Cruz Lotufo & Carlos Amílcar Parada. (2020) Peripheral Inflammatory Hyperalgesia Depends on P2X7 Receptors in Satellite Glial Cells. Frontiers in Physiology 11.
Crossref
Yutong Dong, Yueqi Chen, Lincheng Zhang, Zhansong Tian & Shiwu Dong. (2020) P2X7 receptor acts as an efficient drug target in regulating bone metabolism system. Biomedicine & Pharmacotherapy 125, pages 110010.
Crossref
Mahmoud G. Khalafalla, Lucas T. Woods, Kimberly J. Jasmer, Kevin Muñoz Forti, Jean M. Camden, Janicke L. Jensen, Kirsten H. Limesand, Hilde K. Galtung & Gary A. Weisman. (2020) P2 Receptors as Therapeutic Targets in the Salivary Gland: From Physiology to Dysfunction. Frontiers in Pharmacology 11.
Crossref
Paulina Stokłosa, Anna Borgström, Sven Kappel & Christine Peinelt. (2020) TRP Channels in Digestive Tract Cancers. International Journal of Molecular Sciences 21:5, pages 1877.
Crossref
Jean L.G. da Silva, Daniela F. Passos, Viviane M. Bernardes & Daniela B.R. Leal. (2019) ATP and adenosine: Role in the immunopathogenesis of rheumatoid arthritis. Immunology Letters 214, pages 55-64.
Crossref
Laurie Erb, Lucas T. Woods, Mahmoud G. Khalafalla & Gary A. Weisman. (2019) Purinergic signaling in Alzheimer’s disease. Brain Research Bulletin 151, pages 25-37.
Crossref
Fan Cao, Li-Qin Hu, Shu-Ran Yao, Yan Hu, De-Guang Wang, Yin-Guang Fan, Gui-Xia Pan, Sha-Sha Tao, Qin Zhang, Hai-Feng Pan & Guo-Cui Wu. (2019) P2X7 receptor: A potential therapeutic target for autoimmune diseases. Autoimmunity Reviews 18:8, pages 767-777.
Crossref
Federica Gasparri, Jesper Wengel, Thomas Grutter & Stephan A. Pless. (2019) Molecular determinants for agonist recognition and discrimination in P2X2 receptors. Journal of General Physiology 151:7, pages 898-911.
Crossref
Qing-Chun Li, Yun Liang & Zhen-Bo Su. (2019) Prophylactic treatment with MSC-derived exosomes attenuates traumatic acute lung injury in rats. American Journal of Physiology-Lung Cellular and Molecular Physiology 316:6, pages L1107-L1117.
Crossref
Camila Guerra Martinez. (2019) P2X7 receptor in cardiovascular disease: The heart side. Clinical and Experimental Pharmacology and Physiology 46:6, pages 513-526.
Crossref
Kristy E. Gilman, Jean M. Camden, Rob R. Klein, Qionghui Zhang, Gary A. Weisman & Kirsten H. Limesand. (2019) P2X7 receptor deletion suppresses γ-radiation-induced hyposalivation. American Journal of Physiology-Regulatory, Integrative and Comparative Physiology 316:5, pages R687-R696.
Crossref
Lara Vargas Becker, Daniela Ferreira Passos, Daniela Bitencourt Rosa Leal, Vera Maria Morsch & Maria Rosa Chitolina Schetinger. (2019) ATP signaling and NTPDase in Systemic Lupus Erythematosus (SLE). Immunobiology 224:3, pages 419-426.
Crossref
Daniel T. G. Gonzaga, Felipe H. Oliveira, N. L. von Ranke, G. Q. Pinho, Juliana P. Salles, Murilo L. Bello, Carlos R. Rodrigues, Helena C. Castro, Hellen V. C. M. de Souza, Caroline R. C. Reis, Rennan P. P. Leme, João C. M. Mafra, Luiz C. S. Pinheiro, Lucas V. B. Hoelz, Nubia Boechat & Robson X. Faria. (2019) Synthesis, Biological Evaluation, and Molecular Modeling Studies of New Thiadiazole Derivatives as Potent P2X7 Receptor Inhibitors. Frontiers in Chemistry 7.
Crossref
Joel Linden, Friedrich Koch-NolteGerhard Dahl. (2019) Purine Release, Metabolism, and Signaling in the Inflammatory Response. Annual Review of Immunology 37:1, pages 325-347.
Crossref
Elena S. Haight, Thomas E. Forman, Stephanie A. Cordonnier, Michelle L. JamesVivianne L. Tawfik. (2019) Microglial Modulation as a Target for Chronic Pain: From the Bench to the Bedside and Back. Anesthesia & Analgesia 128:4, pages 737-746.
Crossref
Luping Wang, Sarah Schmidt, Petra P. Larsen, Johanna H. Meyer, William R. Roush, Eicke Latz, Frank G. Holz & Tim U. Krohne. (2019) Efficacy of novel selective NLRP3 inhibitors in human and murine retinal pigment epithelial cells. Journal of Molecular Medicine 97:4, pages 523-532.
Crossref
Yan Zhang, Yi-Shu Zhang, Xiao-Juan Li, Chao-Rong Huang, Hui-Jin Yu, Xiao-Xia Yang & Bin-Xiong Wang. (2019) Overexpression of miR-150 Inhibits the NF-κB Signal Pathway in Intervertebral Disc Degeneration through Targeting <b><i>P2X7</i></b>. Cells Tissues Organs 207:3-4, pages 165-176.
Crossref
Ben-Wen Cui, Ting Bai, Yong Yang, Yu Zhang, Min Jiang, Hong-Xu Yang, Mei Wu, Jian Liu, Chun-Ying Qiao, Zi-Ying Zhan, Yan-Ling Wu, Dong-Zhou Kang, Li-Hua Lian & Ji-Xing Nan. (2019) Thymoquinone Attenuates Acetaminophen Overdose-Induced Acute Liver Injury and Inflammation Via Regulation of JNK and AMPK Signaling Pathway. The American Journal of Chinese Medicine 47:03, pages 577-594.
Crossref
Maarten Timmers, Paulien Ravenstijn, Liwen Xi, Gallen Triana-Baltzer, Maura Furey, Sandy Van Hemelryck, Jeike Biewenga, Marc Ceusters, Anindya Bhattacharya, Maarten van den Boer, Luc van Nueten & Peter de Boer. (2018) Clinical pharmacokinetics, pharmacodynamics, safety, and tolerability of JNJ-54175446, a brain permeable P2X7 antagonist, in a randomised single-ascending dose study in healthy participants. Journal of Psychopharmacology 32:12, pages 1341-1350.
Crossref
Rai Khalid Farooq, Arnaud Tanti, Samia Ainouche, Sébastien Roger, Catherine Belzung & Vincent Camus. (2018) A P2X7 receptor antagonist reverses behavioural alterations, microglial activation and neuroendocrine dysregulation in an unpredictable chronic mild stress (UCMS) model of depression in mice. Psychoneuroendocrinology 97, pages 120-130.
Crossref
Francesco Di Virgilio, Alba Clara Sarti, Simonetta Falzoni, Elena De Marchi & Elena Adinolfi. (2018) Extracellular ATP and P2 purinergic signalling in the tumour microenvironment. Nature Reviews Cancer 18:10, pages 601-618.
Crossref
Anja Pfalzgraff, Sergio Bárcena-Varela, Lena Heinbockel, Thomas Gutsmann, Klaus Brandenburg, Guillermo Martinez-de-Tejada & Günther Weindl. (2018) Antimicrobial endotoxin-neutralizing peptides promote keratinocyte migration via P2X7 receptor activation and accelerate wound healing in vivo . British Journal of Pharmacology 175:17, pages 3581-3593.
Crossref
Michael Mousseau, Nicole E. Burma, Kwan Yeop LeeHeather Leduc-Pessah, Charlie H. T. KwokAllison R. ReidMelissa O’Brien, Boriss Sagalajev, Jo Anne StrattonNatalya PatrickPatrick L. StemkowskiJeff Biernaskie, Gerald W. ZamponiPaul SaloJason J. McDougall, Steven A. Prescott, John R. Matyas & Tuan Trang. (2018) Microglial pannexin-1 channel activation is a spinal determinant of joint pain. Science Advances 4:8.
Crossref
Shao-jun Li, Yu-fen Zhang, Se-hui Ma, Yao Yi, Hong-yan Yu, Lei Pei & Dan Feng. (2018) The role of NLRP3 inflammasome in stroke and central poststroke pain. Medicine 97:33, pages e11861.
Crossref
Marco Tozzi, Anna T. Larsen, Sofie C. Lange, Andrea Giannuzzo, Martin N. Andersen & Ivana Novak. (2018) The P2X7 receptor and pannexin-1 are involved in glucose-induced autocrine regulation in β-cells. Scientific Reports 8:1.
Crossref
Oleg Kambur, Mari A. Kaunisto, Bendik S. Winsvold, Tom Wilsgaard, Audun Stubhaug, John A. Zwart, Eija Kalso & Christopher S. Nielsen. (2018) Genetic variation in P2RX7 and pain tolerance. Pain 159:6, pages 1064-1073.
Crossref
Francesco Di Virgilio, Alba Clara Sarti & Fabio Grassi. (2018) Modulation of innate and adaptive immunity by P2X ion channels. Current Opinion in Immunology 52, pages 51-59.
Crossref
Ivana Novak & Anna Solini. (2018) P2X receptor-ion channels in the inflammatory response in adipose tissue and pancreas — potential triggers in onset of type 2 diabetes?. Current Opinion in Immunology 52, pages 1-7.
Crossref
Danlu Jiang, Sheng Chen, Ruyu Sun, Xue Zhang & Di Wang. (2018) The NLRP3 inflammasome: Role in metabolic disorders and regulation by metabolic pathways. Cancer Letters 419, pages 8-19.
Crossref
Diego Dal Ben, Luca Antonioli, Catia Lambertucci, Matteo Fornai, Corrado Blandizzi & Rosaria Volpini. (2018) Purinergic Ligands as Potential Therapeutic Tools for the Treatment of Inflammation-Related Intestinal Diseases. Frontiers in Pharmacology 9.
Crossref
Jingnian Song, Yanlu Ying, Wei Wang, Xianguo Liu, Xuebing Xu, Xuhong Wei & Xiangcai Ruan. (2018) The role of P2X7R/ERK signaling in dorsal root ganglia satellite glial cells in the development of chronic postsurgical pain induced by skin/muscle incision and retraction (SMIR). Brain, Behavior, and Immunity 69, pages 180-189.
Crossref
Luiz E. B. Savio, Paola de Andrade Mello, Cleide Gonçalves da Silva & Robson Coutinho-Silva. (2018) The P2X7 Receptor in Inflammatory Diseases: Angel or Demon?. Frontiers in Pharmacology 9.
Crossref
Saleela M. Ruwanpura, Sarah Rosli & Michelle D. Tate. 2018. Inflammasomes: Clinical and Therapeutic Implications. Inflammasomes: Clinical and Therapeutic Implications 61 84 .
Michael Kasper & Kathrin Barth. (2017) Potential contribution of alveolar epithelial type I cells to pulmonary fibrosis. Bioscience Reports 37:6.
Crossref
Joaquín Amores-Iniesta, Maria Barberà-Cremades, Carlos M. Martínez, José A. Pons, Beatriz Revilla-Nuin, Laura Martínez-Alarcón, Francesco Di Virgilio, Pascual Parrilla, Alberto Baroja-Mazo & Pablo Pelegrín. (2017) Extracellular ATP Activates the NLRP3 Inflammasome and Is an Early Danger Signal of Skin Allograft Rejection. Cell Reports 21:12, pages 3414-3426.
Crossref
Shradha Mawatwal, Assirbad Behura, Abhirupa Ghosh, Saqib Kidwai, Abtar Mishra, Amar Deep, Sakshi Agarwal, Sudipto Saha, Ramandeep Singh & Rohan Dhiman. (2017) Calcimycin mediates mycobacterial killing by inducing intracellular calcium-regulated autophagy in a P2RX7 dependent manner. Biochimica et Biophysica Acta (BBA) - General Subjects 1861:12, pages 3190-3200.
Crossref
Altaf Mohammed, Naveena B. Janakiram, Venkateshwar Madka, Gopal Pathuri, Qian Li, Rebekah Ritchie, Laura Biddick, Hannah Kutche, Yuting Zhang, Anil Singh, Hariprasad Gali, Stan Lightfoot, Vernon E. Steele, Chen S. Suen & Chinthalapally V. Rao. (2017) Lack of chemopreventive effects of P2X7R inhibitors against pancreatic cancer. Oncotarget 8:58, pages 97822-97834.
Crossref
Mahmoud G. Khalafalla, Lucas T. Woods, Jean M. Camden, Aslam A. Khan, Kirsten H. Limesand, Michael J. Petris, Laurie Erb & Gary A. Weisman. (2017) P2X7 receptor antagonism prevents IL-1β release from salivary epithelial cells and reduces inflammation in a mouse model of autoimmune exocrinopathy. Journal of Biological Chemistry 292:40, pages 16626-16637.
Crossref
Daniel Tadeu Gomes Gonzaga, Leonardo Braga Gomes Ferreira, Thadeu Estevam Moreira Maramaldo Costa, Natalia Lidmar von Ranke, Paulo Anastácio Furtado Pacheco, Ana Paula Sposito Simões, Juliana Carvalho Arruda, Luiza Pereira Dantas, Hércules Rezende de Freitas, Ricardo Augusto de Melo Reis, Carmen Penido, Murilo Lamim Bello, Helena Carla Castro, Carlos Rangel Rodrigues, Vitor Francisco Ferreira, Robson Xavier Faria & Fernando de Carvalho da Silva. (2017) 1-Aryl-1 H - and 2-aryl-2 H -1,2,3-triazole derivatives blockade P2X7 receptor in vitro and inflammatory response in vivo. European Journal of Medicinal Chemistry 139, pages 698-717.
Crossref
Geoffrey Burnstock. (2017) Purinergic Signalling: Therapeutic Developments. Frontiers in Pharmacology 8.
Crossref
Itzhak Binderman, Nasir Gadban & Avinoam Yaffe. (2017) Extracellular ATP is a key modulator of alveolar bone loss in periodontitis. Archives of Oral Biology 81, pages 131-135.
Crossref
Young-Hwan JungYeo Ok KimJung Hyun HanYong-Chul KimMyung Ha Yoon. (2017) Isobolographic Analysis of Drug Combinations With Intrathecal BRL52537 (κ-Opioid Agonist), Pregabalin (Calcium Channel Modulator), AF 353 (P2X3 Receptor Antagonist), and A804598 (P2X7 Receptor Antagonist) in Neuropathic Rats. Anesthesia & Analgesia 125:2, pages 670-677.
Crossref
Tai Yeon Koo, Jae-Ghi Lee, Ji-Jing Yan, Joon Young Jang, Kyung Don Ju, Miyeun Han, Kook-Hwan Oh, Curie Ahn & Jaeseok Yang. (2017) The P2X7 receptor antagonist, oxidized adenosine triphosphate, ameliorates renal ischemia-reperfusion injury by expansion of regulatory T cells. Kidney International 92:2, pages 415-431.
Crossref
Binan Zhu, Yuting Lu, Leilin Chen, Binbin Yu, Yuexin Liu, Min Song & Taijun Hang. (2017) Identification and characterization of related substances in EVT-401 by hyphenated LC–MS techniques. Journal of Pharmaceutical Analysis 7:4, pages 223-230.
Crossref
Huguette Gaelle Ngassa Mbenda, Antonia Wadley, Zane Lombard, Catherine Cherry, Patricia Price & Peter Kamerman. (2017) Genetics of HIV-associated sensory neuropathy and related pain in Africans. Journal of NeuroVirology 23:4, pages 511-519.
Crossref
Maria Barberà-Cremades, Ana I. Gómez, Alberto Baroja-Mazo, Laura Martínez-Alarcón, Carlos M. Martínez, Carlos de Torre-Minguela & Pablo Pelegrín. (2017) P2X7 Receptor Induces Tumor Necrosis Factor-α Converting Enzyme Activation and Release to Boost TNF-α Production. Frontiers in Immunology 8.
Crossref
Maria Lombardi, Maria Elena Mantione, Domenico Baccellieri, David Ferrara, Renata Castellano, Roberto Chiesa, Ottavio Alfieri & Chiara Foglieni. (2017) P2X7 receptor antagonism modulates IL-1β and MMP9 in human atherosclerotic vessels. Scientific Reports 7:1.
Crossref
Francesco Di Virgilio, Diego Dal Ben, Alba Clara Sarti, Anna Lisa Giuliani & Simonetta Falzoni. (2017) The P2X7 Receptor in Infection and Inflammation. Immunity 47:1, pages 15-31.
Crossref
Frances M. Munoz, Ruby Gao, Yuzhen Tian, Brian A. Henstenburg, James E. Barrett & Huijuan Hu. (2017) Neuronal P2X7 receptor-induced reactive oxygen species production contributes to nociceptive behavior in mice. Scientific Reports 7:1.
Crossref
Yong Zhang, Yanyan Zhang, Hao Li, Xiao Jia, Xiuying Zhang, Yan Xia, YuZhong Wang, Linlin Fu, Chenghua Xiao & Deqin Geng. (2017) Increased expression of P2X7 receptor in peripheral blood mononuclear cells correlates with clinical severity and serum levels of Th17-related cytokines in patients with myasthenia gravis. Clinical Neurology and Neurosurgery 157, pages 88-94.
Crossref
Diana Sofia Marques Nascimento, Catarina Soares Potes, Miguel Luz Soares, António Carlos Ferreira, Marzia Malcangio, José Manuel Castro-Lopes & Fani Lourença Moreira Neto. (2017) Drug-Induced HSP90 Inhibition Alleviates Pain in Monoarthritic Rats and Alters the Expression of New Putative Pain Players at the DRG. Molecular Neurobiology.
Crossref
Anne-Sofie Greve, Marianne Skals, Steen K. Fagerberg, Wulf Tonnus, Svend Ellermann-Eriksen, Richard J. Evans, Andreas Linkermann & Helle A. Praetorius. (2017) P2X1, P2X4, and P2X7 Receptor Knock Out Mice Expose Differential Outcome of Sepsis Induced by α-Haemolysin Producing Escherichia coli. Frontiers in Cellular and Infection Microbiology 7.
Crossref
Thomas Gicquel, Brendan Le Daré, Elisabeth Boichot & Vincent Lagente. (2017) Purinergic receptors: new targets for the treatment of gout and fibrosis. Fundamental & Clinical Pharmacology 31:2, pages 136-146.
Crossref
Paolo Pevarello, Silvia Bovolenta, Paola Tarroni, Lorena Za, Elda Severi, Domenica Torino & Rocco Vitalone. (2017) P2X7 antagonists for CNS indications: recent patent disclosures. Pharmaceutical Patent Analyst 6:2, pages 61-76.
Crossref
Bin Zheng, Renchun Lai, Jun Li & Zhiyi Zuo. (2017) Critical role of P2X7 receptors in the neuroinflammation and cognitive dysfunction after surgery. Brain, Behavior, and Immunity 61, pages 365-374.
Crossref
Szu‐Wei Huang, Catherine Walker, Joanne Pennock, Kathryn Else, Werner Muller, Michael JD Daniels, Carolina Pellegrini, David Brough, Gloria Lopez‐Castejon & Sheena M Cruickshank. (2016) P2X7 receptor‐dependent tuning of gut epithelial responses to infection. Immunology & Cell Biology 95:2, pages 178-188.
Crossref
Sean Nelson, Hiroshi Kiyono & Yosuke Kurashima. (2016) Epithelial extracellular ATP: an initiator of immunity to parasitic infections. Immunology & Cell Biology 95:2, pages 117-118.
Crossref
Marta Barniol-Xicota, Seung-Hwa Kwak, So-Deok Lee, Emily Caseley, Elena Valverde, Lin-Hua Jiang, Yong-Chul Kim & Santiago Vázquez. (2017) Escape from adamantane: Scaffold optimization of novel P2X7 antagonists featuring complex polycycles. Bioorganic & Medicinal Chemistry Letters 27:4, pages 759-763.
Crossref
Kenneth R. Cooke, Leo Luznik, Stefanie Sarantopoulos, Frances T. Hakim, Madan Jagasia, Daniel H. Fowler, Marcel R.M. van den Brink, John A. Hansen, Robertson Parkman, David B. Miklos, Paul J. Martin, Sophie Paczesny, Georgia Vogelsang, Steven Pavletic, Jerome Ritz, Kirk R. Schultz & Bruce R. Blazar. (2017) The Biology of Chronic Graft-versus-Host Disease: A Task Force Report from the National Institutes of Health Consensus Development Project on Criteria for Clinical Trials in Chronic Graft-versus-Host Disease. Biology of Blood and Marrow Transplantation 23:2, pages 211-234.
Crossref
Francisco M. Nadal-Nicolás, Caridad Galindo-Romero, Francisco J. Valiente-Soriano, María Barberà-Cremades, Carlos deTorre-Minguela, Manuel Salinas-Navarro, Pablo Pelegrín & Marta Agudo-Barriuso. (2016) Involvement of P2X7 receptor in neuronal degeneration triggered by traumatic injury. Scientific Reports 6:1.
Crossref
Alistair G. Fryatt, Sudad Dayl, Paul M. Cullis, Ralf Schmid & Richard J. Evans. (2016) Mechanistic insights from resolving ligand-dependent kinetics of conformational changes at ATP-gated P2X1R ion channels. Scientific Reports 6:1.
Crossref
Xiaomin Zhong, Feng Zhu, Jianlin Qiao, Kai Zhao, Shengyun Zhu, Lingyu Zeng, Xiaofei Chen & Kailin Xu. (2016) The impact of P2X7 receptor antagonist, brilliant blue G on graft-versus-host disease in mice after allogeneic hematopoietic stem cell transplantation. Cellular Immunology 310, pages 71-77.
Crossref
K. Milewski & M. Oria. (2015) What we know: the inflammatory basis of hepatic encephalopathy. Metabolic Brain Disease 31:6, pages 1239-1247.
Crossref
Andrea Giannuzzo, Mara Saccomano, Joanna Napp, Maria Ellegaard, Frauke Alves & Ivana Novak. (2016) Targeting of the P2X7 receptor in pancreatic cancer and stellate cells. International Journal of Cancer 139:11, pages 2540-2552.
Crossref
Welbeck DanquahCatherine Meyer-SchwesingerBjörn RissiekCarolina PintoArnau Serracant-PratMiriam AmadiDomenica IacendaJan-Hendrik KnopAnna HammelPhiline BergmannNicole SchwarzJoana AssunçãoWendy RotthierFriedrich HaagEva TolosaPeter BannasEric Boué-GrabotTim MagnusToon LaeremansCatelijne StortelersFriedrich Koch-Nolte. (2016) Nanobodies that block gating of the P2X7 ion channel ameliorate inflammation. Science Translational Medicine 8:366.
Crossref
Giovanna Sociali, Davide Visigalli, Thomas Prukop, Ilaria Cervellini, Elena Mannino, Consuelo Venturi, Santina Bruzzone, Michael W. Sereda & Angelo Schenone. (2016) Tolerability and efficacy study of P2X7 inhibition in experimental Charcot-Marie-Tooth type 1A (CMT1A) neuropathy. Neurobiology of Disease 95, pages 145-157.
Crossref
Zhi-Dan Fan, Ya-Yuan Zhang, Yi-Hong Guo, Na Huang, Hui-Hui Ma, Hui Huang & Hai-Guo Yu. (2016) Involvement of P2X7 receptor signaling on regulating the differentiation of Th17 cells and type II collagen-induced arthritis in mice. Scientific Reports 6:1.
Crossref
Francesco Di Virgilio & Anna Lisa Giuliani. (2016) Purinergic signalling in autoimmunity: A role for the P2X7R in systemic lupus erythematosus?. Biomedical Journal 39:5, pages 326-338.
Crossref
W.M. BaldwinIIIIII & A.E. Morelli. (2016) Strategically Altering the Balance of Macrophage Subpopulations to Inhibit Chronic Rejection. American Journal of Transplantation 16:9, pages 2510-2511.
Crossref
C. Wu, Y. Zhao, X. Xiao, Y. Fan, M. Kloc, W. Liu, R.M. Ghobrial, P. Lan, X. He & X.C. Li. (2016) Graft-Infiltrating Macrophages Adopt an M2 Phenotype and Are Inhibited by Purinergic Receptor P2X7 Antagonist in Chronic Rejection. American Journal of Transplantation 16:9, pages 2563-2573.
Crossref
Priyank A. Shenoy, Andy Kuo, Irina Vetter & Maree T. Smith. (2016) The Walker 256 Breast Cancer Cell- Induced Bone Pain Model in Rats. Frontiers in Pharmacology 7.
Crossref
Francesca Amoroso, Erica Salaro, Simonetta Falzoni, Paola Chiozzi, Anna Lisa Giuliani, Giorgio Cavallesco, Pio Maniscalco, Andrea Puozzo, Ilaria Bononi, Fernanda Martini, Mauro Tognon & Francesco Di Virgilio. (2016) P2×7 targeting inhibits growth of human mesothelioma. Oncotarget 7:31, pages 49664-49676.
Crossref
Hayley Goullee, Antonia L. Wadley, Catherine L. Cherry, Richard J. N. Allcock, Michael Black, Peter R. Kamerman & Patricia Price. (2016) Polymorphisms in CAMKK2 may predict sensory neuropathy in African HIV patients. Journal of NeuroVirology 22:4, pages 508-517.
Crossref
Ronglan Zhao, Dongchun Liang & Deming Sun. (2016) Blockade of Extracellular ATP Effect by Oxidized ATP Effectively Mitigated Induced Mouse Experimental Autoimmune Uveitis (EAU). PLOS ONE 11:5, pages e0155953.
Crossref
Lucas T. Woods, Deepa Ajit, Jean M. Camden, Laurie Erb & Gary A. Weisman. (2016) Purinergic receptors as potential therapeutic targets in Alzheimer's disease. Neuropharmacology 104, pages 169-179.
Crossref
Christa C. Chrovian, Akinola Soyode-Johnson, Hong Ao, Genesis M. Bacani, Nicholas I. Carruthers, Brian Lord, Leslie Nguyen, Jason C. Rech, Qi Wang, Anindya Bhattacharya & Michael A. Letavic. (2016) Novel Phenyl-Substituted 5,6-Dihydro-[1,2,4]triazolo[4,3- a ]pyrazine P2X7 Antagonists with Robust Target Engagement in Rat Brain . ACS Chemical Neuroscience 7:4, pages 490-497.
Crossref
Lakshmi Galam, Ashna Rajan, Athena Failla, Ramani Soundararajan, Richard F. Lockey & Narasaiah Kolliputi. (2016) Deletion of P2X7 attenuates hyperoxia-induced acute lung injury via inflammasome suppression. American Journal of Physiology-Lung Cellular and Molecular Physiology 310:6, pages L572-L581.
Crossref
James Won Suk Jahng, Erfei Song & Gary Sweeney. (2016) Crosstalk between the heart and peripheral organs in heart failure. Experimental & Molecular Medicine 48:3, pages e217-e217.
Crossref
Lifang Zou, Guihua Tu, Wei Xie, Shiyao Wen, Qiuyu Xie, Shuangmei Liu, Guilin Li, Yun Gao, Hong Xu, Shouyu Wang, Yun Xue, Bing Wu, Qiulan Lv, Mofeng Ying, Xi Zhang & Shangdong Liang. (2015) LncRNA NONRATT021972 involved the pathophysiologic processes mediated by P2X7 receptors in stellate ganglia after myocardial ischemic injury. Purinergic Signalling 12:1, pages 127-137.
Crossref
Herbert Zimmermann. (2015) Extracellular ATP and other nucleotides—ubiquitous triggers of intercellular messenger release. Purinergic Signalling 12:1, pages 25-57.
Crossref
János Peti-PeterdiBellamkonda K. KishoreJennifer L. Pluznick. (2016) Regulation of Vascular and Renal Function by Metabolite Receptors. Annual Review of Physiology 78:1, pages 391-414.
Crossref
Martha Triantafilou, Timothy R. Hughes, Bryan Paul Morgan & Kathy Triantafilou. (2016) Complementing the inflammasome. Immunology 147:2, pages 152-164.
Crossref
Amma Owusu-Ansah, Chibueze A. Ihunnah, Aisha L. Walker & Solomon F. Ofori-Acquah. (2016) Inflammatory targets of therapy in sickle cell disease. Translational Research 167:1, pages 281-297.
Crossref
Flávia Sarmento Vieira, Hayandra Ferreira Nanini, Christina Maeda Takiya & Robson Coutinho-Silva. (2016) P2X7 receptor knockout prevents streptozotocin-induced type 1 diabetes in mice. Molecular and Cellular Endocrinology 419, pages 148-157.
Crossref
Xudong Jiang, Wenjuan Mao, Ziyi Yang, Jia Zeng, Yi Zhang, Yang Song, Ying Kong, Shuangyi Ren & Yunfei Zuo. (2015) Silencing P2X7 receptor downregulates the expression of TCP-1 involved in lymphoma lymphatic metastasis. Oncotarget 6:39, pages 42105-42117.
Crossref
Chang-Hong Li, Xin-Jiang Lu, Ming-Yun Li & Jiong Chen. (2015) Cathelicidin modulates the function of monocytes/macrophages via the P2X7 receptor in a teleost, Plecoglossus altivelis. Fish & Shellfish Immunology 47:2, pages 878-885.
Crossref
Daniela Gentile, Mariarita Natale, Pietro Enea Lazzerini, Pier Leopoldo Capecchi & Franco Laghi-Pasini. (2015) The role of P2X7 receptors in tissue fibrosis: a brief review. Purinergic Signalling 11:4, pages 435-440.
Crossref
Talia H. Swartz, George R. Dubyak & Benjamin K. Chen. (2015) Purinergic Receptors: Key Mediators of HIV-1 Infection and Inflammation. Frontiers in Immunology 6.
Crossref
Robert I. Menzies, Amelia R. Howarth, Robert J. Unwin, Frederick W.K. Tam, John J. Mullins & Matthew A. Bailey. (2015) Inhibition of the purinergic P2X7 receptor improves renal perfusion in angiotensin-II-infused rats. Kidney International 88:5, pages 1079-1087.
Crossref
Manju Tewari & Pankaj Seth. (2015) Emerging role of P2X7 receptors in CNS health and disease. Ageing Research Reviews 24, pages 328-342.
Crossref
Anthony Sinadinos, Christopher N. J. Young, Rasha Al-Khalidi, Anna Teti, Pawe? Kalinski, Shafini Mohamad, L?onore Floriot, Tiphaine Henry, Gianluca Tozzi, Taiwen Jiang, Olivier Wurtz, Alexis Lefebvre, Mikhail Shugay, Jie Tong, David Vaudry, Stephen Arkle, Jean-Claude doRego & Dariusz C. G?recki. (2015) P2RX7 Purinoceptor: A Therapeutic Target for Ameliorating the Symptoms of Duchenne Muscular Dystrophy. PLOS Medicine 12:10, pages e1001888.
Crossref
Jingya Yu, Yong Chen, Mingcai Li, Qiaoyan Gao, Yong Peng, Qiongyao Gong, Zhen Zhang & Xiudi Wu. (2015) Paeoniflorin down-regulates ATP-induced inflammatory cytokine production and P2X7R expression on peripheral blood mononuclear cells from patients with primary Sjögren's syndrome. International Immunopharmacology 28:1, pages 115-120.
Crossref
Amelia R. Howarth, Bryan R. Conway & Matthew A. Bailey. (2015) Vascular and inflammatory actions of P2X receptors in renal injury. Autonomic Neuroscience 191, pages 135-140.
Crossref
Yan Deng, Xue-Ling Guo, Xiao Yuan, Jin Shang, Die Zhu & Hui-Guo Liu. (2015) P2X7 Receptor Antagonism Attenuates the Intermittent Hypoxia-induced Spatial Deficits in a Murine Model of Sleep Apnea Via Inhibiting Neuroinflammation and Oxidative Stress. Chinese Medical Journal 128:16, pages 2168-2175.
Crossref
Emily A. Caseley, Stephen P. Muench, Stephen A. Baldwin, Katie Simmons, Colin W. Fishwick & Lin-Hua Jiang. (2015) Docking of competitive inhibitors to the P2X7 receptor family reveals key differences responsible for changes in response between rat and human. Bioorganic & Medicinal Chemistry Letters 25:16, pages 3164-3167.
Crossref
Leonardo Ferreira, Luíza Pereira & Robson Faria. (2015) Fluorescent dyes as a reliable tool in P2X7 receptor-associated pore studies. Journal of Bioenergetics and Biomembranes 47:4, pages 283-307.
Crossref
Alexander Eser, Jean-Frederic Colombel, Paul Rutgeerts, Severine Vermeire, Harald Vogelsang, Martin Braddock, Tore Persson & Walter Reinisch. (2015) Safety and Efficacy of an Oral Inhibitor of the Purinergic Receptor P2X7 in Adult Patients with Moderately to Severely Active Crohn?s Disease. Inflammatory Bowel Diseases, pages 1.
Crossref
Neha Soni, Prashant Koushal, B.V.K. Reddy, Rahul Deshmukh & Puneet Kumar. (2015) Effect of GLT-1 modulator and P2X7 antagonists alone and in combination in the kindling model of epilepsy in rats. Epilepsy & Behavior 48, pages 4-14.
Crossref
Tilmann Kallinich. (2015) Regulating against the dysregulation: new treatment options in autoinflammation. Seminars in Immunopathology 37:4, pages 429-437.
Crossref
Yaoping Tang, Yongchao Wang, Kyoung-mi Park, Qiuping Hu, Jian-peng Teoh, Zuzana Broskova, Punithavathi Ranganathan, Calpurnia Jayakumar, Jie Li, Huabo Su, Yaoliang Tang, Ganesan Ramesh & Il-man Kim. (2015) MicroRNA-150 protects the mouse heart from ischaemic injury by regulating cell death. Cardiovascular Research 106:3, pages 387-397.
Crossref
Ramasri Sathanoori, Karl Sw?rd, Bj?rn Olde & David Erlinge. (2015) The ATP Receptors P2X7 and P2X4 Modulate High Glucose and Palmitate-Induced Inflammatory Responses in Endothelial Cells. PLOS ONE 10:5, pages e0125111.
Crossref
Stefan FeskeHeike Wulff & Edward Y. Skolnik. (2015) Ion Channels in Innate and Adaptive Immunity. Annual Review of Immunology 33:1, pages 291-353.
Crossref
Yanli Yan, Jianwen BaiXiaoxu Zhou, Jinhua Tang, Chunming Jiang, Evelyn Tolbert, George Bayliss, Rujun Gong, Ting C. Zhao & Shougang Zhuang. (2015) P2X7 receptor inhibition protects against ischemic acute kidney injury in mice. American Journal of Physiology-Cell Physiology 308:6, pages C463-C472.
Crossref
SeungHye Han & Rama K. Mallampalli. (2015) The Acute Respiratory Distress Syndrome: From Mechanism to Translation. The Journal of Immunology 194:3, pages 855-860.
Crossref
Samantha L. Schneider, Andrew L. Ross & James M. Grichnik. (2015) Do inflammatory pathways drive melanomagenesis?. Experimental Dermatology 24:2, pages 86-90.
Crossref
Blandine Maître, Stéphanie Magnenat, Véronique Heim, Catherine Ravanat, Richard J. Evans, Henri de la Salle, Christian Gachet & Béatrice Hechler. (2015) The P2X1 Receptor Is Required for Neutrophil Extravasation during Lipopolysaccharide-Induced Lethal Endotoxemia in Mice. The Journal of Immunology 194:2, pages 739-749.
Crossref
Sae-Hae KimHa-Yan LeeYong-Suk Jang. (2015) Expression of the ATP-gated P2X 7 Receptor on M Cells and Its Modulating Role in the Mucosal Immune Environment . Immune Network 15:1, pages 44.
Crossref
Humaira Masood, Ruochen Che & Aihua Zhang. (2015) Inflammasomes in the Pathophysiology of Kidney Diseases. Kidney Diseases 1:3, pages 187-193.
Crossref
Clare M Turner, Nishkantha Arulkumaran, Mervyn Singer, Robert J Unwin & Frederick WK Tam. (2014) Is the inflammasome a potential therapeutic target in renal disease?. BMC Nephrology 15:1.
Crossref
Labchan Rajbhandari, Million Adane Tegenge, Shiva Shrestha, Nishant Ganesh Kumar, Adeel Malik, Aditya Mithal, Suneil Hosmane & Arun Venkatesan. (2014) Toll-like receptor 4 deficiency impairs microglial phagocytosis of degenerating axons. Glia 62:12, pages 1982-1991.
Crossref
Yuanyuan Zhang, Fahuan Yuan, Xuejiao Cao, Zhifang Zhai, GangHuang, Xiang Du, Yiqin Wang, Jingbo zhang, Yunjian Huang, Jinghong Zhao & Weiping Hou. (2014) P2X7 receptor blockade protects against cisplatin-induced nephrotoxicity in mice by decreasing the activities of inflammasome components, oxidative stress and caspase-3. Toxicology and Applied Pharmacology 281:1, pages 1-10.
Crossref
Luiz Anastacio Alves, Ricardo Augusto de Melo Reis, Cristina Alves Magalhães de Souza, Monica Santos de Freitas, Pedro Celso Nogueira Teixeira, Dinarte Neto Moreira Ferreira & Robson Faria Xavier. (2014) The P2X7 receptor: Shifting from a low- to a high-conductance channel — An enigmatic phenomenon?. Biochimica et Biophysica Acta (BBA) - Biomembranes 1838:10, pages 2578-2587.
Crossref
Bernd L. Fiebich, Shamima Akter & Ravi Shankar Akundi. (2014) The two-hit hypothesis for neuroinflammation: role of exogenous ATP in modulating inflammation in the brain. Frontiers in Cellular Neuroscience 8.
Crossref
Min Wan, Oliver Soehnlein, Xiao Tang, Anne M. Does, Erik Smedler, Per Uhlén, Lennart Lindbom, Birgitta Agerberth & Jesper Z. Haeggström. (2014) Cathelicidin LL‐37 induces time‐resolved release of LTB 4 and TXA 2 by human macrophages and triggers eicosanoid generation in vivo . The FASEB Journal 28:8, pages 3456-3467.
Crossref
Fernando Ochoa-Cortes, Andromeda Liñán-Rico, Kenneth A. Jacobson & Fievos L. Christofi. (2014) Potential for Developing Purinergic Drugs for Gastrointestinal Diseases. Inflammatory Bowel Diseases 20:7, pages 1259-1287.
Crossref
Guy G. Brusselle, Sharen Provoost, Ken R. Bracke, Anna Kuchmiy & Mohamed Lamkanfi. (2014) Inflammasomes in Respiratory Disease. Chest 145:5, pages 1121-1133.
Crossref
Kaifeng Liu, Andrea Vergani, Picheng Zhao, Moufida Ben Nasr, Xiao Wu, Khadija Iken, Dawei Jiang, Xiaofeng Su, Carmen Fotino, Paolo Fiorina & Gary A Visner. (2014) Inhibition of the Purinergic Pathway Prolongs Mouse Lung Allograft Survival. American Journal of Respiratory Cell and Molecular Biology, pages 140324142513008.
Crossref
Zhongshuang Hu, Taisuke Murakami, Kaori Suzuki, Hiroshi Tamura, Kyoko Kuwahara-Arai, Toshiaki Iba & Isao Nagaoka. (2014) Antimicrobial Cathelicidin Peptide LL-37 Inhibits the LPS/ATP-Induced Pyroptosis of Macrophages by Dual Mechanism. PLoS ONE 9:1, pages e85765.
Crossref
Torben Madsen Kvist, Peter Schwarz & Niklas Rye Jørgensen. (2014) The P2X7 Receptor: A Key Player in Immune-Mediated Bone Loss?. The Scientific World Journal 2014, pages 1-10.
Crossref
Suvarthi DasRatanesh Kumar SethAshutosh KumarMaria B. KadiiskaGregory Michelotti, Anna Mae Diehl & Saurabh Chatterjee. (2013) Purinergic receptor X7 is a key modulator of metabolic oxidative stress-mediated autophagy and inflammation in experimental nonalcoholic steatohepatitis. American Journal of Physiology-Gastrointestinal and Liver Physiology 305:12, pages G950-G963.
Crossref
Sheng Chen, Qingyi Ma, Paul R. Krafft, Yujie Chen, Jiping Tang, Jianmin Zhang & John H. Zhang. (2013) P2X7 Receptor Antagonism Inhibits p38 Mitogen-Activated Protein Kinase Activation and Ameliorates Neuronal Apoptosis After Subarachnoid Hemorrhage in Rats. Critical Care Medicine 41:12, pages e466-e474.
Crossref
Luiz Alves, Rômulo Bezerra, Robson Faria, Leonardo Ferreira & Valber da Silva Frutuoso. (2013) Physiological Roles and Potential Therapeutic Applications of the P2X7 Receptor in Inflammation and Pain. Molecules 18:9, pages 10953-10972.
Crossref
Stefania Muzzachi, Antonella Blasi, Elena Ciani, Maria Favia, Rosa A. Cardone, Domenico Marzulli, Stephan J. Reshkin, Giulia Merizzi, Valeria Casavola, Antonio Soleti & Lorenzo Guerra. (2013) MED1101: A new dialdehydic compound regulating P2×7 receptor cell surface expression in U937 cells. Biology of the Cell 105:9, pages 399-413.
Crossref
David Yang-Wei Fann, Seung-Yoon Lee, Silvia Manzanero, Prasad Chunduri, Christopher G. Sobey & Thiruma V. Arumugam. (2013) Pathogenesis of acute stroke and the role of inflammasomes. Ageing Research Reviews 12:4, pages 941-966.
Crossref
Fenila Jacob, Claudina Pérez Novo, Claus Bachert & Koen Van Crombruggen. (2013) Purinergic signaling in inflammatory cells: P2 receptor expression, functional effects, and modulation of inflammatory responses. Purinergic Signalling 9:3, pages 285-306.
Crossref
Alberto Baroja-Mazo, Maria Barber?-Cremades & Pablo Pelegr?n. (2013) P2X7 Receptor Activation Impairs Exogenous MHC Class I Oligopeptides Presentation in Antigen Presenting Cells. PLoS ONE 8:8, pages e70577.
Crossref
Chin-Wei Chiao, J. Eduardo da Silva-Santos, Fernanda R. GiachiniRita C. Tostes, Ming-Jai Su & R. Clinton Webb. (2013) P2X7 receptor activation contributes to an initial upstream mechanism of lipopolysaccharide-induced vascular dysfunction. Clinical Science 125:3, pages 131-141.
Crossref
Francesco Di Virgilio. (2013) The Therapeutic Potential of Modifying Inflammasomes and NOD-Like Receptors. Pharmacological Reviews 65:3, pages 872-905.
Crossref
Andrea Vergani, Carmen Fotino, Francesca D’Addio, Sara Tezza, Michele Podetta, Francesca Gatti, Melissa Chin, Roberto Bassi, Ruth D. Molano, Domenico Corradi, Rita Gatti, Maria E. Ferrero, Antonio Secchi, Fabio GrassiCamillo Ricordi, Mohamed H. Sayegh, Paola Maffi, Antonello Pileggi & Paolo Fiorina. (2013) Effect of the Purinergic Inhibitor Oxidized ATP in a Model of Islet Allograft Rejection. Diabetes 62:5, pages 1665-1675.
Crossref
Moritz Haneklaus, Luke AJ O’Neill & Rebecca C Coll. (2013) Modulatory mechanisms controlling the NLRP3 inflammasome in inflammation: recent developments. Current Opinion in Immunology 25:1, pages 40-45.
Crossref
Elena De Santis, Maura Di Vito, Giulietta Anna Perrone, Emanuela Mari, Maria Osti, Enrico De Antoni, Luigi Coppola, Marco Tafani, Angelo Carpi & Matteo A. Russo. (2013) Overexpression of pro-inflammatory genes and down-regulation of SOCS-1 in human PTC and in hypoxic BCPAP cells. Biomedicine & Pharmacotherapy 67:1, pages 7-16.
Crossref
Andrea VerganiSara TezzaFrancesca D’AddioCarmen FotinoKaifeng LiuMonika NiewczasRoberto BassiR. Damaris MolanoSonja KleffelAlessandra PetrelliAntonio SoletiEnrico AmmiratiMaria FrigerioGary VisnerFabio GrassiMaria E. FerreroDomenico CorradiReza AbdiCamillo RicordiMohamed H. SayeghAntonello PileggiPaolo Fiorina. (2013) Long-Term Heart Transplant Survival by Targeting the Ionotropic Purinergic Receptor P2X7. Circulation 127:4, pages 463-475.
Crossref
Iman Jalilian, Mari Spildrejorde, Aine Seavers, Belinda L. Curtis, Jason D. McArthur & Ronald Sluyter. (2012) Functional expression of the damage-associated molecular pattern receptor P2X7 on canine kidney epithelial cells. Veterinary Immunology and Immunopathology 150:3-4, pages 228-233.
Crossref
Surina Zheng, Shunsuke Sugita, Shizuka Hirai & Yukari Egashira. (2012) Protective effect of low molecular fraction of MGN-3, a modified arabinoxylan from rice bran, on acute liver injury by inhibition of NF-κB and JNK/MAPK expression. International Immunopharmacology 14:4, pages 764-769.
Crossref
Paul Kubes & Wajahat Z. Mehal. (2012) Sterile Inflammation in the Liver. Gastroenterology 143:5, pages 1158-1172.
Crossref
Xu Ji, Yukiko Naito, Huachun Weng, Kosuke Endo, Xiao Ma & Naoharu Iwai. (2012) P2X 7 deficiency attenuates hypertension and renal injury in deoxycorticosterone acetate-salt hypertension . American Journal of Physiology-Renal Physiology 303:8, pages F1207-F1215.
Crossref
Lucas T. Woods, Jean M. Camden, Josef M. BatekMichael J. Petris, Laurie Erb & Gary A. Weisman. (2012) P2X7 receptor activation induces inflammatory responses in salivary gland epithelium. American Journal of Physiology-Cell Physiology 303:7, pages C790-C801.
Crossref
Iman Jalilian, Michelle Peranec, Belinda L. Curtis, Aine Seavers, Mari Spildrejorde, Vanessa Sluyter & Ronald Sluyter. (2012) Activation of the damage-associated molecular pattern receptor P2X7 induces interleukin-1β release from canine monocytes. Veterinary Immunology and Immunopathology 149:1-2, pages 86-91.
Crossref
Gary A. Weisman, Jean M. Camden, Troy S. Peterson, Deepa Ajit, Lucas T. Woods & Laurie Erb. (2012) P2 Receptors for Extracellular Nucleotides in the Central Nervous System: Role of P2X7 and P2Y2 Receptor Interactions in Neuroinflammation. Molecular Neurobiology 46:1, pages 96-113.
Crossref
Maria Barberà‐CremadesAlberto Baroja‐MazoAna I. GomezFrancisco Machado, Francesco Di Virgilio & Pablo Pelegrín. (2012) P2X7 receptor‐stimulation causes fever via PGE2 and IL‐1β release . The FASEB Journal 26:7, pages 2951-2962.
Crossref
Matthew A. Bailey, Robert J. Unwin & David G. Shirley. (2012) P2X receptors and kidney function. Wiley Interdisciplinary Reviews: Membrane Transport and Signaling 1:4, pages 503-511.
Crossref
Dejan Risti?Jens Ellrich. (2012) P2X7 receptor blockade reverses purinergic facilitation of neck muscle nociception in mice. Cephalalgia 32:7, pages 544-553.
Crossref
Lauren Nicotra, Lisa C. Loram, Linda R. Watkins & Mark R. Hutchinson. (2012) Toll-like receptors in chronic pain. Experimental Neurology 234:2, pages 316-329.
Crossref
Elena Adinolfi, Francesca Amoroso & Anna Lisa Giuliani. (2012) P2X7 Receptor Function in Bone-Related Cancer. Journal of Osteoporosis 2012, pages 1-10.
Crossref
Alberto Baroja-Mazo & Pablo Pelegrín. (2012) Modulating P2X7 Receptor Signaling during Rheumatoid Arthritis: New Therapeutic Approaches for Bisphosphonates. Journal of Osteoporosis 2012, pages 1-7.
Crossref
Gustavo B. Menezes, Daniel S. Mansur, Braedon McDonald, Paul Kubes & Mauro M. Teixeira. (2011) Sensing sterile injury: Opportunities for pharmacological control. Pharmacology & Therapeutics 132:2, pages 204-214.
Crossref

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.