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Cyclin-dependent kinase inhibitor therapy for hematologic malignancies

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Pages 723-738 | Published online: 06 May 2013

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Shaban Ahmad, Mussuvir Pasha KM, Khalid Raza, Misbahuddin M. Rafeeq, Alaa Hamed Habib, Murugesh Eswaran & Manoj Kumar Yadav. (2023) Reporting dinaciclib and theodrenaline as a multitargeted inhibitor against SARS-CoV-2: an in-silico study. Journal of Biomolecular Structure and Dynamics 41:9, pages 4013-4023.
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S.S. Liang, X.G. Liu, Y.X. Cui, S.L. Zhang, Q.G. Zhang & J.Z. Chen. (2021) Molecular mechanism concerning conformational changes of CDK2 mediated by binding of inhibitors using molecular dynamics simulations and principal component analysis. SAR and QSAR in Environmental Research 32:7, pages 573-594.
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Lubaid Saleh, Caroline Wilson & Ingunn Holen. (2020) CDK4/6 inhibitors in breast cancer – from in vitro models to clinical trials. Acta Oncologica 59:2, pages 219-232.
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Xin Wang, Kaiyuan Deng, Cheng Wang, Yao Li, Tianqi Wang, Zhi Huang, Yakun Ma, Peiqing Sun, Yi Shi, Shengyong Yang, Yan Fan & Rong Xiang. (2020) Novel CDKs inhibitors for the treatment of solid tumour by simultaneously regulating the cell cycle and transcription control. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 414-423.
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Eran Tallis & Gautam Borthakur. (2019) Novel treatments for relapsed/refractory acute myeloid leukemia with FLT3 mutations. Expert Review of Hematology 12:8, pages 621-640.
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Joan Rou-En Choo & Soo-Chin Lee. (2018) CDK4-6 inhibitors in breast cancer: current status and future development. Expert Opinion on Drug Metabolism & Toxicology 14:11, pages 1123-1138.
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Prithviraj Bose, Varsha Gandhi & Marina Konopleva. (2017) Pathways and mechanisms of venetoclax resistance. Leukemia & Lymphoma 58:9, pages 2026-2039.
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P. Carrasco Salas, L. Fernández, M. Vela, D. Bueno, B. González, J. Valentín, P. Lapunzina & A. Pérez-Martínez. (2016) The role of CDKN2A/B deletions in pediatric acute lymphoblastic leukemia. Pediatric Hematology and Oncology 33:7-8, pages 415-422.
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Jeffrey D Altenburg & Sherif S Farag. (2015) The potential role of PD0332991 (Palbociclib) in the treatment of multiple myeloma. Expert Opinion on Investigational Drugs 24:2, pages 261-271.
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Tomi K Sawyer, Joe C Wu, Jonathon R Sawyer & Jessie M English. (2013) Protein kinase inhibitors: breakthrough medicines and the next generation. Expert Opinion on Investigational Drugs 22:6, pages 675-678.
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