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Drug Evaluation

A review of montelukast in the treatment of asthma and allergic rhinitis

Pages 679-686 | Published online: 02 Mar 2005

Keep up to date with the latest research on this topic with citation updates for this article.

Read on this site (6)

Yong Chen, Tingting Feng, Yong Li, Bin Du & Weiyu Weng. (2017) Formulation and evaluation of a montelukast sodium orally disintegrating tablet with a similar dissolution profile as the marketed product. Pharmaceutical Development and Technology 22:2, pages 168-172.
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Priyanka Jain, Vaibhav Rajoriya & Varsha Kashaw. (2015) Development and Validation of Simultaneous RP-HPLC Method for the Estimation of Theophylline and Motelukast in Pharmaceutical Formulation. Analytical Chemistry Letters 5:3, pages 172-182.
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Glenis Scadding. (2009) Pediatric allergy medications: review of currently available formulations. Current Medical Research and Opinion 25:8, pages 2069-2079.
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Lieven Dupont, Emmanuel Potvin, Dana Korn, Albert Lachman, Michèle Dramaix, Julie Gusman & Rudi Peché. (2005) Improving asthma control in patients suboptimally controlled on inhaled steroids and long-acting β2‐agonists: addition of montelukast in an open-label pilot study. Current Medical Research and Opinion 21:6, pages 863-869.
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Graziano Riccioni, Carmine Di Ilio & Nicolantonio D’Orazio. (2004) An update of the leukotriene modulators for the treatment of asthma. Expert Opinion on Investigational Drugs 13:7, pages 763-776.
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Basma M. Ahmed, Noha O. Mansour, Rehab A. Sallam & Moetaza M. Soliman. (2023) Efficacy of montelukast as an adjuvant therapy in rheumatoid arthritis patients: A randomized controlled study. International Immunopharmacology 124, pages 110959.
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Diana M. Ardila, Diego F. Rodríguez, Alirio Palma, Iván Díaz Costa, Justo Cobo & Christopher Glidewell. (2022) Synthesis, and spectroscopic and structural characterization of three new styrylquinoline–benzimidazole hybrids. Acta Crystallographica Section C Structural Chemistry 78:11, pages 671-680.
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Arjun Anant, Moumita Saha, Shubham Dhiman, Priti Singh, Balak Das Kurmi, Ghanshyam Das Gupta & Vivek Asati. (2022) An analytical review for the estimation of montelukast sodium. SEPARATION SCIENCE PLUS 5:5, pages 120-137.
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Amany A. Azouz, Dina A. Hanna, Ali A. Abo-Saif & Basim Anwar Shehata Messiha. (2022) Interference with megalin expression/endocytic function by montelukast mitigates gentamicin nephrotoxicity: Downregulation of ClC-5 expression. Saudi Pharmaceutical Journal 30:2, pages 150-161.
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Neeli Satyanarayana, Kota Sathish, Sakkani Nagaraju, Ravinder Pawar, Mohmmad Faizan, Murgan Arumugavel, Thangellapally Shirisha & Dhurke Kashinath. (2022) Metal-free, one-pot synthesis of 2-styrylquinolines via Friedländer annulation and sp 3 C–H activation using 1,3-dimethylurea and l -tartaric acid (3 : 1) as a deep eutectic solvent . New Journal of Chemistry 46:4, pages 1637-1642.
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Miaomiao Zhao, Hao Li & Hui Li. (2021) The relevance of CYSLTR1 gene polymorphism to the severity of allergic rhinitis and clinical responsiveness of montelukast in children. European Archives of Oto-Rhino-Laryngology 278:12, pages 4847-4853.
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Charles Frank Schuler IV & Jenny Maribel Montejo. (2021) Allergic Rhinitis in Children and Adolescents. Immunology and Allergy Clinics of North America 41:4, pages 613-625.
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Antonietta Siciliano, Marco Guida, Maria Rosaria Iesce, Giovanni Libralato, Fabio Temussi, Emilia Galdiero, Federica Carraturo, Flavio Cermola & Marina DellaGreca. (2021) Ecotoxicity and photodegradation of Montelukast (a drug to treat asthma) in water. Environmental Research 202, pages 111680.
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Wei-Jie Li, Yun Zhao, Yuan Gao, Ling-Ling Dong, Yin-Fang Wu, Zhi-Hua Chen & Hua-Hao Shen. (2021) Lipid metabolism in asthma: Immune regulation and potential therapeutic target. Cellular Immunology 364, pages 104341.
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Johanna Michael, Diana Bessa de Sousa, Justin Conway, Erick Gonzalez-Labrada, Rodolphe Obeid, Julia Tevini, Thomas Felder, Birgit Hutter-Paier, Horst Zerbe, Nadine Paiement & Ludwig Aigner. (2020) Improved Bioavailability of Montelukast through a Novel Oral Mucoadhesive Film in Humans and Mice. Pharmaceutics 13:1, pages 12.
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N.G. Astafieva, A.A. Baranov, E.A. Vishneva, N.A. Daikhes, A.V. Zhestkov, N.I. Ilyina, O.V. Karneeva, E.P. Karpova, I.A. Kim, A.I. Kryukov, O.M. Kurbacheva, R.Ya. Meshkova, L.S. Namazova-Baranova, N.M. Nenasheva, G.A. Novik, E.V. Nosulya, K.S. Pavlova, A.N. Pampura, V.M. Svistushkin, L.R. Selimzyanova, M.R. Khaitov & R.M. Khaitov. (2020) Allergic rhinitis. Rossiiskaya rinologiya 28:4, pages 246.
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Mohammad S. Hareedy, Esraa A. Ahmed & Marwa F. Ali. (2019) Montelukast modifies simvastatin‐induced myopathy and hepatotoxicity. Drug Development Research 80:7, pages 1000-1009.
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Charles Frank Schuler IV & Jenny Maribel Montejo. (2019) Allergic Rhinitis in Children and Adolescents. Pediatric Clinics of North America 66:5, pages 981-993.
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Kunti Abhishek Shah & Vijaykumar Kunvarji Parmar. (2019) Quality by Design Based Method Development for Simultaneous Estimation of Montelukast Sodium and Theophylline in Tablet Dosage Form. Current Pharmaceutical Analysis 15:6, pages 612-623.
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Ju‑Hee Kang, Hyungsik Lim, Dong‑Seok Lee & Mijung Yim. (2018) Montelukast inhibits RANKL‑induced osteoclast formation and bone loss via CysLTR1 and P2Y12. Molecular Medicine Reports.
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Mark S. Dykewicz, Dana V. Wallace, Fuad Baroody, Jonathan Bernstein, Tim Craig, Ira Finegold, Faith Huang, Desiree Larenas-Linnemann, Eli Meltzer, Gary Steven, David I. Bernstein, Joann Blessing-Moore, Chitra Dinakar, Matthew Greenhawt, Caroline C. Horner, David A. Khan, David Lang, John Oppenheimer, Jay M. Portnoy, Christopher R. Randolph, Matthew A. Rank, Mark S. Dykewicz & Dana V. Wallace. (2017) Treatment of seasonal allergic rhinitis. Annals of Allergy, Asthma & Immunology 119:6, pages 489-511.e41.
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