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Drug Safety Evaluation

The safety of istradefylline for the treatment of Parkinson’s disease

, MD

Keep up to date with the latest research on this topic with citation updates for this article.

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F. Javier Álvarez. (2016) Parkinson’s disease, antiparkinson medicines, and driving. Expert Review of Neurotherapeutics 16:9, pages 1023-1032.
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Ruxandra Julia Vorovenci & Angelo Antonini. (2015) The efficacy of oral adenosine A2A antagonist istradefylline for the treatment of moderate to severe Parkinson’s disease. Expert Review of Neurotherapeutics 15:12, pages 1383-1390.
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Articles from other publishers (15)

Yuxin Huang. (2023) A review on the current status and development of Parkinson's clinical drugs. A review on the current status and development of Parkinson's clinical drugs.
Yuemei Wang, Yuanbing Zhu, Junmeng Wang, Longcong Dong, Shuqing Liu, Sihui Li & Qiaofeng Wu. (2023) Purinergic signaling: A gatekeeper of blood-brain barrier permeation. Frontiers in Pharmacology 14.
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Xiaoqin Hu, Jinhuan Ni, Nanyong Gao, Zhize Ye, Guoxin Hu, Jianping Cai & Jianchang Qian. (2022) The effect of CYP3A4 genetic polymorphism and drug interaction on the metabolism of istradefylline. Chemico-Biological Interactions 366, pages 110123.
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Ernesto Alberto Rendón-Ochoa, Montserrat Padilla-Orozco, Vladimir Melesio Calderon, Victor Hugo Avilés-Rosas, Omar Hernández-González, Teresa Hernández-Flores, María Belén Perez-Ramirez, Marcela Palomero-Rivero, Elvira Galarraga & José Bargas. (2022) Dopamine D 2 and Adenosine A 2A Receptors Interaction on Ca 2+ Current Modulation in a Rodent Model of Parkinsonism . ASN Neuro 14, pages 175909142211020.
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Min Shin, Madhavi Pandya, Kristan Espinosa, Ravindra Telang, Jordi Boix, Peter R. Thorne & Srdjan M. Vlajkovic. (2021) Istradefylline Mitigates Age-Related Hearing Loss in C57BL/6J Mice. International Journal of Molecular Sciences 22:15, pages 8000.
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Xiang Li, Wenjun Wang, Jianghong Yan & Fancai Zeng. (2021) Glutamic Acid Transporters: Targets for Neuroprotective Therapies in Parkinson’s Disease. Frontiers in Neuroscience 15.
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Angela Valderrama Parizotto, Ana Paula Ferro, Rogério Marchiosi, Flávia Carolina Moreira-Vilar, Jennifer Munik Bevilaqua, Wanderley Dantas dos Santos, Flávio Augusto Vicente Seixas & Osvaldo Ferrarese-Filho. (2020) Entacapone improves saccharification without affecting lignin and maize growth: An in silico, in vitro, and in vivo approach. Plant Physiology and Biochemistry 151, pages 421-428.
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Francisco M. Mouro, Attila Köfalvi, Luís A. André, Younis Baqi, Christa E. Müller, Joaquim A. Ribeiro & Ana M. Sebastião. (2019) Memory deficits induced by chronic cannabinoid exposure are prevented by adenosine A2AR receptor antagonism. Neuropharmacology 155, pages 10-21.
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Marina Cerrone, Chantal J. M. van Opbergen, Kabir Malkani, Natasha Irrera, Mingliang Zhang, Toon A. B. Van Veen, Bruce Cronstein & Mario Delmar. (2018) Blockade of the Adenosine 2A Receptor Mitigates the Cardiomyopathy Induced by Loss of Plakophilin-2 Expression. Frontiers in Physiology 9.
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Fabiana Núñez, Jaume Taura, Juan Camacho, Marc López-Cano, Víctor Fernández-Dueñas, Naomi Castro, Julio Castro & Francisco Ciruela. (2018) PBF509, an Adenosine A2A Receptor Antagonist With Efficacy in Rodent Models of Movement Disorders. Frontiers in Pharmacology 9.
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Jaume Taura, Ernest G. Nolen, Gisela Cabré, Jordi Hernando, Lucia Squarcialupi, Marc López-Cano, Kenneth A. Jacobson, Víctor Fernández-Dueñas & Francisco Ciruela. (2018) Remote control of movement disorders using a photoactive adenosine A2A receptor antagonist. Journal of Controlled Release 283, pages 135-142.
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Caio M. Massari, Marc López-Cano, Fabiana Núñez, Víctor Fernández-Dueñas, Carla I. Tasca & Francisco Ciruela. (2017) Antiparkinsonian Efficacy of Guanosine in Rodent Models of Movement Disorder. Frontiers in Pharmacology 8.
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Paulo A. de Oliveira, James A. R. Dalton, Marc López-Cano, Adrià Ricarte, Xavier Morató, Filipe C. Matheus, Andréia S. Cunha, Christa E. Müller, Reinaldo N. Takahashi, Víctor Fernández-Dueñas, Jesús Giraldo, Rui D. Prediger & Francisco Ciruela. (2017) Angiotensin II type 1/adenosine A 2A receptor oligomers: a novel target for tardive dyskinesia. Scientific Reports 7:1.
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Sergi Ferré. 2017. Adenosine Receptors in Neurodegenerative Diseases. Adenosine Receptors in Neurodegenerative Diseases 231 255 .
Lakshmi Jayashankar & Richard Hafner. (2016) Adjunct Strategies for Tuberculosis Vaccines: Modulating Key Immune Cell Regulatory Mechanisms to Potentiate Vaccination. Frontiers in Immunology 7.
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