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Time-controlled oral delivery systems for colon targeting

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Pages 583-597 | Published online: 01 Sep 2006

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Monica R. P. Rao, Rohit Vidyadhar Godbole, Sameer G. Borate, Sanskar Mahajan & Tejal Gangwal. (2021) Nanosuspension coated multiparticulates for controlled delivery of albendazole. Drug Development and Industrial Pharmacy 47:3, pages 367-376.
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Alessandra Maroni, Saliha Moutaharrik, Lucia Zema & Andrea Gazzaniga. (2017) Enteric coatings for colonic drug delivery: state of the art. Expert Opinion on Drug Delivery 14:9, pages 1027-1029.
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Mayur M. Patel & Avani F. Amin. (2013) Development of a novel tablet-in-capsule formulation of mesalamine for inflammatory bowel disease. Pharmaceutical Development and Technology 18:2, pages 390-400.
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Bo Xiao & Didier Merlin. (2012) Oral colon-specific therapeutic approaches toward treatment of inflammatory bowel disease. Expert Opinion on Drug Delivery 9:11, pages 1393-1407.
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Yellela S. R. Krishnaiah & Mansoor A. Khan. (2012) Strategies of targeting oral drug delivery systems to the colon and their potential use for the treatment of colorectal cancer. Pharmaceutical Development and Technology 17:5, pages 521-540.
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Arik Dahan, Gordon L Amidon & Ellen M Zimmermann. (2010) Drug targeting strategies for the treatment of inflammatory bowel disease: a mechanistic update. Expert Review of Clinical Immunology 6:4, pages 543-550.
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Youness Karrout, Christel Neut, Daniel Wils, Florence Siepmann, Laetitia Deremaux, Pierre Desreumaux & Juergen Siepmann. (2009) Characterization of ethylcellulose: starch-based film coatings for colon targeting. Drug Development and Industrial Pharmacy 35:10, pages 1190-1200.
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Heba S. Abd-Ellah, Ramesh Mudududdla, Glen P. Carter & Jonathan B. Baell. (2023) Design, Development, and Optimisation of Smart Linker Chemistry for Targeted Colonic Delivery—In Vitro Evaluation. Pharmaceutics 15:1, pages 303.
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Susan Hua & Ephraem C. Lye. (2022) Impact of gastric and bowel surgery on gastrointestinal drug delivery. Drug Delivery and Translational Research 13:1, pages 37-53.
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Alessia Favaron, Laura E. McCoubrey, Moe Elbadawi, Abdul W. Basit & Mine Orlu. 2023. Pharmaceutical Formulations for Older Patients. Pharmaceutical Formulations for Older Patients 191 230 .
Zih-Sian Yang, Hung-Yi Song, Kai-Min Yang & Po-Yuan Chiang. (2022) The physicochemical properties and the release of sodium caseinate/ polysaccharide gum chlorophyll multiple-layer particles by rotary side-spray fluid bed technology. Food Chemistry 394, pages 133442.
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Ankita N. Yawalkar, Manoj A. Pawar & Pradeep R. Vavia. (2022) Microspheres for targeted drug delivery- A review on recent applications. Journal of Drug Delivery Science and Technology 75, pages 103659.
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Atheer Awad, Christine M. Madla, Laura E. McCoubrey, Fabiana Ferraro, Francesca K.H. Gavins, Asma Buanz, Simon Gaisford, Mine Orlu, Florence Siepmann, Juergen Siepmann & Abdul W. Basit. (2022) Clinical translation of advanced colonic drug delivery technologies. Advanced Drug Delivery Reviews 181, pages 114076.
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Hossein Shahdadi Sardou, Abbas Akhgari, Amir Hooshang Mohammadpour, Ali Beheshti Namdar, Hossein Kamali, Amir Hossein Jafarian, Hadi Afrasiabi Garekani & Fatemeh Sadeghi. (2022) Optimization study of combined enteric and time-dependent polymethacrylates as a coating for colon targeted delivery of 5-ASA pellets in rats with ulcerative colitis. European Journal of Pharmaceutical Sciences 168, pages 106072.
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Shabnam Hosseini, Oliver Wetzel, Kathrin Kostka, Marc Heggen, Kateryna Loza & Matthias Epple. (2021) Pathways for Oral and Rectal Delivery of Gold Nanoparticles (1.7 nm) and Gold Nanoclusters into the Colon: Enteric-Coated Capsules and Suppositories. Molecules 26:16, pages 5069.
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Alice Melocchi, Marco Uboldi, Francesco Briatico-Vangosa, Saliha Moutaharrik, Matteo Cerea, Anastasia Foppoli, Alessandra Maroni, Luca Palugan, Lucia Zema & Andrea Gazzaniga. (2021) The Chronotopic™ System for Pulsatile and Colonic Delivery of Active Molecules in the Era of Precision Medicine: Feasibility by 3D Printing via Fused Deposition Modeling (FDM). Pharmaceutics 13:5, pages 759.
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Rayan Sabra & Nashiru Billa. (2021) Soliciting the Oral Route as a Logical Approach to Managing Colon Cancer. Frontiers in Bioengineering and Biotechnology 9.
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Susan Hua. (2020) Advances in Oral Drug Delivery for Regional Targeting in the Gastrointestinal Tract - Influence of Physiological, Pathophysiological and Pharmaceutical Factors. Frontiers in Pharmacology 11.
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Minh N.U. Nguyen, Phuong H.L. Tran & Thao T.D. Tran. (2019) A single-layer film coating for colon-targeted oral delivery. International Journal of Pharmaceutics 559, pages 402-409.
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Priyanka Bhatt, Deepa Patel, Ankita Patel, Akanksha Patel & Aishwarya Nagarsheth. 2019. Novel Drug Delivery Technologies. Novel Drug Delivery Technologies 73 120 .
V. V. Golotiuk. (2018) PROSPECTS OF APPLICATION OF PECTIN MODIFICATIONS IN THE COMPLEX MEDICAMENT THERAPY OF COLORECTAL CANCER. Bulletin of Problems Biology and Medicine 1.1:142, pages 25.
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Rouslan I. Moustafine, Alexander Y. Sitenkov, Alexandra V. Bukhovets, Shamil F. Nasibullin, Bernard Appeltans, Tatiana V. Kabanova, Vitaliy V. Khutoryanskiy & Guy Van den Mooter. (2017) Indomethacin-containing interpolyelectrolyte complexes based on Eudragit® E PO/S 100 copolymers as a novel drug delivery system. International Journal of Pharmaceutics 524:1-2, pages 121-133.
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Serena Mazzucchelli & Fabio Corsi. (2017) Diabetes management strategies: can nanoparticles be used to therapeutically deliver insulin?. Therapeutic Delivery 8:2, pages 49-51.
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Alessandra Maroni, Maria Dorly Del Curto, Stefano Salmaso, Lucia Zema, Alice Melocchi, Paolo Caliceti & Andrea Gazzaniga. (2016) In vitro and in vivo evaluation of an oral multiple-unit formulation for colonic delivery of insulin. European Journal of Pharmaceutics and Biopharmaceutics 108, pages 76-82.
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Lucia Salvioni, Luisa Fiandra, Maria Dorly Del Curto, Serena Mazzucchelli, Raffaele Allevi, Marta Truffi, Luca Sorrentino, Benedetta Santini, Matteo Cerea, Luca Palugan, Fabio Corsi & Miriam Colombo. (2016) Oral delivery of insulin via polyethylene imine-based nanoparticles for colonic release allows glycemic control in diabetic rats. Pharmacological Research 110, pages 122-130.
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Sheng Qi & Duncan Craig. (2016) Recent developments in micro- and nanofabrication techniques for the preparation of amorphous pharmaceutical dosage forms. Advanced Drug Delivery Reviews 100, pages 67-84.
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Alessandra Maroni, Lucia Zema, Matteo Cerea, Anastasia Foppoli, Luca Palugan & Andrea Gazzaniga. (2016) Erodible drug delivery systems for time-controlled release into the gastrointestinal tract. Journal of Drug Delivery Science and Technology 32, pages 229-235.
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Elena Macchi, Lucia Zema, Preetanshu Pandey, Andrea Gazzaniga & Linda A. Felton. (2016) Influence of temperature and relative humidity conditions on the pan coating of hydroxypropyl cellulose molded capsules. European Journal of Pharmaceutics and Biopharmaceutics 100, pages 47-57.
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E. Macchi, L. Zema, A. Maroni, A. Gazzaniga & L.A. Felton. (2015) Enteric-coating of pulsatile-release HPC capsules prepared by injection molding. European Journal of Pharmaceutical Sciences 70, pages 1-11.
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Luca Palugan, Matteo Cerea, Lucia Zema, Andrea Gazzaniga & Alessandra Maroni. (2015) Coated pellets for oral colon delivery. Journal of Drug Delivery Science and Technology 25, pages 1-15.
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Bibi F. Choonara, Yahya E. Choonara, Pradeep Kumar, Divya Bijukumar, Lisa C. du Toit & Viness Pillay. (2014) A review of advanced oral drug delivery technologies facilitating the protection and absorption of protein and peptide molecules. Biotechnology Advances 32:7, pages 1269-1282.
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Maria Dorly Del Curto, Luca Palugan, Anastasia Foppoli, Lucia Zema, Andrea Gazzaniga & Alessandra Maroni. (2014) Erodible Time‐Dependent Colon Delivery Systems with Improved Efficiency in Delaying the Onset of Drug Release. Journal of Pharmaceutical Sciences 103:11, pages 3585-3593.
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Rajesh A Keraliya & Madhabhai M Patel. (2014) Effect of viscosity of hydrophilic coating polymer on lag time of atenolol pulsatile press coated tablets. Journal of Pharmaceutical Chemistry 1:1, pages 15-21.
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Alessandra Maroni, Maria Dorly Del Curto, Lucia Zema, Anastasia Foppoli & Andrea Gazzaniga. (2013) Film coatings for oral colon delivery. International Journal of Pharmaceutics 457:2, pages 372-394.
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Alessandra Maroni, Maria Dorly Del Curto, Matteo Cerea, Lucia Zema, Anastasia Foppoli & Andrea Gazzaniga. (2013) Polymeric coatings for a multiple-unit pulsatile delivery system: Preliminary study on free and applied films. International Journal of Pharmaceutics 440:2, pages 256-263.
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Lucia Zema, Giulia Loreti, Alice Melocchi, Alessandra Maroni, Luca Palugan & Andrea Gazzaniga. (2013) Gastroresistant capsular device prepared by injection molding. International Journal of Pharmaceutics 440:2, pages 264-272.
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Jing Liu, Liangke Zhang, Yuntao Jia, Wenjing Hu, Jingqing Zhang & Huiming Jiang. (2012) Preparation and evaluation of pectin-based colon-specific pulsatile capsule in vitro and in vivo. Archives of Pharmacal Research 35:11, pages 1927-1934.
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B. M. Ursekar, P. S. Soni, Abhijit A. Date & M. S. Nagarsenker. (2012) Characterization of Soy Polysaccharide and Its In Vitro and In Vivo Evaluation for Application in Colon Drug Delivery. AAPS PharmSciTech 13:3, pages 934-943.
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Lucia Zema, Giulia Loreti, Alice Melocchi, Alessandra Maroni & Andrea Gazzaniga. (2012) Injection Molding and its application to drug delivery. Journal of Controlled Release 159:3, pages 324-331.
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Alessandra Maroni, Lucia Zema, Maria Dorly Del Curto, Anastasia Foppoli & Andrea Gazzaniga. (2012) Oral colon delivery of insulin with the aid of functional adjuvants. Advanced Drug Delivery Reviews 64:6, pages 540-556.
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Jing Liu, Liangke Zhang, Wenjing Hu, Rui Tian, Yongzhen Teng & Chengyuan Wang. (2012) Preparation of konjac glucomannan-based pulsatile capsule for colonic drug delivery system and its evaluation in vitro and in vivo. Carbohydrate Polymers 87:1, pages 377-382.
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