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Regulation of human hepatic drug transporter expression by pro-inflammatory cytokines

, PharmD PhD &
Pages 1469-1481 | Published online: 28 Sep 2009

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Karima Alim, Arnaud Bruyère, Alain Lescoat, Elodie Jouan, Valérie Lecureur, Marc Le Vée & Olivier Fardel. (2021) Interactions of janus kinase inhibitors with drug transporters and consequences for pharmacokinetics and toxicity. Expert Opinion on Drug Metabolism & Toxicology 17:3, pages 259-271.
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Eva Ramboer, Tamara Vanhaecke, Vera Rogiers & Mathieu Vinken. (2013) Primary hepatocyte cultures as prominent in vitro tools to study hepatic drug transporters. Drug Metabolism Reviews 45:2, pages 196-217.
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Olivier Fardel. (2013) Cytokines as molecular targets for aryl hydrocarbon receptor ligands: implications for toxicity and xenobiotic detoxification. Expert Opinion on Drug Metabolism & Toxicology 9:2, pages 141-152.
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Tommy B Andersson, Kajsa P Kanebratt & John Gerry Kenna. (2012) The HepaRG cell line: a unique in vitro tool for understanding drug metabolism and toxicology in human. Expert Opinion on Drug Metabolism & Toxicology 8:7, pages 909-920.
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Alexander M Cressman, Vanja Petrovic & Micheline Piquette-Miller. (2012) Inflammation-mediated changes in drug transporter expression/activity: implications for therapeutic drug response. Expert Review of Clinical Pharmacology 5:1, pages 69-89.
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Olivier Fardel, Elise Kolasa & Marc Le Vee. (2012) Environmental chemicals as substrates, inhibitors or inducers of drug transporters: implication for toxicokinetics, toxicity and pharmacokinetics. Expert Opinion on Drug Metabolism & Toxicology 8:1, pages 29-46.
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Neill James Liptrott & Andrew Owen. (2011) The role of cytokines in the regulation of drug disposition: extended functional pleiotropism?. Expert Opinion on Drug Metabolism & Toxicology 7:3, pages 341-352.
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