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Expert Opinion on Drug Discovery Volume 6, 2011 - Issue 5
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Approaches to the rational design of selective melanocortin receptor antagonists

Victor J HrubyUniversity of Arizona, Department of Chemistry and Biochemistry, 1306 E. University Blvd., Tucson, AZ 85721, [email protected]
,
Minying CaiUniversity of Arizona, Department of Chemistry and Biochemistry, 1306 E. University Blvd., Tucson, AZ 85721, [email protected]
,
Joel NybergUniversity of Arizona, Department of Chemistry and Biochemistry, 1306 E. University Blvd., Tucson, AZ 85721, [email protected]
&
Dhanasekaran MuthuUniversity of Arizona, Department of Chemistry and Biochemistry, 1306 E. University Blvd., Tucson, AZ 85721, [email protected]
Pages 543-557 | Published online: 24 Mar 2011

Citations (7)

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Read on this site (1)

Yang Zhou & Minying Cai. (2017) Novel approaches to the design of bioavailable melanotropins. Expert Opinion on Drug Discovery 12:10, pages 1023-1030.
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Articles from other publishers (6)

Uru Malik, Lai Yue Chan, Minying Cai, Victor J. Hruby, Quentin Kaas, Norelle L. Daly & David J. Craik. (2020) Development of novel frog‐skin peptide scaffolds with selectivity towards melanocortin receptor subtypes. Peptide Science 113:4.
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Charlotte Martin, Luis E. Gimenez, Savannah Y. Williams, Yu Jing, Yiran Wu, Charlie Hollanders, Olivier Van der Poorten, Simon Gonzalez, Kevin Van holsbeeck, Santo Previti, Arthur Lamouroux, Suwen Zhao, Dirk Tourwé, Raymond C. Stevens, Roger D. Cone & Steven Ballet. (2020) Structure-Based Design of Melanocortin 4 Receptor Ligands Based on the SHU-9119-hMC4R Cocrystal Structure. Journal of Medicinal Chemistry 64:1, pages 357-369.
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Francesco Merlino, Yang Zhou, Minying Cai, Alfonso Carotenuto, Ali M. Yousif, Diego Brancaccio, Salvatore Di Maro, Silvia Zappavigna, Antonio Limatola, Ettore Novellino, Paolo Grieco & Victor J. Hruby. (2018) Development of Macrocyclic Peptidomimetics Containing Constrained α,α-Dialkylated Amino Acids with Potent and Selective Activity at Human Melanocortin Receptors. Journal of Medicinal Chemistry 61:9, pages 4263-4269.
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Shanthi Kanthala, Sashikanth Banappagari, Ameya Gokhale, Yong-Yu Liu, Gu Xin, Yunfeng Zhao & Seetharama Jois. (2015) Novel Peptidomimetics for Inhibition of HER2:HER3 Heterodimerization in HER2-Positive Breast Cancer. Chemical Biology & Drug Design 85:6, pages 702-714.
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Shanthi Kanthala, Ted Gauthier & Seetharama Satyanarayanajois. (2014) Structure-activity relationships of peptidomimetics that inhibit PPI of HER2-HER3. Biopolymers 101:6, pages 693-702.
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Minying Cai, Magda Stankova, Dhanasekaran Muthu, Alexander Mayorov, Zhehui Yang, Devendra Trivedi, Christopher Cabello & Victor J. Hruby. (2013) An Unusual Conformation of γ-Melanocyte-Stimulating Hormone Analogues Leads to a Selective Human Melanocortin 1 Receptor Antagonist for Targeting Melanoma Cells. Biochemistry 52:4, pages 752-764.
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