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Mostafa M. M. El-Miligy, Marwa E. Abdelaziz, Salwa M. Fahmy, Tamer M. Ibrahim, Marwa M. Abu-Serie, Mona A. Mahran & Aly A. Hazzaa. (2023) Discovery of new pyridine-quinoline hybrids as competitive and non-competitive PIM-1 kinase inhibitors with apoptosis induction and caspase 3/7 activation capabilities. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Gubbi M Arunesh, Ekambaram Shanthi, Mudeenahally H Krishna, Jegatheesan Sooriya Kumar & Vellarkad N Viswanadhan. (2014) Small molecule inhibitors of PIM1 kinase: July 2009 to February 2013 patent update. Expert Opinion on Therapeutic Patents 24:1, pages 5-17.
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Samy Mohamady, Ahmed F. Khalil, Bassem H. Naguib, Mohamed S. Nafie, Haytham O. Tawfik & Moataz A. Shaldam. (2024) Tailored horseshoe-shaped nicotinonitrile scaffold as dual promising c-Met and Pim-1 inhibitors: Design, synthesis, SAR and in silico study. Bioorganic Chemistry 143, pages 106988.
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Zhao Deng & Des R. Richardson. (2023) The Myc Family and the Metastasis Suppressor NDRG1: Targeting Key Molecular Interactions with Innovative Therapeutics. Pharmacological Reviews 75:5, pages 1007-1035.
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Haifa Almukadi, Gada Ali Jadkarim, Arif Mohammed, Majid Almansouri, Nasreen Sultana, Noor Ahmad Shaik & Babajan Banaganapalli. (2023) Combining machine learning and structure-based approaches to develop oncogene PIM kinase inhibitors. Frontiers in Chemistry 11.
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Jing Huang, Ye Yuan, Xiaoxiao Zhu, Guodong Li, Ya Xu, Wenlin Chen & Ying Zhu. (2022) Identification of Pim-1 Kinase Inhibitors by Pharmacophore Model, Molecular
Docking-based Virtual Screening, and Biological Evaluation. Current Computer-Aided Drug Design 18:3, pages 240-246.
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Vinayak Walhekar, Chandrakant Bagul, Dileep Kumar, Amol Muthal, Garlapati Achaiah & Ravindra Kulkarni. (2022) Topical advances in PIM kinases and their inhibitors: Medicinal chemistry perspectives. Biochimica et Biophysica Acta (BBA) - Reviews on Cancer 1877:3, pages 188725.
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Youyi Zhao, Aziz ur Rehman Aziz, Hangyu Zhang, Zhengyao Zhang, Na Li & Bo Liu. (2022) A systematic review on active sites and functions of PIM-1 protein. Human Cell 35:2, pages 427-440.
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Hafez Razmazma, Ali Ebrahimi & Mohammad Hashemi. (2020) Structural insights for rational design of new PIM-1 kinase inhibitors based on 3,5-disubstituted indole derivatives: An integrative computational approach. Computers in Biology and Medicine 118, pages 103641.
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Ronja Bjørnstad, Reidun Aesoy, Øystein Bruserud, Annette K. Brenner, Francis Giraud, Tara Helen Dowling, Gro Gausdal, Pascale Moreau, Stein Ove Døskeland, Fabrice Anizon & Lars Herfindal. (2019) A Kinase Inhibitor with Anti-Pim Kinase Activity is a Potent and Selective Cytotoxic Agent Toward Acute Myeloid Leukemia. Molecular Cancer Therapeutics 18:3, pages 567-578.
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Lubna Swellmeen, Rand Shahin, Yusuf Al-Hiari, Amani Alamiri, Alaa Hasan & Omar Shaheen. (2017) Structure based drug design of Pim-1 kinase followed by pharmacophore guided synthesis of quinolone-based inhibitors. Bioorganic & Medicinal Chemistry 25:17, pages 4855-4875.
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Jong-Eun Kim, Joe Eun Son, Hyein Jeong, Dong Joon Kim, Sang Gwon Seo, Eunjung Lee, Tae Gyu Lim, Jong Rhan Kim, Yengo Raymond Kimbung, Hanyong Chen, Ann M. Bode, Ki Won Lee & Zigang Dong. (2015) A Novel Cinnamon-Related Natural Product with Pim-1 Inhibitory Activity Inhibits Leukemia and Skin Cancer. Cancer Research 75:13, pages 2716-2728.
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Wei Li, Xiaobo Wan, Fanqi Zeng, Yuting Xie, Yanli Wang, Wei Zhang, Li Li & Niu Huang. (2014) More than just a GPCR ligand: structure-based discovery of thioridazine derivatives as Pim-1 kinase inhibitors. Med. Chem. Commun. 5:4, pages 507-511.
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Ramesh Ekambaram, Erki Enkvist, Ganesh babu Manoharan, Mihkel Ugandi, Marje Kasari, Kaido Viht, Stefan Knapp, Olaf-Georg Issinger & Asko Uri. (2014) Benzoselenadiazole-based responsive long-lifetime photoluminescent probes for protein kinases. Chem. Commun. 50:31, pages 4096-4098.
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Mingzhang Gao, Min Wang, Kathy D. Miller & Qi-Huang Zheng. (2013) Synthesis of (Z)-2-((1H-indazol-3-yl)methylene)-6-[11C]methoxy-7-(piperazin-1-ylmethyl)benzofuran-3(2H)-one as a new potential PET probe for imaging of the enzyme PIM1. Bioorganic & Medicinal Chemistry Letters 23:15, pages 4342-4346.
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Ramesh Ekambaram, Erki Enkvist, Angela Vaasa, Marje Kasari, Gerda Raidaru, Stefan Knapp & Asko Uri. (2013) Selective Bisubstrate Inhibitors with Sub-nanomolar Affinity for Protein Kinase Pim-1. ChemMedChem 8:6, pages 909-913.
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