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Takeru Ehara, Osamu Irie, Takatoshi Kosaka, Takanori Kanazawa, Werner Breitenstein, Philipp Grosche, Nils Ostermann, Masaki Suzuki, Shimpei Kawakami, Kazuhide Konishi, Yuko Hitomi, Atsushi Toyao, Hiroki Gunji, Frederic Cumin, Nikolaus Schiering, Trixie Wagner, Dean F. Rigel, Randy L. Webb, Jürgen Maibaum & Fumiaki Yokokawa. (2014) Structure-Based Design of Substituted Piperidines as a New Class of Highly Efficacious Oral Direct Renin Inhibitors. ACS Medicinal Chemistry Letters 5:7, pages 787-792.
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