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Recent developments in the use of differential scanning fluorometry in protein and small molecule discovery and characterization

Pages 1071-1082 | Published online: 06 Jun 2013

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Thamires Quadros Froes, Bianca Trindade Chaves, Marina Sena Mendes, Rafael Matos Ximenes, Ivanildo Mangueira da Silva, Priscila Brandão Gomes da Silva, Julianna Ferreira Cavalcanti de Albuquerque & Marcelo Santos Castilho. (2021) Synthesis and biological evaluation of thiazolidinedione derivatives with high ligand efficiency to P. aeruginosa PhzS. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 1217-1229.
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Chuanhu Han, Yuanrong Zheng, Changyu Zhou, Yiqi Liang, Siqiang Huang, Yangying Sun, Jinxuan Cao, Jun He, Francisco J. Barba, Jiqiang Liu, Daodong Pan & Qiang Xia. (2023) Pressurization-induced molten globule-like protein as a regulatory target for off-flavor controlling: Thermodynamic evidence and molecular modeling. Food Control 154, pages 110022.
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Poppy Llowarch, Laura Usselmann, Delyan Ivanov & Geoffrey A. Holdgate. (2023) Thermal unfolding methods in drug discovery. Biophysics Reviews 4:2.
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Emma R. Wolf-Saxon, Chad C. Moorman, Anthony Castro, Alfredo Ruiz-Rivera, Jeremy P. Mallari & Jason R. Burke. (2023) Regulatory ligand binding in plant chalcone isomerase–like (CHIL) proteins. Journal of Biological Chemistry 299:6, pages 104804.
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Paula Leandro, Paulo R. Lino, Raquel Lopes, João Leandro, Mariana P. Amaro, Paulo Sousa, João B. Vicente & António J. Almeida. (2023) Isothermal denaturation fluorimetry vs differential scanning fluorimetry as tools for screening of stabilizers for protein freeze-drying: Human phenylalanine hydroxylase as the case study. European Journal of Pharmaceutics and Biopharmaceutics 187, pages 1-11.
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Emilia Christofi & Perdita Barran. (2023) Ion Mobility Mass Spectrometry (IM-MS) for Structural Biology: Insights Gained by Measuring Mass, Charge, and Collision Cross Section. Chemical Reviews 123:6, pages 2902-2949.
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Filipa S. S. Engrola, João Paquete-Ferreira, Teresa Santos-Silva, Márcia A. S. Correia, Francisco Leisico & Marino F. A. Santos. 2023. Advanced Methods in Structural Biology. Advanced Methods in Structural Biology 199 213 .
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Petar Iliev, Danielle Hanke & Brent D. G. Page. (2022) STAT Protein Thermal Shift Assays to Monitor Protein‐Inhibitor Interactions. ChemBioChem 23:20.
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Zhao Cui, Peng Chen, Caifeng Li, Shiwen Deng & Hongjun Yang. (2022) Chip-DSF: A rapid screening strategy for drug protein targets. Pharmacological Research 182, pages 106346.
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Brice A. P. Wilson, Christopher C. Thornburg, Curtis J. Henrich, Tanja Grkovic & Barry R. O'Keefe. (2020) Creating and screening natural product libraries. Natural Product Reports 37:7, pages 893-918.
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