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Xenobiotica
the fate of foreign compounds in biological systems
Volume 41, 2011 - Issue 9
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General Xenobiochemistry

Interaction of sirolimus and everolimus with hepatic and intestinal organic anion-transporting polypeptide transporters

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Pages 752-757 | Received 29 Dec 2010, Accepted 17 Mar 2011, Published online: 27 Apr 2011

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Hallvard Holdaas, Karsten Midtvedt & Anders Åsberg. (2012) A drug safety evaluation of everolimus in kidney transplantation. Expert Opinion on Drug Safety 11:6, pages 1013-1022.
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Ashwin Kamath, Suresh Kumar Srinivasamurthy, Mukta N. Chowta, Sheetal D. Ullal, Youssef Daali & Uppugunduri S. Chakradhara Rao. (2022) Role of Drug Transporters in Elucidating Inter-Individual Variability in Pediatric Chemotherapy-Related Toxicities and Response. Pharmaceuticals 15:8, pages 990.
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Taleah Farasyn, Alexandra Crowe, Oliver Hatley, Sibylle Neuhoff, Khondoker Alam, Jean Kanyo, TuKiet T. Lam, Kai Ding & Wei Yue. (2019) Preincubation With Everolimus and Sirolimus Reduces Organic Anion-Transporting Polypeptide (OATP)1B1- and 1B3-Mediated Transport Independently of mTOR Kinase Inhibition: Implication in Assessing OATP1B1- and OATP1B3-Mediated Drug-Drug Interactions. Journal of Pharmaceutical Sciences 108:10, pages 3443-3456.
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Konrad MeissnerJane BloodAmber M. FrancisViktar YermolenkaEvan D. Kharasch. (2014) Cyclosporine-inhibitable Cerebral Drug Transport Does Not Influence Clinical Methadone Pharmacodynamics. Anesthesiology 121:6, pages 1281-1291.
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Margarida Estudante, José G. Morais, Graça Soveral & Leslie Z. Benet. (2013) Intestinal drug transporters: An overview. Advanced Drug Delivery Reviews 65:10, pages 1340-1356.
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Fabien Lamoureux, Nicolas Picard, Belkacem Boussera, François‐Ludovic Sauvage & Pierre Marquet. (2011) Sirolimus and everolimus intestinal absorption and interaction with calcineurin inhibitors: a differential effect between cyclosporine and tacrolimus. Fundamental & Clinical Pharmacology 26:4, pages 463-472.
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K Mandery, H Glaeser & MF Fromm. (2011) Interaction of innovative small molecule drugs used for cancer therapy with drug transporters. British Journal of Pharmacology 165:2, pages 345-362.
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