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Xenobiotica
the fate of foreign compounds in biological systems
Volume 42, 2012 - Issue 10
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General Xenobiochemistry

Identification of human cytochrome P450 isoforms and esterases involved in the metabolism of mirabegron, a potent and selective β3-adrenoceptor agonist

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Pages 957-967 | Received 02 Feb 2012, Accepted 08 Mar 2012, Published online: 18 Apr 2012

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Danyi Lu, Dong Dong, Zhong Liu, Yifei Wang & Baojian Wu. (2015) Metabolism elucidation of BJ-B11 (a heat shock protein 90 inhibitor) by human liver microsomes: identification of main contributing enzymes. Expert Opinion on Drug Metabolism & Toxicology 11:7, pages 1029-1040.
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Emilio Sacco, Riccardo Bientinesi, Daniele Tienforti, Marco Racioppi, Gaetano Gulino, Daniele D'Agostino, Matteo Vittori & Pierfrancesco Bassi. (2014) Discovery history and clinical development of mirabegron for the treatment of overactive bladder and urinary incontinence. Expert Opinion on Drug Discovery 9:4, pages 433-448.
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Umberto Leone Roberti Maggiore, Linda Cardozo, Simone Ferrero, Filomena Sileo, Alice Cola, Marco Torella, Nicola Colacurci, Massimo Candiani & Stefano Salvatore. (2014) Mirabegron in the treatment of overactive bladder. Expert Opinion on Pharmacotherapy 15:6, pages 873-887.
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Karl-Erik Andersson. (2013) New developments in the management of overactive bladder: focus on mirabegron and onabotulinumtoxinA. Therapeutics and Clinical Risk Management 9, pages 161-170.
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Raymond T Lee, Mitchell Bamberger & Pamela Ellsworth. (2013) Impact of mirabegron extended-release on the treatment of overactive bladder with urge urinary incontinence, urgency, and frequency. Research and Reports in Urology 5, pages 147-157.
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Mahendra Kashyap & Pradeep Tyagi. (2013) The pharmacokinetic evaluation of mirabegron as an overactive bladder therapy option. Expert Opinion on Drug Metabolism & Toxicology 9:5, pages 617-627.
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