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Drug Development and Industrial Pharmacy Volume 37, 2011 - Issue 7
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Research Article

Polymorphic transformation of anhydrous caffeine under compression and grinding: a re-evaluation.

Vincent MazelEA 401 “Matériaux et Santé”, UFR de Pharmacie, Université Paris-sud 11, 5, avenue Jean Baptiste Clément, 92296 Châtenay Malabry Cedex, FranceCorrespondence[email protected]
,
Céline DelplaceEA 401 “Matériaux et Santé”, UFR de Pharmacie, Université Paris-sud 11, 5, avenue Jean Baptiste Clément, 92296 Châtenay Malabry Cedex, France
,
Virginie BusigniesEA 401 “Matériaux et Santé”, UFR de Pharmacie, Université Paris-sud 11, 5, avenue Jean Baptiste Clément, 92296 Châtenay Malabry Cedex, France
,
Vincent FaivreUMR 8612, Laboratoire de Physico-Chimie des Systèmes Polyphasés, UFR de Pharmacie, Université Paris-sud 11, 5, avenue Jean Baptiste Clément, 92296 Châtenay Malabry Cedex, France
,
Pierre TchoreloffEA 401 “Matériaux et Santé”, UFR de Pharmacie, Université Paris-sud 11, 5, avenue Jean Baptiste Clément, 92296 Châtenay Malabry Cedex, France
&
Najet YagoubiEA 401 “Matériaux et Santé”, UFR de Pharmacie, Université Paris-sud 11, 5, avenue Jean Baptiste Clément, 92296 Châtenay Malabry Cedex, France
Pages 832-840 | Received 05 Jul 2010, Accepted 01 Dec 2010, Published online: 10 Jan 2011

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Maria Betânia de Freitas-Marques, Talita Santos do Valle, Bárbara Caroline Rodrigues de Araujo, Rita de Cássia de Oliveira Sebastião, Wagner da Nova Mussel, Maria Irene Yoshida & Christian Fernandes. (2023) Thermal energy and tableting effects in benznidazole product: the impacts of industrial processing. Drug Development and Industrial Pharmacy 49:6, pages 416-428.
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Tingting Meng, Fangxia Qiao, Shijie Ma, Ting Gao, Li Li, Yanhui Hou & Jianhong Yang. (2021) Exploring the influence factors and improvement strategies of drug polymorphic transformation combined kinetic and thermodynamic perspectives during the formation of nanosuspensions. Drug Development and Industrial Pharmacy 47:12, pages 1867-1880.
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Audrey Juban, Stephanie Briancon & François Puel. (2016) Processing-induced-transformations (PITs) during direct compression: impact of compression speeds on phase transition of caffeine. Drug Development and Industrial Pharmacy 42:11, pages 1857-1864.
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Mengran Guo, Shugang Qin, Shiyan Wang, Min Sun, Huiling Yang, Xinchun Wang, Ping Fan & Zhaohui Jin. (2023) Herbal Medicine Nanocrystals: A Potential Novel Therapeutic Strategy. Molecules 28:17, pages 6370.
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Heejun Park, Jeong-Soo Kim, Seongwoo Hong, Eun-Sol Ha, Haichen Nie, Qi Tony Zhou & Min-Soo Kim. (2022) Tableting process-induced solid-state polymorphic transition. Journal of Pharmaceutical Investigation 52:2, pages 175-194.
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Qin Shi, Haibiao Chen, Yanan Wang, Jia Xu, Ziying Liu & Chen Zhang. (2022) Recent advances in drug polymorphs: Aspects of pharmaceutical properties and selective crystallization. International Journal of Pharmaceutics 611, pages 121320.
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Taichiro TogoToshiya TaniguchiYoshitaka Nakata. (2018) The Effect of Compaction Force on the Transition to Hydrate of Anhydrous Aripiprazole. Chemical and Pharmaceutical Bulletin 66:3, pages 263-269.
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Tinne Monteyne, Jochem Vancoillie, Jean-Paul Remon, Chris Vervaet & Thomas De Beer. (2016) Continuous melt granulation: Influence of process and formulation parameters upon granule and tablet properties. European Journal of Pharmaceutics and Biopharmaceutics 107, pages 249-262.
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Alain Hedoux. 2016. Disordered Pharmaceutical Materials. Disordered Pharmaceutical Materials 361 392 .
Tinne Monteyne, Liza Heeze, Klaus Oldörp, Chris Vervaet, Jean-Paul Remon & Thomas De Beer. (2016) Vibrational spectroscopy to support the link between rheology and continuous twin-screw melt granulation on molecular level: A case study. European Journal of Pharmaceutics and Biopharmaceutics 103, pages 127-135.
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Audrey Juban, Stéphanie Briançon & François Puel. (2016) Processing-induced-transformations (PITs) during direct compression: Impact of tablet composition and compression load on phase transition of caffeine. International Journal of Pharmaceutics 501:1-2, pages 253-264.
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Marija Zba?nik, Ivana Nogalo, Dominik Cin?i? & Branko Kaitner. (2015) Polymorphism control in the mechanochemical and solution-based synthesis of a thermochromic Schiff base. CrystEngComm 17:41, pages 7870-7877.
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Jatin Sood, Bharti Sapra, Sameer Bhandari, Manish Jindal & Ashok K Tiwary. (2014) Understanding pharmaceutical polymorphic transformations I: influence of process variables and storage conditions. Therapeutic Delivery 5:10, pages 1123-1142.
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Sharmistha Pal, B. N. Roopa, Khalid Abu, Sulur G. Manjunath & Sudhir Nambiar. (2013) Thermal studies of furosemide–caffeine binary system that forms a cocrystal. Journal of Thermal Analysis and Calorimetry 115:3, pages 2261-2268.
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William Jones & Mark D. Eddleston. (2014) Introductory Lecture: Mechanochemistry, a versatile synthesis strategy for new materials. Faraday Discuss. 170, pages 9-34.
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Alain Hédoux, Yannick Guinet, Laurent Paccou, Florence Danède & Patrick Derollez. (2013) Polymorphic Transformation of Anhydrous Caffeine upon Grinding and Hydrostatic Pressurizing Analyzed by Low-Frequency Raman Spectroscopy. Journal of Pharmaceutical Sciences 102:1, pages 162-170.
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Gerti Weber Brun, Ángel Martín, Eduardo Cassel, Rubem Mário Figueiró Vargas & María José Cocero. (2012) Crystallization of Caffeine by Supercritical Antisolvent (SAS) Process: Analysis of Process Parameters and Control of Polymorphism. Crystal Growth & Design 12:4, pages 1943-1951.
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