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Drug Development and Industrial Pharmacy Volume 20, 1994 - Issue 18
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Research Article

X-Ray Powder Diffraction Study on the Grinding Effect of the Polymorphs of a Novel and Orally Effective Uricosuric Agent: FR76505

Akira Miyamae Analytical Research Laboratories, Fujisawa Pharmaceutical Co., Ltd., Kashima, Yodogawa-ku, Osaka, 532, Japan
,
Hisami Kema Analytical Research Laboratories, Fujisawa Pharmaceutical Co., Ltd., Kashima, Yodogawa-ku, Osaka, 532, Japan
,
Tetsuo Kawabata Analytical Research Laboratories, Fujisawa Pharmaceutical Co., Ltd., Kashima, Yodogawa-ku, Osaka, 532, Japan
,
Tsutomu Yasuda Analytical Research Laboratories, Fujisawa Pharmaceutical Co., Ltd., Kashima, Yodogawa-ku, Osaka, 532, Japan
,
Makoto Otsuka Department of Pharmaceutical Technology, Kobe Women's College of Pharmacy, Motoyamakitamachi, Higashinada-ku, Kobe, 658, Japan
&
And Yoshihisa Matsuda Department of Pharmaceutical Technology, Kobe Women's College of Pharmacy, Motoyamakitamachi, Higashinada-ku, Kobe, 658, Japan
Pages 2881-2897 | Published online: 20 Oct 2008

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Naewon Kang, Jangmi Lee, Ji Na Choi, Chen Mao & Eun Hee Lee. (2015) Cryomilling-induced solid dispersion of poor glass forming/poorly water-soluble mefenamic acid with polyvinylpyrrolidone K12. Drug Development and Industrial Pharmacy 41:6, pages 978-988.
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Paola Mura, Maria Teresa Faucci & Pier Luigi Parrini. (2001) Effects of Grinding with Microcrystalline Cellulose and Cyclodextrins on the Ketoprofen Physicochemical Properties. Drug Development and Industrial Pharmacy 27:2, pages 119-128.
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Articles from other publishers (16)

Mingdi Liu, Jichao Liu, Qiuhong Wang, Ping Song, Haichao Li, Songgu Wu & Junbo Gong. (2023) Quantitative analysis of low content polymorphic impurities in canagliflozin tablets by PXRD, NIR, ATR-FITR and Raman solid-state analysis techniques combined with stoichiometry. Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy 293, pages 122458.
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Jin Feng, Changjin Lim, Sihyun Nam, Woojin Yoon, Hoseop Yun, Woo-Sik Kim & Ji-Hun An. (2023) Investigation of Solid-State Hydrate-Anhydrous Phase Transformations of Dabigatran Etexilate Hemi-Edisylate. Crystals 13:3, pages 424.
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Mingdi Liu, Peng Shi, Guangle Wang, Gang Wang, Ping Song, Yumin Liu, Songgu Wu & Junbo Gong. (2021) Quantitative analysis of binary mixtures of entecavir using solid-state analytical techniques with chemometric methods. Arabian Journal of Chemistry 14:10, pages 103360.
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Valmala Bhavana, Rahul B. Chavan, M.K. Chaitanya Mannava, Ashwini Nangia & Nalini R. Shastri. (2019) Quantification of niclosamide polymorphic forms – A comparative study by Raman, NIR and MIR using chemometric techniques. Talanta 199, pages 679-688.
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Peter L.D. Wildfong, Rahul V. Haware, Ting Xu & Kenneth R. Morris. 2018. Pharmaceutical Crystals. Pharmaceutical Crystals 361 426 .
Fumie Kato, Yoshihisa Matsuda & Satoru Watano. (2014) Effect of Grinding on Solid State Stability of Mefenamic Acid Polymorphs. Journal of the Society of Powder Technology, Japan 51:10, pages 678-685.
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Christian Muehlenfeld, Birthe Kann, Maike Windbergs & Markus Thommes. (2013) Solid Dispersions Prepared by Continuous Cogrinding in an Air Jet Mill. Journal of Pharmaceutical Sciences 102:11, pages 4132-4139.
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Lauretta Maggi, Giovanna Bruni, Mariarosa Maietta, Andrea Canobbio, Andrea Cardini & Ubaldo Conte. (2013) II. Technological approaches to improve the dissolution behavior of nateglinide, a lipophilic insoluble drug: Co-milling. International Journal of Pharmaceutics 454:1, pages 568-572.
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Balasubramaniam Jagadish, Rajesh Yelchuri, Bindu K, Hemalatha Tangi, Swetha Maroju & Vinay Umesh Rao. (2010) Enhanced Dissolution and Bioavailability of Raloxifene Hydrochloride by Co-grinding with Different Superdisintegrants. Chemical and Pharmaceutical Bulletin 58:3, pages 293-300.
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Eugene Y. Cheung & Matthew L. Peterson. (2009) Reconciling thermal and structural data from the polymorphic transitions of malonamide. Thermochimica Acta 482:1-2, pages 57-61.
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Sharmistha Datta & David J. W. Grant. (2004) Crystal structures of drugs: advances in determination, prediction and engineering. Nature Reviews Drug Discovery 3:1, pages 42-57.
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Shuichi Yada, Masaoki Ohya, Yuko Ohuchi, Takeshi Hamaura, Naoki Wakiyama, Fusao Usui, Akira Kusai & Keiji Yamamoto. (2003) Solid phase transition of CS-891 enantiotropes during grinding. International Journal of Pharmaceutics 255:1-2, pages 69-79.
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Sanjay Garg, Raghupathi Kandarapu, Kavita Vermani, Kaustubh R. Tambwekar, Alka Garg, Donald P. Waller & Lourens J.D. Zaneveld. (2003) Development Pharmaceutics of Microbicide Formulations. Part I: Preformulation Considerations and Challenges. AIDS Patient Care and STDs 17:1, pages 17-32.
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P Mura, M Cirri, M.T Faucci, J.M Ginès-Dorado & G.P Bettinetti. (2002) Investigation of the effects of grinding and co-grinding on physicochemical properties of glisentide. Journal of Pharmaceutical and Biomedical Analysis 30:2, pages 227-237.
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Kenneth R. Morris, Ulrich J. Griesser, Craig J. Eckhardt & Joseph G. Stowell. (2001) Theoretical approaches to physical transformations of active pharmaceutical ingredients during manufacturing processes. Advanced Drug Delivery Reviews 48:1, pages 91-114.
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. 1999. Industrial Applications of X-Ray Diffraction. Industrial Applications of X-Ray Diffraction 457 467 .

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