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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 26, 2011 - Issue 4
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Original Article

Bifunctional phenolic-choline conjugates as anti-oxidants and acetylcholinesterase inhibitors

Jaroslav ŠebestíkCentro de Química Estrutural, Instituto Superior Técnico, Av. Rovisco Pais 1, 1049-001 Lisboa, Portugal
,
Sérgio M. MarquesCentro de Química Estrutural, Instituto Superior Técnico, Av. Rovisco Pais 1, 1049-001 Lisboa, Portugal
,
Pedro L. Falé
,
Susana SantosCentro de Química e Bioquímica, Faculdade de Ciências da Universidade de Lisboa, Campo Grande, 1749-016 Lisboa, Portugal
,
Daniela M. ArduínoCentro de Neurociências e Biologia Celular, Universidade de Coimbra, 3030 Coimbra, Portugal
,
Sandra M. Cardoso
,
Catarina R. Oliveira
,
M. Luísa M. SerralheiroCentro de Química e Bioquímica, Faculdade de Ciências da Universidade de Lisboa, Campo Grande, 1749-016 Lisboa, Portugal
&
M. Amélia SantosCentro de Química Estrutural, Instituto Superior Técnico, Av. Rovisco Pais 1, 1049-001 Lisboa, PortugalCorrespondence[email protected]
 show all
Pages 485-497 | Received 28 Apr 2010, Accepted 04 Oct 2010, Published online: 11 Nov 2010

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Gaia Fancellu, Karam Chand, Daniel Tomás, Elisabetta Orlandini, Luca Piemontese, Diana F. Silva, Sandra M. Cardoso, Sílvia Chaves & M. Amélia Santos. (2020) Novel tacrine–benzofuran hybrids as potential multi-target drug candidates for the treatment of Alzheimer’s Disease. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 211-226.
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Luca Piemontese, Daniel Tomás, Asha Hiremathad, Vito Capriati, Emanuel Candeias, Sandra M. Cardoso, Sílvia Chaves & M. Amélia Santos. (2018) Donepezil structure-based hybrids as potential multifunctional anti-Alzheimer’s drug candidates. Journal of Enzyme Inhibition and Medicinal Chemistry 33:1, pages 1212-1224.
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Marina Costa, Romane Josselin, Diana F. Silva, Sandra M. Cardoso, Nóra V. May, Sílvia Chaves & M. Amélia Santos. (2020) Donepezil-based hybrids as multifunctional anti-Alzheimer's disease chelating agents: Effect of positional isomerization. Journal of Inorganic Biochemistry 206, pages 111039.
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