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Research Article

Molecular modeling study bioactive natural product of khellin analogues as a novel potential pharmacophore of EGFR inhibitors

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Pages 1171-1181 | Received 07 Jan 2012, Accepted 05 Aug 2012, Published online: 01 Oct 2012

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Raj P. Shah, Priya Wazir, Utpal Nandi & Sonali S. Bharate. (2023) Self‐Emulsifying Drug Delivery of Khellin for Improving Its Oral Bioavailability. ChemistrySelect 8:46.
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N. M. Fawzy, K. M. Ahmed, H. M. Abo-Salem & M. S. Aly. (2022) Novel Furochromone Derivatives of Potential Anticancer Activity Targeting EGFR Tyrosine Kinase. Synthesis and Molecular Docking Study. Russian Journal of Bioorganic Chemistry 48:4, pages 749-767.
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Adli A. Selim, Basma M. Essa, Islam M. Abdelmonem, Mohamed A. Amin & Mona O. Sarhan. (2021) Extraction, purification and radioiodination of Khellin as cancer theranostic agent. Applied Radiation and Isotopes 178, pages 109970.
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Thi Thu Tram Nguyen, Van Anh Le, Pascal Retailleau & Thanh Binh Nguyen. (2019) Access to 2‐Amino‐3‐Arylthiophenes by Base‐Catalyzed Redox Condensation Reaction Between Arylacetonitriles, Chalcones, and Elemental Sulfur. Advanced Synthesis & Catalysis 362:1, pages 160-165.
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Ameen Abu-Hashem. (2018) Synthesis of New Furothiazolo Pyrimido Quinazolinones from Visnagenone or Khellinone and Antimicrobial Activity. Molecules 23:11, pages 2793.
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Rajni Sharma, Ibidapo S. WilliamsLinda GatchieVinay R. SonawaneBhabatosh Chaudhuri & Sandip B. Bharate. (2018) Khellinoflavanone, a Semisynthetic Derivative of Khellin, Overcomes Benzo[ a ]pyrene Toxicity in Human Normal and Cancer Cells That Express CYP1A1 . ACS Omega 3:8, pages 8553-8566.
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Khurshed Bozorov, Li Fei Nie, Jiangyu Zhao & Haji A. Aisa. (2017) 2-Aminothiophene scaffolds: Diverse biological and pharmacological attributes in medicinal chemistry. European Journal of Medicinal Chemistry 140, pages 465-493.
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Ameen A. Abu-Hashem & Mohamed El-Shazly. (2015) Synthesis, reactions and biological activities of furochromones: A review. European Journal of Medicinal Chemistry 90, pages 633-665.
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