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Mateusz Kciuk, Adrianna Gielecińska, Somdutt Mujwar, Mariusz Mojzych, Beata Marciniak, Rafał Drozda & Renata Kontek. (2022) Targeting carbonic anhydrase IX and XII isoforms with small molecule inhibitors and monoclonal antibodies. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 1278-1298.
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Muhammad Umair Amin, Sajid Ali, Muhammad Yasir Ali, Dominik C. Fuhrmann, Imran Tariq, Benjamin S. Seitz, Eduard Preis, Jana Brüßler, Bernhard Brüne & Udo Bakowsky. (2022) Co-delivery of carbonic anhydrase IX inhibitor and doxorubicin as a promising approach to address hypoxia-induced chemoresistance. Drug Delivery 29:1, pages 2072-2085.
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Helga Helseth Hektoen, Anne Hansen Ree, Kathrine Røe Redalen & Kjersti Flatmark. (2016) Sulfamate inhibitor S4 influences carbonic anhydrase IX ectodomain shedding in colorectal carcinoma cells. Journal of Enzyme Inhibition and Medicinal Chemistry 31:5, pages 779-786.
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Claudiu T. Supuran. (2016) Drug interaction considerations in the therapeutic use of carbonic anhydrase inhibitors. Expert Opinion on Drug Metabolism & Toxicology 12:4, pages 423-431.
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Murat Bozdag, Fabrizio Carta, Daniela Vullo, Semra Isik, Zeid AlOthman, Sameh M. Osman, Andrea Scozzafava & Claudiu T. Supuran. (2016) Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase. Journal of Enzyme Inhibition and Medicinal Chemistry 31:1, pages 132-136.
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Namrata Singasane, Prashant S. Kharkar, Mariangela Ceruso, Claudiu T. Supuran & Mrunmayee P. Toraskar. (2015) Inhibition of carbonic anhydrase isoforms I, II, IX and XII with Schiff’s bases incorporating iminoureido moieties. Journal of Enzyme Inhibition and Medicinal Chemistry 30:6, pages 901-907.
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Daniela Vullo, Semra Isik, Murat Bozdag, Fabrizio Carta & Claudiu T. Supuran. (2015) 7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring. Journal of Enzyme Inhibition and Medicinal Chemistry 30:5, pages 773-777.
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Erik O. Pettersen, Peter Ebbesen, Roben G. Gieling, Kaye J. Williams, Ludwig Dubois, Philippe Lambin, Carol Ward, James Meehan, Ian H. Kunkler, Simon P. Langdon, Anne H. Ree, Kjersti Flatmark, Heidi Lyng, Maria J. Calzada, Luis del Peso, Manuel O. Landazuri, Agnes Görlach, Hubert Flamm, Jochen Kieninger, Gerald Urban, Andreas Weltin, Dean C. Singleton, Syed Haider, Francesca M. Buffa, Adrian L. Harris, Andrea Scozzafava, Claudiu T. Supuran, Isabella Moser, Gerhard Jobst, Morten Busk, Kasper Toustrup, Jens Overgaard, Jan Alsner, Jacques Pouyssegur, Johanna Chiche, Nathalie Mazure, Ibtissam Marchiq, Scott Parks, Afshan Ahmed, Margaret Ashcroft, Silvia Pastorekova, Yihai Cao, Kasper M. Rouschop, Brad G. Wouters, Marianne Koritzinsky, Hilda Mujcic & Dan Cojocari. (2015) Targeting tumour hypoxia to prevent cancer metastasis. From biology, biosensing and technology to drug development: the METOXIA consortium. Journal of Enzyme Inhibition and Medicinal Chemistry 30:5, pages 689-721.
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Claudiu T Supuran & Jean-Yves Winum. (2015) Designing carbonic anhydrase inhibitors for the treatment of breast cancer. Expert Opinion on Drug Discovery 10:6, pages 591-597.
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Articles from other publishers (63)
Md. Abu Sufian, Sabina Zamanova, Ahmed M. Shabana, Brianna Kemp, Utpal K. Mondal, Claudiu T. Supuran & Marc A. Ilies. (2023) Expression Dynamics of CA IX Epitope in Cancer Cells under Intermittent Hypoxia Correlates with Extracellular pH Drop and Cell Killing by Ureido-Sulfonamide CA IX Inhibitors. International Journal of Molecular Sciences 24:5, pages 4595.
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Phuong Linh Nguyen, Ahmed Elkamhawy, Young Hee Choi, Chang Hoon Lee, Kyeong Lee & Jungsook Cho. (2022) Suppression of Tumor Growth and Cell Migration by Indole-Based Benzenesulfonamides and Their Synergistic Effects in Combination with Doxorubicin. International Journal of Molecular Sciences 23:17, pages 9903.
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Xiaojuan Wang, Zhixiong Zhang, Zhenzhen Liu, Xiqi Ma, Qi Dai, Xiaoqiang Wang, Baosheng Ge, Hua He & Fang Huang. (2022) Spectroscopic investigation on the binding interactions between graphene quantum dots and carbonic anhydrase. Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy 265, pages 120369.
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Gregory Fishberger, Nicole Natarelli, Dao Le, Deborah Liaw, Afrin Naz, Caroline Ward, Michael Young & Charles Preuss. 2022. Recent Advances in Therapeutic Drug Monitoring and Clinical Toxicology. Recent Advances in Therapeutic Drug Monitoring and Clinical Toxicology
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Stanislav Kalinin, Anna Malkova, Tatiana Sharonova, Vladimir Sharoyko, Alexander Bunev, Claudiu T. Supuran & Mikhail Krasavin. (2021) Carbonic Anhydrase IX Inhibitors as Candidates for Combination Therapy of Solid Tumors. International Journal of Molecular Sciences 22:24, pages 13405.
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Antje Güttler, Yvonne Eiselt, Anne Funtan, Andreas Thiel, Marina Petrenko, Jacqueline Keßler, Iris Thondorf, Reinhard Paschke, Dirk Vordermark & Matthias Bache. (2021) Betulin Sulfonamides as Carbonic Anhydrase Inhibitors and Anticancer Agents in Breast Cancer Cells. International Journal of Molecular Sciences 22:16, pages 8808.
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Holger M. Becker & Joachim W. Deitmer. (2021) Proton Transport in Cancer Cells: The Role of Carbonic Anhydrases. International Journal of Molecular Sciences 22:6, pages 3171.
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Salvador Harguindey, Khalid Alfarouk, Julián Polo Orozco, Stefano Fais & Jesús Devesa. (2020) Towards an Integral Therapeutic Protocol for Breast Cancer Based upon the New H+-Centered Anticancer Paradigm of the Late Post-Warburg Era. International Journal of Molecular Sciences 21:20, pages 7475.
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Salvador Harguindey, Khalid Alfarouk, Julián Polo Orozco, Kévin Hardonnière, Daniel Stanciu, Stefano Fais & Jesús Devesa. (2020) A New and Integral Approach to the Etiopathogenesis and Treatment of Breast Cancer Based upon Its Hydrogen Ion Dynamics. International Journal of Molecular Sciences 21:3, pages 1110.
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Kaye J. Williams & Roben G. Gieling. (2019) Preclinical Evaluation of Ureidosulfamate Carbonic Anhydrase IX/XII Inhibitors in the Treatment of Cancers. International Journal of Molecular Sciences 20:23, pages 6080.
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Ana Podolski-Renić, Jelena Dinić, Tijana Stanković, Mirna Jovanović, Amra Ramović, Aleksandrs Pustenko, Raivis Žalubovskis & Milica Pešić. (2019) Sulfocoumarins, specific carbonic anhydrase IX and XII inhibitors, interact with cancer multidrug resistant phenotype through pH regulation and reverse P-glycoprotein mediated resistance. European Journal of Pharmaceutical Sciences 138, pages 105012.
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Pradipta Das, Michael D. Delost, Munaum H. Qureshi, David T. Smith & Jon T. Njardarson. (2018) A Survey of the Structures of US FDA Approved Combination Drugs. Journal of Medicinal Chemistry 62:9, pages 4265-4311.
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Tanzeela Abdul Fattah, Silvia Bua, Aamer Saeed, Ghulam Shabir & Claudiu T. Supuran. (2019) 3-Aminobenzenesulfonamides incorporating acylthiourea moieties selectively inhibit the tumor-associated carbonic anhydrase isoform IX over the off-target isoforms I, II and IV. Bioorganic Chemistry 82, pages 123-128.
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Claudiu T. Supuran, Vincenzo Alterio, Anna Di Fiore, Katia D’ Ambrosio, Fabrizio Carta, Simona Maria Monti & Giuseppina De Simone. (2018) Inhibition of carbonic anhydrase IX targets primary tumors, metastases, and cancer stem cells: Three for the price of one. Medicinal Research Reviews 38:6, pages 1799-1836.
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Jennifer M. Sahni & Ruth A. Keri. (2018) Targeting bromodomain and extraterminal proteins in breast cancer. Pharmacological Research 129, pages 156-176.
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Khayal Al-Khayal, Ahmed Alafeefy, Mansoor-Ali Vaali-Mohammed, Amer Mahmood, Ahmed Zubaidi, Omar Al-Obeed, Zahid Khan, Maha Abdulla & Rehan Ahmad. (2017) Novel derivative of aminobenzenesulfonamide (3c) induces apoptosis in colorectal cancer cells through ROS generation and inhibits cell migration. BMC Cancer 17:1.
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Srinivas Angapelly, P.V. Sri Ramya, Andrea Angeli, Sonia Del Prete, Clemente Capasso, Mohammed Arifuddin & Claudiu T. Supuran. (2017) Development of sulfonamides incorporating phenylacrylamido functionalities as carbonic anhydrase isoforms I, II, IX and XII inhibitors. Bioorganic & Medicinal Chemistry 25:20, pages 5726-5732.
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Zhuang Hou, Bin Lin, Yu Bao, Hai-ning Yan, Miao Zhang, Xiao-wei Chang, Xin-xin Zhang, Zi-jie Wang, Gao-fei Wei, Mao-sheng Cheng, Yang Liu & Chun Guo. (2017) Dual-tail approach to discovery of novel carbonic anhydrase IX inhibitors by simultaneously matching the hydrophobic and hydrophilic halves of the active site. European Journal of Medicinal Chemistry 132, pages 1-10.
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Fabrizio Carta, Alexander Birkmann, Tamara Pfaff, Helmut Buschmann, Wilfried Schwab, Holger Zimmermann, Alfonso Maresca & Claudiu T. Supuran. (2017) Lead Development of Thiazolylsulfonamides with Carbonic Anhydrase Inhibitory Action. Journal of Medicinal Chemistry 60:7, pages 3154-3164.
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Amal A. Abd-El Fattah, Hebatallah A. Darwish, Nevine Fathy & Samia A. Shouman. (2017) Carbonic anhydrase inhibition boosts the antitumor effects of Imatinib mesylate via potentiating the antiangiogenic and antimetastatic machineries. Toxicology and Applied Pharmacology 316, pages 123-138.
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L L da Motta, I Ledaki, K Purshouse, S Haider, M A De Bastiani, D Baban, M Morotti, G Steers, S Wigfield, E Bridges, J-L Li, S Knapp, D Ebner, F Klamt, A L Harris & A McIntyre. (2016) The BET inhibitor JQ1 selectively impairs tumour response to hypoxia and downregulates CA9 and angiogenesis in triple negative breast cancer. Oncogene 36:1, pages 122-132.
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Murat Bozdag, Ahmed Mahmoud Alafeefy, Abdul Malik Altamimi, Daniela Vullo, Fabrizio Carta & Claudiu T. Supuran. (2017) Coumarins and other fused bicyclic heterocycles with selective tumor-associated carbonic anhydrase isoforms inhibitory activity. Bioorganic & Medicinal Chemistry 25:2, pages 677-683.
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Kamini Marathe, Nevin McVicar, Alex Li, Miranda Bellyou, Susan Meakin & Robert Bartha. (2016) Topiramate induces acute intracellular acidification in glioblastoma. Journal of Neuro-Oncology 130:3, pages 465-472.
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Javad Garousi, Hadis Honarvar, Ken G. Andersson, Bogdan Mitran, Anna Orlova, Jos Buijs, John Löfblom, Fredrik Y. Frejd & Vladimir Tolmachev. (2016) Comparative Evaluation of Affibody Molecules for Radionuclide Imaging of in Vivo Expression of Carbonic Anhydrase IX. Molecular Pharmaceutics 13:11, pages 3676-3687.
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Simon J. A. van Kuijk, Roben G. Gieling, Raymon Niemans, Natasja G. Lieuwes, Rianne Biemans, Brian A. Telfer, Guido R. M. M. Haenen, Ala Yaromina, Philippe Lambin, Ludwig J. Dubois & Kaye J. Williams. (2016) The Sulfamate Small Molecule CAIX Inhibitor S4 Modulates Doxorubicin Efficacy. PLOS ONE 11:8, pages e0161040.
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Nagwa M. Abdel Gawad, Noha H. Amin, Mohammed T. Elsaadi, Fatma M.M. Mohamed, Andrea Angeli, Viviana De Luca, Clemente Capasso & Claudiu T. Supuran. (2016) Synthesis of 4-(thiazol-2-ylamino)-benzenesulfonamides with carbonic anhydrase I, II and IX inhibitory activity and cytotoxic effects against breast cancer cell lines. Bioorganic & Medicinal Chemistry 24:13, pages 3043-3051.
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Daniela Vullo, Mariaconcetta Durante, Francesco Saverio Di Leva, Sandro Cosconati, Emanuela Masini, Andrea Scozzafava, Ettore Novellino, Claudiu T. Supuran & Fabrizio Carta. (2016) Monothiocarbamates Strongly Inhibit Carbonic Anhydrases in Vitro and Possess Intraocular Pressure Lowering Activity in an Animal Model of Glaucoma. Journal of Medicinal Chemistry 59:12, pages 5857-5867.
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Ahmed M. Alafeefy, Fabrizio Carta, Mariangela Ceruso, Abdul-Malek S. Al-Tamimi, Abdulla A. Al-Kahtani & Claudiu T. Supuran. (2016) Development of 3-(4-aminosulphonyl)-phenyl-2-mercapto-3H-quinazolin-4-ones as inhibitors of carbonic anhydrase isoforms involved in tumorigenesis and glaucoma. Bioorganic & Medicinal Chemistry 24:6, pages 1402-1407.
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Carrie L. Lomelino, Brian P. Mahon, Robert McKenna, Fabrizio Carta & Claudiu T. Supuran. (2016) Kinetic and X-ray crystallographic investigations on carbonic anhydrase isoforms I, II, IX and XII of a thioureido analog of SLC-0111. Bioorganic & Medicinal Chemistry 24:5, pages 976-981.
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Ahmed M. Alafeefy, Rehan Ahmad, Maha Abdulla, Wagdy M. Eldehna, Abdul-Malek S. Al-Tamimi, Hatem A. Abdel-Aziz, Omar Al-Obaid, Fabrizio Carta, Abdulla A. Al-Kahtani & Claudiu T. Supuran. (2016) Development of certain new 2-substituted-quinazolin-4-yl-aminobenzenesulfonamide as potential antitumor agents. European Journal of Medicinal Chemistry 109, pages 247-253.
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Elisabetta Barresi, Silvia Salerno, Anna Maria Marini, Sabrina Taliani, Concettina La Motta, Francesca Simorini, Federico Da Settimo, Daniela Vullo & Claudiu T. Supuran. (2016) Sulfonamides incorporating heteropolycyclic scaffolds show potent inhibitory action against carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry 24:4, pages 921-927.
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Benedetta Cornelio, Marie Laronze-Cochard, Mariangela Ceruso, Marta Ferraroni, Graham A. RanceFabrizio Carta, Andrei N. KhlobystovAntonella Fontana, Claudiu T. Supuran & Janos Sapi. (2016) 4-Arylbenzenesulfonamides as Human Carbonic Anhydrase Inhibitors (hCAIs): Synthesis by Pd Nanocatalyst-Mediated Suzuki–Miyaura Reaction, Enzyme Inhibition, and X-ray Crystallographic Studies. Journal of Medicinal Chemistry 59:2, pages 721-732.
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Marta Ferraroni, Fabrizio Carta, Andrea Scozzafava & Claudiu T. Supuran. (2015) Thioxocoumarins Show an Alternative Carbonic Anhydrase Inhibition Mechanism Compared to Coumarins. Journal of Medicinal Chemistry 59:1, pages 462-473.
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Adel S. El-Azab, Alaa A.-M. Abdel-Aziz, Rezk R. Ayyad, Mariangela Ceruso & Claudiu T. Supuran. (2016) Inhibition of carbonic anhydrase isoforms I, II, IV, VII and XII with carboxylates and sulfonamides incorporating phthalimide/phthalic anhydride scaffolds. Bioorganic & Medicinal Chemistry 24:1, pages 20-25.
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Murat Bozdag, Ahmed M. Alafeefy, Daniela Vullo, Fabrizio Carta, Nurcan Dedeoglu, Abdul-Malek S. Al-Tamimi, Nabila A. Al-Jaber, Andrea Scozzafava & Claudiu T. Supuran. (2015) Benzenesulfonamides incorporating bulky aromatic/heterocyclic tails with potent carbonic anhydrase inhibitory activity. Bioorganic & Medicinal Chemistry 23:24, pages 7751-7764.
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Giuseppe La Regina, Antonio Coluccia, Valeria Famiglini, Sveva Pelliccia, Ludovica Monti, Daniela Vullo, Elisa Nuti, Vincenzo Alterio, Giuseppina De Simone, Simona Maria Monti, Peiwen Pan, Seppo Parkkila, Claudiu T. Supuran, Armando Rossello & Romano Silvestri. (2015) Discovery of 1,1′-Biphenyl-4-sulfonamides as a New Class of Potent and Selective Carbonic Anhydrase XIV Inhibitors. Journal of Medicinal Chemistry 58:21, pages 8564-8572.
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Alessio Nocentini, Fabrizio Carta, Mariangela Ceruso, Gianluca Bartolucci & Claudiu T. Supuran. (2015) Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII. Bioorganic & Medicinal Chemistry 23:21, pages 6955-6966.
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İbrahim Esirden, Ramazan Ulus, Burak Aday, Muhammet Tanç, Claudiu T. Supuran & Muharrem Kaya. (2015) Synthesis of novel acridine bis-sulfonamides with effective inhibitory activity against the carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry 23:20, pages 6573-6580.
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Ludwig J. Dubois, Raymon Niemans, Simon J.A. van Kuijk, Kranthi M. Panth, Nanda-Kumar Parvathaneni, Sarah G.J.A. Peeters, Catharina M.L. Zegers, Nicolle H. Rekers, Marike W. van Gisbergen, Rianne Biemans, Natasja G. Lieuwes, Linda Spiegelberg, Ala Yaromina, Jean-Yves Winum, Marc Vooijs & Philippe Lambin. (2015) New ways to image and target tumour hypoxia and its molecular responses. Radiotherapy and Oncology 116:3, pages 352-357.
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Cenzo Congiu, Valentina Onnis, Alessandro Deplano, Gianfranco Balboni, Nurcan Dedeoglu & Claudiu T. Supuran. (2015) Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity. Bioorganic & Medicinal Chemistry Letters 25:18, pages 3850-3853.
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Cenzo Congiu, Valentina Onnis, Alessandro Deplano, Gianfranco Balboni, Mariangela Ceruso & Claudiu T. Supuran. (2015) Synthesis and carbonic anhydrase I, II, IX and XII inhibitory activity of sulfamates incorporating piperazinyl-ureido moieties. Bioorganic & Medicinal Chemistry 23:17, pages 5619-5625.
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Poonam Khloya, Mariangela Ceruso, Sita Ram, Claudiu T. Supuran & Pawan K. Sharma. (2015) Sulfonamide bearing pyrazolylpyrazolines as potent inhibitors of carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry Letters 25:16, pages 3208-3212.
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Diaa A. Ibrahim, Deena S. Lasheen, Maysoun Y. Zaky, Amany W. Ibrahim, Daniela Vullo, Mariangela Ceruso, Claudiu T. Supuran & Dalal A. Abou El Ella. (2015) Design and synthesis of benzothiazole-6-sulfonamides acting as highly potent inhibitors of carbonic anhydrase isoforms I, II, IX and XII. Bioorganic & Medicinal Chemistry 23:15, pages 4989-4999.
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Mariusz Mojzych, Mariangela Ceruso, Anna Bielawska, Krzysztof Bielawski, Emilia Fornal & Claudiu T. Supuran. (2015) New pyrazolo[4,3-e][1,2,4]triazine sulfonamides as carbonic anhydrase inhibitors. Bioorganic & Medicinal Chemistry 23:13, pages 3674-3680.
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Murat Bozdag, Fabrizio Carta, Daniela Vullo, Atilla Akdemir, Semra Isik, Cecilia Lanzi, Andrea Scozzafava, Emanuela Masini & Claudiu T. Supuran. (2015) Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma action. Bioorganic & Medicinal Chemistry 23:10, pages 2368-2376.
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Jaromir Pastorek & Silvia Pastorekova. (2015) Hypoxia-induced carbonic anhydrase IX as a target for cancer therapy: From biology to clinical use. Seminars in Cancer Biology 31, pages 52-64.
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Daniela Vullo, Viviana De Luca, Sonia Del Prete, Vincenzo Carginale, Andrea Scozzafava, Clemente Capasso & Claudiu T. Supuran. (2015) Sulfonamide inhibition studies of the γ-carbonic anhydrase from the Antarctic cyanobacterium Nostoc commune. Bioorganic & Medicinal Chemistry 23:8, pages 1728-1734.
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Fabrizio Carta, Lorenzo Di Cesare Mannelli, Melissa Pinard, Carla Ghelardini, Andrea Scozzafava, Robert McKenna & Claudiu T. Supuran. (2015) A class of sulfonamide carbonic anhydrase inhibitors with neuropathic pain modulating effects. Bioorganic & Medicinal Chemistry 23:8, pages 1828-1840.
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Aiga Grandane, Muhammet Tanc, Raivis Žalubovskis & Claudiu T. Supuran. (2015) Synthesis of 6-aryl-substituted sulfocoumarins and investigation of their carbonic anhydrase inhibitory action. Bioorganic & Medicinal Chemistry 23:7, pages 1430-1436.
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Joanna Kopecka, Ivana Campia, Andrea Jacobs, Andreas P. Frei, Dario Ghigo, Bernd Wollscheid & Chiara Riganti. (2015) Carbonic anhydrase XII is a new therapeutic target to overcome chemoresistance in cancer cells. Oncotarget 6:9, pages 6776-6793.
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Muhammet Tanc, Fabrizio Carta, Andrea Scozzafava & Claudiu T. Supuran. (2015) α-Carbonic Anhydrases Possess Thioesterase Activity. ACS Medicinal Chemistry Letters 6:3, pages 292-295.
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Brian P. Mahon, Alex M. Hendon, Jenna M. Driscoll, Gregory M. Rankin, Sally-Ann Poulsen, Claudiu T. Supuran & Robert McKenna. (2015) Saccharin: A lead compound for structure-based drug design of carbonic anhydrase IX inhibitors. Bioorganic & Medicinal Chemistry 23:4, pages 849-854.
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Daniela Vullo, Sonia Del Prete, Gillian M. Fisher, Katherine T. Andrews, Sally-Ann Poulsen, Clemente Capasso & Claudiu T. Supuran. (2015) Sulfonamide inhibition studies of the η-class carbonic anhydrase from the malaria pathogen Plasmodium falciparum. Bioorganic & Medicinal Chemistry 23:3, pages 526-531.
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Murat Boztaş, Yasin Çetinkaya, Meryem Topal, İlhami Gülçin, Abdullah Menzek, Ertan Şahin, Muhammet Tanc & Claudiu T. Supuran. (2014) Synthesis and Carbonic Anhydrase Isoenzymes I, II, IX, and XII Inhibitory Effects of Dimethoxybromophenol Derivatives Incorporating Cyclopropane Moieties. Journal of Medicinal Chemistry 58:2, pages 640-650.
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Murat Bozdag, Melissa Pinard, Fabrizio Carta, Emanuela Masini, Andrea Scozzafava, Robert McKenna & Claudiu T. Supuran. (2014) A Class of 4-Sulfamoylphenyl-ω-aminoalkyl Ethers with Effective Carbonic Anhydrase Inhibitory Action and Antiglaucoma Effects. Journal of Medicinal Chemistry 57:22, pages 9673-9686.
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Murat Bozdag, Marta Ferraroni, Fabrizio Carta, Daniela Vullo, Laura Lucarini, Elisabetta Orlandini, Armando Rossello, Elisa Nuti, Andrea Scozzafava, Emanuela Masini & Claudiu T. Supuran. (2014) Structural Insights on Carbonic Anhydrase Inhibitory Action, Isoform Selectivity, and Potency of Sulfonamides and Coumarins Incorporating Arylsulfonylureido Groups. Journal of Medicinal Chemistry 57:21, pages 9152-9167.
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Alaa A.-M. Abdel-Aziz, Adel S. El-Azab, Mariangela Ceruso & Claudiu T. Supuran. (2014) Carbonic anhydrase inhibitory activity of sulfonamides and carboxylic acids incorporating cyclic imide scaffolds. Bioorganic & Medicinal Chemistry Letters 24:22, pages 5185-5189.
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Busra Sarikaya, Mariangela Ceruso, Fabrizio Carta & Claudiu T. Supuran. (2014) Inhibition of carbonic anhydrase isoforms I, II, IX and XII with novel Schiff bases: Identification of selective inhibitors for the tumor-associated isoforms over the cytosolic ones. Bioorganic & Medicinal Chemistry 22:21, pages 5883-5890.
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Ahmed M. Alafeefy, Mariangela Ceruso, Abdul-Malek S. Al-Tamimi, Sonia Del Prete, Clemente Capasso & Claudiu T. Supuran. (2014) Quinazoline–sulfonamides with potent inhibitory activity against the α-carbonic anhydrase from Vibrio cholerae. Bioorganic & Medicinal Chemistry 22:19, pages 5133-5140.
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Tineke W. H. Meijer, Johan Bussink, Miriam Zatovicova, Paul N. Span, Jasper Lok, Claudiu T. Supuran & Johannes H. A. M. Kaanders. (2014) Tumor Microenvironmental Changes Induced by the Sulfamate Carbonic Anhydrase IX Inhibitor S4 in a Laryngeal Tumor Model. PLoS ONE 9:9, pages e108068.
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Paul C. McDonald & Shoukat Dedhar. 2014. Carbonic Anhydrase: Mechanism, Regulation, Links to Disease, and Industrial Applications. Carbonic Anhydrase: Mechanism, Regulation, Links to Disease, and Industrial Applications
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Silvia Pastorekova & Claudiu T. Supuran. 2014. Hypoxia and Cancer. Hypoxia and Cancer
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Ludwig Dubois, Sarah G.J.A. Peeters, Simon J.A. van Kuijk, Ala Yaromina, Natasja G. Lieuwes, Ruchi Saraya, Rianne Biemans, Marouan Rami, Nanda Kumar Parvathaneni, Daniela Vullo, Marc Vooijs, Claudiu T. Supuran, Jean-Yves Winum & Philippe Lambin. (2013) Targeting carbonic anhydrase IX by nitroimidazole based sulfamides enhances the therapeutic effect of tumor irradiation: A new concept of dual targeting drugs. Radiotherapy and Oncology 108:3, pages 523-528.
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