Publication Cover
Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 37, 2007 - Issue 2
277
Views
15
CrossRef citations to date
0
Altmetric
Original Articles

Synthesis, Structure, and Biological Activity of Novel 1H‐1,2,4‐Triazol‐1‐yl‐thiazole Derivatives

, , , , &
Pages 199-207 | Received 25 May 2006, Published online: 25 Jul 2007

References

  • Smia , M. S. , Maghray , A. S. , Mohamed , A. R. and Mohamed , A. K. 2000 . Heteroatom Chem. , 11 : 362 – 369 .
  • Bilodeau , M. T. , Balitza , A. E. , Koester , T. J. , Manley , P. J. , Rodman , L. D. , Buser-Doepner , C. , Coll , K. E. , Fernandes , C. , Gibbs , J. B. , Heimbrook , D. C. , Huckle , W. R. , Kohl , N. , Lynch , J. J. , Mao , X. , McFall , R. C. , McLoughlin , D. , Miller-Stein , C. M. , Rickert , K. W. , Sepp-Lorenzino , L. , Shipman , J. M. , Subramanian , R. , Thomas , K. A. , Wong , B. K. , Yu , S. and Hartman , G. D. 2004 . Potent N‐(1,3‐thiazole‐2‐yl)pyridin‐2‐amine vascular endothelial growth factor receptor tyrosine kinase inhibitors with excellent pharmacokinetics and low affinity for the hERG ion channel . J. Med. Chem. , 47 ( 25 ) : 6363 – 6372 .
  • Wang , S. , Meads , C. , Wood , G. , Osnowski , A. , Anderson , S. , Yuill , R. , Thomas , M. , Mwzna , M. , Jackson , W. , Midgley , C. , Griffiths , G. , Fleming , I. , Green , S. , McNae , I. , Wu , S. Y. , Mclnness , C. , Zheleva , D. , Walkinshaw , M. D. and Fischer , P. M. 2004 . 2‐Anilino‐4‐(thiazol‐5‐yl)pyrimidine CDK inhibitors: Synthesis, SAR Analysis, X‐ray crystallography, and biological activity . J. Med. Chem. , 47 ( 7 ) : 1662 – 1675 .
  • Dayan , F. E. , Vincent , A. C. , Romagni , J. G. , Allen , S. N. , Duke , S. O. , Duke , M. V. , Bowling , J. J. and Zjawiony , J. K. 2004 . Amino‐ and urea‐substituted thiazoles inhibit photosynthetic electron transfer . J. Agric. Food Chem. , 48 ( 8 ) : 3689 – 3693 .
  • Miyauchi , H. , Kozuki , K. , Tanio , T. and Ohashi , N. 1995 . Bioorg. Med. Chem. Lett. , 5 ( 14 ) : 1479 – 1482 .
  • Jin , Z. , Huo , A. H. , Li , T. , Hu , Y. , Liu , J. B. and Fang , J. X. 2005 . Synthesis, structures and biological activity research of novel ferrocenyl‐containing 1H‐1,2,4‐triazole derivatives . J. Organomet. Chem. , 690 : 1226 – 1232 .
  • Fang , J. X. , Jin , Z. , Li , Z. M. and Liu , W. 2003 . Preparation, characterization and biological activities of novel ferrocenyl‐substituted azaheterocycle compounds . Appl. Organomet. Chem. , 17 : 145 – 153 .
  • Shao , L. , Hu , Y. , Tao , W. F. , Jin , Z. and Fang , J. X. 2005 . [2‐(4‐Nitophenoxyl)‐2‐(1H‐1,2,4‐triazol‐1‐yl) acetyl]ferrocene . Acta Cryst. E , 61 : m1837 – m1839 .
  • Sakata , M. , Shirakawa , Y. , Kamata , N. , Sakaguchi , Y. , Nishino , H. , Ouyang , J. and Kurosawa , K. 2000 . J. Heterocycl. Chem. , 37 : 269 – 274 .
  • Joshi , K. C. , Pathak , V. N. and Sharma , S. 1985 . Org. Prep. Proc. Int. , 17 : 146
  • Timmler , H. , Krämer , W. , Büchel , K. H. , Kaspers , H. and Brandes , W. US Patent 4 776 877 . 1988 .

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.