Cyclocondensation of Thioamides and Haloacetic Acid Derivatives Provides Only 4-Thiazolidinones; Isomeric 5-Thiazolidinones Were Not observed

REFERENCES

• Lesyk , R. B. ; Zimenkovsky , B. S. 4-Thiazolidones: Centenarian history, current status, and perspectives for modern organic and medicinal chemistry . Curr. Org. Chem. 2004 , 8 , 1547 – 1577 .
   Web of Science ®Google Scholar
• Jain , A. K. ; Vaidya , A. ; Ravichandran , V. ; Kashaw , S. K. ; Agrawal , R. K. Recent developments and biological activities of thiazolidinone derivatives: A review . Bioorg. Med. Chem. 2012 , 20 , 3378 – 3395 .
   PubMed Web of Science ®Google Scholar
• Prabhakar , Y. S. ; Solomon , V. R. ; Gupta , M. K. ; Katti , S. B. QSAR studies on thiazolidines: A biologically privileged scaffold . Top. Heterocycl. Chem. 2006 , 4 , 161 – 249 .
   Google Scholar
• Tomasic , T. ; Masic , L. P. Rhodanine as a privileged scaffold in drug discovery . Curr. Med. Chem. 2009 , 16 , 1596 – 1629 .
   PubMed Web of Science ®Google Scholar
• Lesyk , R. B. ; Zimenkovsky , B. S. ; Kaminskyy , D. V. ; Kryshchyshyn , A. P. ; Havryluk , D. Ya. ; Atamanyuk , D. V. ; Subtel'na , I. Yu. ; Khyluk , D. V. Thiazolidinone motif in anticancer drug discovery: Experience of DH LNMU medicinal chemistry scientific group . Biopolym. Cell. 2011 , 27 , 107 – 117 .
   Web of Science ®Google Scholar
• Kaminskyy , D. V. ; Lesyk , R. B. Structure–anticancer activity relationships among 4-azolidinone-3-carboxylic acids derivatives . Biopolym. Cell. 2010 , 26 , 136 – 145 .
   Google Scholar
• Metwally , M. A. ; Keshk , E. M. ; Fekry , A. ; Etman , H. A. Synthesis of some new thiazolidin-5-one derivatives of pharmaceutical interest . Phosphorus, Sulfur Silicon Relat. Elem. 2004 , 179 , 2067 – 2079 .
   Web of Science ®Google Scholar
• Metwally , M. A. ; Etman , H. A. ; Keshk , E. M. ; Fekry , A. Thiazolidin-5-ones: Synthesis and reactions. Phosphorus, Sulfur Silicon Relat. Elem. 2006, 181, 1039–1058.
   Web of Science ®Google Scholar
• El-Desoky , S. I. ; Bondock , S. B. ; Etman , H. A. ; Fadda , A. A. ; Metwally , M. A. Synthesis of some new thiazole derivatives of pharmaceutical interest . Sulfur Lett. 2003 , 26 , 127 – 135 .
   Google Scholar
• Kaminskyy , D. ; Khyluk , D. ; Vasylenko , O. ; Zaprutko , L. ; Lesyk , R. A facile synthesis and anticancer activity evaluation of spiro[thiazolidinone-isatin] conjugates . Sci. Pharm. 2011 , 79 , 763 – 777 .
   PubMedGoogle Scholar
• Bukowski , L. Some reactions of 2-cyanomethyl-3-3H-imidazol[4,5-b]pyridine with isothiocyanates: Antituberculotic activity of the obtained compounds . Pharmazie 2001 , 56 , 23 – 31 .
   PubMed Web of Science ®Google Scholar
• Grabenko , A. D. ; Kulaeva , L. N. ; Pel'kis , P. S. Substituted arylamides of dithiocarboxylic acids, XIII: Synthesis of 2,3-disubstituted thiazolidin-4-ones . Chem. Heterocyc. Compd. 1970 , 6 , 1513 – 1514 .
   Google Scholar
• Fadda , A. A. ; Bondock , S. ; Rabie , R. ; Etman , H. A. Cyanoacetamide derivatives as synthons in heterocyclic synthesis . Turk. J. Chem. 2008 , 32 , 259 – 286 .
   Web of Science ®Google Scholar
• Khalil , M. ; Berghot , M. A. ; Gouda , M. A. Synthesis and antibacterial activity of some new thiazole and thiophene derivatives . Eur. J. Med. Chem. 2009 , 44 , 4434 – 4440 .
   PubMed Web of Science ®Google Scholar
• Metwally , M. A. ; Khalifa , M. E. ; Attia , E. A. ; Amer , F. A. New arylhydrazonothiazolidin-5-one disperse dyes for dyeing polyester fibers . Pol. J. Chem. Technol. 2010 , 12 , 1 – 6 .
   Web of Science ®Google Scholar
• Dabholkar , V. V. ; Tripathi , D. R. Synthesis and antibacterial activity of isochromene and isoquinoline derivative . J. Heterocycl. Chem. 2011 , 48 , 529 – 532 .
   Web of Science ®Google Scholar
• Mohareb , R. M. ; Sherif , S. M. Heterocyclic synthesis with isothiocyantes: Synthesis of several new polyfunctionally substituted thiophene, 4-thiazoline, and thiazolidinone derivatives . Arch. Pharm. 1991 , 324 , 469 – 471 .
   Web of Science ®Google Scholar
• Hernandez , R. P. ; Rodriguez , J. D. ; De-Armas , H. N. ; Toscano , R. A. Ethyl cyano(4-oxo-3-phenyl-l,3-thiazolidin-2-ylidene)acetate . Acta Cryst. 1996 , C52 , 1731 – 1733 .
   Google Scholar
• Sidwell , R. W. ; Smee , D. F. In vitro and in vivo assay systems for study of influenza virus inhibitors . Antiviral. Res. 2000 , 48 , 1 – 16 .
   PubMed Web of Science ®Google Scholar
• Ram , V. J. ; Haque , N. ; Singh , S. K. ; Nath , M. ; Shoeb , A. Polarized ketene dithioacetals, part II: Synthesis of S,S- and S,N-cyclic ketene to azoles and 1,3-dithiole-2-thiones . Phosphorus, Sulfur Silicon Relat. Elem. 1994 , 88 , 155 – 161 .
   Web of Science ®Google Scholar