Utilization of Chloroagetone in the Synthesis of 3-Methylindoles

References

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• In the few instances where chloroacetone was reported to have been used earlier in the literature, the yields are rather poor (ref. 1, p 166). Dialkylated anilines appeared to be better (ref. 1, p 169)
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• Compound 1 is made by the reductive animation of m-phenetidine with benzaldehyde using NaBH4/phthalic acid
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• Compounds 6 and 7 give spectral data identical to those reported in ref. 6.
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