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- In some cases, most notably 4e and 4f hydrolysis and decarboxylation was accompanied by some scrambling of the bromine. This could be minimized (< 5%) by addition of the bromoketoester to a refluxing solution solution of benzene containing 1 eq. of TsOH or Amberlyst resin
- Rasmussen , C. R. , Press , J. B. , Boyd , R. E. , Scott , M. K. , Reynolds , B. E. , Paragamian , V. , Plampin , J. N. , Hortenstine , J. T. , Gardocki , J. F. , Bennett , D. , Connelly , C. , Martinez , R. , Shupsky , J. , Codd , E. and Raffa , R. B. J. Med. Chem. , manuscript in preparation