95
Views
12
CrossRef citations to date
0
Altmetric
Research Article

Microsphere-based once-daily modified release matrix tablets for oral administration in angina pectoris

, &
Pages 257-266 | Received 19 Apr 2007, Accepted 05 Feb 2008, Published online: 08 Oct 2008

References

  • Amperiadou A, Georgarakis M. Controlled release salbutamol sulphate microcapsules prepared by emulsion solvent-evaporation technique and study on the release affected parameters. Int J Pharm 1995; 115: 1–8
  • Bayomi MA, Al-Suwayeh SA, El-heiw AM, Mesnad AF. Preparation of casein-chitosan microspheres containing diltiazem hydrochloride by an aqueous coacervation technique. Pharm Acta Helv 1998; 73: 187–192
  • Bhalerao SS, Lalla JK, Rane MS. Study of processing parameters influencing the properties of diltiazem hydrochloride microspheres. J Microencapsulation 2001; 18: 299–307
  • Cavallari C, Albertini B, Rodriquez L, Rabasco AM, Fini A. Release of indomethacin from ultrasound dry granules containing lactose-based excipients. J Cont Rel 2005; 102: 39–47
  • Çomoğlu T, Gönül N, Baykara T. The effects of pressure and direct compression on tabletting of microsponges. Int J Pharm 2002; 242: 191–195
  • Das SK, Das NG. Preparation and in vitro dissolution profile of dual polymer (Eudragit®RS100 and RL100) microparticles of diltiazem hydrochloride. J Microencapsulation 1998; 15: 445–452
  • EP. European Pharmacopoeia 5.0. Aubin-France 2005; 233
  • Halder A, Sa B. Preparation and in-vitro evaluation of polystyrene-coated diltiazem-resin complex by oil-in-water emulsion solvent evaporation method. AAPS PharmSciTech 2006; 7: E1–E8
  • Hasçiçek C, Gönül N, Erk N. Mucoadhesive microspheres containing gentamicin sulfate for nasal administration: Preparation and in vitro characterization. Il Farmaco 2003; 58: 11–16
  • Hoffman BB. Therapy of hypertension. The pharmacological basis of therapeutics, 11th ed, Brunton LL, Lazo JS, Parker KL. McGraw-Hill Companies, New York 2006; 845–868
  • Horoz BB, K·l·çarslan M, Yüksel N, Baykara T. Influence of aluminium tristearate and sucrose stearate as the dispersing agents on physical properties and release characteristics of Eudragit RS microspheres. AAPS PharmSciTech 2006; 7: E1–E7
  • Huang H, Ghebre-Sellassie I. Preparation of microspheres of water-soluble pharmaceuticals. J Microencapsulation 1989; 6: 219–225
  • Hutt V, Janik F, Kappler J, Pabst G, Ravelli V, Maccari M, Jaeger H. Evaluation of pharmacokinetics, bioavaliability and dose linearity of diltiazem in healthy volunteers. Arzneimittel-Forschung 1993; 43: 737–743
  • Kakish HF, Tashtoush B, Ibrahim HG, Najib NM. A novel approach for the preparation of highly loaded polymeric controlled release dosage forms of diltiazem HCl and diclofenac sodium. Eur J Pharm Biopharm 2002; 54: 75–81
  • Kawata M, Nakamura M, Goto S, Aoyama T. Preparation and dissolution pattern of Eudragit RS microcapsules containing ketoprofen. Chem Pharm Bull 1986; 34: 2618–2623
  • Kim CK, Kim MJ, Oh KH. Preparation and evaluation of sustained release microspheres of terbutaline sulfate. Int J Pharm 1994; 106: 213–219
  • Kristmundsdóttir T, Gudmundsson ÓS, Ingvarsdóttir K. Release of diltiazem from Eudragit microparticles prepared by spray-drying. Int J Pharm 1996; 137: 159–165
  • Mateovic T, Kriznar B, Bogataj M, Mrhar A. The influence of stirring rate on biopharmaceutical properties of Eudragit RS microspheres. J Microencapsulation 2002; 19: 29–36
  • Michel T. Treatment of myocardial ischemia. The pharmacological basis of therapeutics, 11th ed, Brunton LL, Lazo JS, Parker KL. McGraw-Hill Companies, New York 2006; 823–844
  • Obaidat AA, Obaidat RM. Controlled release of tramadol hydrochloride from matrices prepared using glyceryl behenate. Eur J Pharm Biopharm 2001; 52: 231–235
  • Pather SI, Russell I, Syce JA, Neau SH. Sustained release theophylline tablets by direct compression Part 1: Formulation and in vitro testing. Int J Pharm 1998; 164: 1–10
  • Pignatello R, Consoli P, Puglisi G. In vitro release kinetics of Tolmetin from tabletted Eudragit microparticles. J Microencapsulation 2000; 17: 373–383
  • Reddy KR, Mutalik S, Reddy S. Once-daily sustained release matrix tablets of nicorandil: Formulation and in vitro evaluation. AAPS PharmSciTech 2003; 4: 1–9
  • Schall R, Müller FR, Müller FO, Luus HG. Bioequivalance of controlled-release calcium antagonists. Clin Pharmacokinetics 1997; 32: 75–89
  • Şengel CT, Hasçiçek C, Gönül N. Development and in-vitro evaluation of modified release tablets including ethylcellulose microspheres loaded with diltiazem hydrochloride. J Microencapsulation 2006; 23: 135–152
  • Shimpi S, Chauhan B, Mahadik KR, Paradkar A. Preparation and evaluation of diltiazem HCl-Gelucire 43/01 floating granules prepared by melt granulation. AAPS PharmSciTech 2004; 5: 1–6
  • Sood A, Pachagnula R. Drug release evaluation of diltiazem CR preparations. Int J Pharm 1998; 175: 95–107
  • Souto EB, Mehnert W, Müller RH. Polymorphic behaviour of Compritol®888 ATO as bulk lipid and as SLN and NLC. J Microencapsulation 2006; 23: 417–433
  • Sveinsson SJ, Kristmundsdóttir T, Ingvarsdóttir K. The effect of tableting on the release characteristics of naproxen and ibuprofen microcapsules. Int J Pharm 1993; 92: 29–34
  • Sweetman SC. Cardiovascular drugs. Martindale the complete drug reference, 33rd ed, Sweetman SC. Pharmaceutical Press, Chicago 2002; 874–877
  • USP 24/NF 19. 2000. United States of Pharmacopoeia Convention Inc., RockvilleUSA, 574–575
  • USP 30/NF 25. 2007. United States of Pharmacopoeia Convention Inc., RockvilleUSA, 680–683
  • Zhang YE, Schwartz JB. Effect of diluents on tablet integrity and controlled drug release. Drug Dev Ind Pharm 2000; 26: 761–765

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.