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Research Articles

Enhanced in vitro and ex vivo transdermal permeation of microemulsion gel of tapentadol hydrochloride

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Pages 127-139 | Received 22 Jul 2023, Accepted 12 Feb 2024, Published online: 27 Feb 2024

References

  • Alkilani, A.Z., McCrudden, M.T., and Donnelly, R.F., 2015. Transdermal drug delivery: innovative pharmaceutical developments based on disruption of the barrier properties of the stratum corneum. Pharmaceutics, 7 (4), 438–470. doi: 10.3390/pharmaceutics7040438.
  • Alvi, M.M. and Chatterjee, P.A., 2014. Prospective analysis of co-processed non-ionic surfactants in enhancing permeability of a model hydrophilic drug. AAPS PharmSciTech, 15 (2), 339–353. doi: 10.1208/s12249-013-0065-8.
  • Available from: https://www.accessdata.fda.gov/drugsatfda_docs/label/2021/200533s023lbl.pdf.
  • Available from: https://www.drugs.com/tapentadol.html [Accessed 01 October 2023].
  • Badawy, M.E.I., et al., 2017. Optimization and characterization of the formation of oil-in-water diazinon nanoemulsions: modeling and influence of the oil phase, surfactant and sonication. Journal of environmental science and health. Part. B, pesticides, food contaminants, and agricultural wastes, 52 (12), 896–911. doi: 10.1080/03601234.2017.1362941.
  • Basalious, E.B., Shawky, N., and Badr-Eldin, S.M., 2010. SNEDDS containing bioenhancers for improvement of dissolution and oral absorption of lacidipine. I: development and optimization. International journal of pharmaceutics, 391 (1-2), 203–211. doi: 10.1016/j.ijpharm.2010.03.008.
  • Chien, Y.W., 1992. Novel drug delivery system. 2nd ed., revised and expanded. CRC Press, 302–344.
  • Chien, Y.W., et al., 1990. Facilitated transdermal delivery of therapeutic peptides and proteins by iontophoretic delivery devices. Journal of controlled release, 13 (2-3), 263–278. doi: 10.1016/0168-3659(90)90017-N.
  • Costa, P. and Lobo, J.M.S., 2001. Modeling and comparison of dissolution profiles. European journal of pharmaceutical sciences: official journal of the European federation for pharmaceutical sciences, 13 (2), 123–133. doi: 10.1016/s0928-0987(01)00095-1.
  • Craig, D., 1995. An investigation into the mechanisms of self-emulsification using particle size analysis and low frequency dielectric spectroscopy. International journal of pharmaceutics, 114 (1), 103–110. doi: 10.1016/0378-5173(94)00222-Q.
  • Elias, P.M., 1991. Epidermal barrier function: intercellular lamellar lipid structures, origin, composition and metabolism. Journal of controlled release, 15 (3), 199–208. doi: 10.1016/0168-3659(91)90111-P.
  • Gannu, R., et al., 2010. Enhanced bioavailability of lacidipine via microemulsion based transdermal gels: formulation optimization, ex vivo and in vivo characterization. International journal of pharmaceutics, 388 (1-2), 231–241. doi: 10.1016/j.ijpharm.2009.12.050.
  • Heuschkel, S., Goebel, A., and Neubert, R.H., 2008. Microemulsions–modern colloidal carrier for dermal and transdermal drug delivery. Journal of pharmaceutical sciences, 97 (2), 603–631. doi: 10.1002/jps.20995.
  • Hoar, T.P. and Schulman, J.H., 1943. Transparent water-in-oil dispersions: the oleopathic hydro-micelle. Nature, 152 (3847), 102–103. doi: 10.1038/152102a0.
  • ICH guidelines: stability testing of new drug substances and products Q1A(R2). 2003.
  • Jagdale, S.C., Patil, S., and Kuchekar, B.S., 2013. Application of design of experiment for floating drug delivery of tapentadol hydrochloride. Computational and mathematical methods in medicine, 2013, 625729–625727. doi: 10.1155/2013/625729.
  • Jain, D. and Basniwal, P.K., 2013. Tapentadol, a novel analgesic: review of recent trends in synthesis, related substances, analytical methods. Pharmacodynamics and pharmacokinetics, 51 (2), 283–289. doi: 10.1016/j.bfopcu.2013.04.003.
  • Johannes, K.F., 2013. Chapter 6 – emulsifiers. Hydraulic Fracturing Chemicals and Fluids Technology, Gulf Professional Publishing, 81–88. doi: 10.1016/B978-0-12-411491-3.00006-6.
  • Kantarci, G., et al., 2007. Comparison of different water/oil microemulsions containing diclofenac sodium: Preparation, characterization, release rate, and skin irritation studies. AAPS pharm sci tech, 8 (4), E91.
  • Khurana, S., Jain, N.K., and Bedi, P.M., 2013. Development and characterization of a novel controlled release drug delivery system based on nanostructured lipid carriers gel for meloxicam. Life sciences, 93 (21), 763–772. doi: 10.1016/j.lfs.2013.09.027.
  • Kogan, A., Aserin, A., and Garti, N., 2007. Improved solubilization of carbamazepine and structural transitions in nonionic microemulsions upon aqueous phase dilution. Journal of colloid and interface science, 315 (2), 637–647. doi: 10.1016/j.jcis.2007.06.087.
  • Kogan, A. and Garti, N., 2006. Microemulsions as transdermal drug delivery vehicles. Advances in colloid and interface science, 123-126, 369–385. doi: 10.1016/j.cis.2006.05.014.
  • Mezei, M. and Gulasekharam, V., 1980. Liposomes–a selective drug delivery system for the topical route of administration. Lotion dosage form. Life sciences, 26 (18), 1473–1477. doi: 10.1016/0024-3205(80)90268-4.
  • Mitragotri, S., Blankschtein, D., and Langer, R., 1995. Ultrasound-mediated transdermal protein delivery. Science, 269 (5225), 850–853. doi: 10.1126/science.7638603.
  • Moore, J.W. and Flanner, H.H., 1996. Mathematical comparison of curves with an emphasis on in vitro dissolution profiles. Pharmaceutical technology, 20, 64–74.
  • Morgan, T.M., et al., 1998. Transdermal delivery of estradiol in postmenopausal women with a novel topical aerosol. Journal of pharmaceutical sciences, 87 (10), 1226–1228. doi: 10.1021/js9800275.
  • Pellett, M., et al., 2002. The application of supersaturated systems to percutaneous drug delivery. In: Transdermal drug delivery systems. CRC Press, 320–341.
  • Potts, R.O., and Francoeur, M.L., 1991. The influence of stratum corneum morphology on water permeability. The journal of investigative dermatology, 96 (4), 495–499. doi: 10.1111/1523-1747.ep12470197.
  • Potts, R.O., and Guy, R.H., 1992. Predicting skin permeability. Pharmaceutical research, 9 (5), 663–669. doi: 10.1023/a:1015810312465.
  • Remington, J. P., 2006. Remington: the science and practice of pharmacy. Lippincott Williams & Wilkins.
  • Shukla, T., et al., 2018. Biomedical applications of microemulsion through dermal and transdermal route. Biomedicine & pharmacotherapy = biomedecine & pharmacotherapie, 108, 1477–1494. doi: 10.1016/j.biopha.2018.10.021.
  • Sudhakar, B., Varma, J.N., and Murthy, K.V., 2014. Formulation characterization and ex vivo studies of terbinafine HCl liposomes for cutaneous delivery. Current drug delivery, 11 (4), 521–530. doi: 10.2174/1567201810666140109113830.
  • Tartaro, G., et al., 2020. Microemulsion microstructure(s): a tutorial review. Nanomaterials, 10 (9), 1657. doi: 10.3390/nano10091657.
  • Weaver, J.C., Pliquett, U., and Vaughan, T., 1999. Apparatus and method for electroporation of tissue. Google Patents.
  • W.H.O. Series, 2009. Stability testing of active pharmaceutical ingredients and finished pharmaceutical products, 953, 87–123.
  • Williams, A.C., and Barry, B.W., 2012. Penetration enhancers. Advanced drug delivery reviews, 64, 128–137. doi: 10.1016/j.addr.2012.09.032.
  • Zakaria, M.Y., et al., 2022. Employment of PEGylated ultra-deformable transferosomes for transdermal delivery of tapentadol with boosted bioavailability and analgesic activity in post-surgical pain. International journal of pharmaceutics, 628, 122274. doi: 10.1016/j.ijpharm.2022.122274.

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