Enhanced Percutaneous Permeability of Diclofenac Using a New U-Type Dilutable Microemulsion

REFERENCES

• Alvarez-Figueroa M. J., Blanco-Mendez J. Transdermal delivery of methotrexate: Iontophoretic delivery from hydrogels and passive delivery from microemulsions. Int. J. Pharmaceut. 2001; 215: 57–65
   PubMed Web of Science ®Google Scholar
• Arellano A., Santoyo S., Martin C., Ygartua P. Influence of propylene glycol and isopropyl myristate on the in vitro percuntaneous penetration of diclofenac sodium from Carbopol gels. Europ. J. Pharm. Sci. 1998; 7: 129–135
   Web of Science ®Google Scholar
• Bonina F. P., Puglia C., Barbuzzi T., deCaprariis P., Palagiano F., Rimoli M. G., Saija A. In vitro and in vivo evaluation of polyoxyethylene esters as dermal prodrugs of ketoprofen, naproxen and diclofenac. Europ. J. Pharm. Sci. 2001; 14: 123–134
   PubMed Web of Science ®Google Scholar
• Cabos C., Delord P., Marignan J. C. Local lamellar structure in dense microemulsions. J. Phys. Rev. B. 1988; 37: 9796–9799
   PubMed Web of Science ®Google Scholar
• Chen S.-H., Chang S.-L. Microemulsions. Structure and dynamics of strongly interacting colloids and supra-molecular aggregates in solution, S.-H. Chen, J.S. Huang, P. Tartaglia. Kluwer Academic, DordrechtThe Netherlands 1992; 659–689
   Google Scholar
• Chen S. H., Chang S. L., Strey R., Samseth J., Mortensen K. Structural evolution of bicontinuous microemulsions. J. Phys. Chem. 1991; 95: 7429–7432
   Google Scholar
• Chiu Y. C., Yang W. L. Preparation of vitamin E microemulsion possessing high resistance to oxidation in air. Colloids Surfaces 1992; 63: 311–322
   Web of Science ®Google Scholar
• Delgado-Charro M. B., Iglesias-Vilas G., Blanco-Mendez J., Lopez-Quintela M. A., Marty J.-P., Guy R. H. Delivery of a hydrophilic solute through the skin from novel microemulsion systems. Eur. J. Pharm. Biopharm. 1997; 43: 37–42
   Web of Science ®Google Scholar
• Dreher F., Walde P., Walther P., Wehrli E. Interaction of a lecithin microemulsion gel with human stratum corneum and its effect on transdermal transport. J. Control. Rel. 1997; 45: 131–140
   Web of Science ®Google Scholar
• El-Laithy H. M., El-Shaboury K. M. F. The development of cutina lipogels and gel microemulsion for topical administration of fluconazole. AAPS Pharm. Sci.Tech. 2003; 3, article 35.
   Google Scholar
• Ezrahi S., Wachtel E., Aserin A., Garti N. Structural polymorphism in a four-component nonionic microemulsion. J. Colloid Interface Sci. 1997; 191: 277–290
   PubMed Web of Science ®Google Scholar
• Fini A., Fazio G., Gonzales-Rodriguez M., Cavallari C., Passerini N., Rodriguez L. Formation of ion-pairs in aqueous solutions of diclofenac sodium. Int. J. Pharm. 1999; 187: 163–173
   PubMed Web of Science ®Google Scholar
• Garti N., Aserin A., Ezrahi S., Wachtel E. Water solubilization and chain length compatibility in nonionic microemulsions. J. Colloid Interface Sci. 1995; 169: 428–436
   Web of Science ®Google Scholar
• Gradzielski M., Hoffman H. Rheological properties of microemulsions. Handbook of microemulsion science and technology, P. Kumar, K. L. Mittal. Marcel Dekker, New York 1999; 161–192
   Google Scholar
• Holmberg K. Quarter century progress and new horizons in microemulsions. Micelles, microemulsions, and monolayers, O. Shah. Marcel Dekker, New York 1998; 161–192
   Google Scholar
• Kemken J., Ziegler A., Mueller B. W. Influence of supersaturation on the pharmacodynamic effect of bupranolol after dermal administration using microemulsions as vehicle. Pharm. Res. 1992; 9: 554–558
   PubMed Web of Science ®Google Scholar
• Kreilgaard M. Dermal pharmacokinetics of microemulsion formulations determined by in vitro microdialysis. Pharm. Res. 2001; 18: 367–373
   PubMed Web of Science ®Google Scholar
• Kreilgaard M., Kemme M. J. B., Burggraaf J., Schoemaker R. C., Cohen A. F. Influence of a microemulsion vehicle on cutaneous bioequivalence of a lipophilic model drug assessed by microdialysis and pharmacodynamics. Pharm. Res. 2001; 18: 593–599
   PubMed Web of Science ®Google Scholar
• Kreilgaard M., Pedersen E. J., Jaroszewski J. W. NMR characterization and transdermal drug delivery potential of microemulsion systems. J. Control. Rel. 2000; 69: 421–433
   PubMed Web of Science ®Google Scholar
• Lee P. J., Langer R., Shastri V. P. Novel microemulsion enhancer formulation for simultaneous transdermal delivery of hydrophilic and hydrophobic drugs. Pharm. Res. 2003; 20: 264–269
   PubMed Web of Science ®Google Scholar
• Malmsten M. Microemulsions. Surfactants and polymers in drug delivery, drugs and pharmaceutical sciences, J. Swarbrick. Marcel Dekker, New York 2002; 133–159
   Google Scholar
• Osborne D. W., Ward A. J., O'Neill K. J. Microemulsions as topical drug delivery vehicles: In vitro transdermal studies of a model hydrophilic drug. J. Pharm. Pharmacol. 1991; 43: 450–454
   PubMed Web of Science ®Google Scholar
• Parra J. L., Coderch L., Yuste I., de la Maza A. Incorporation of non-steroidal anti-inflammatory drugs into specific monophasic formulations. Colloids and Surfaces A: Physicochem. Eng. Aspects 1997; 123–124; 114–124
   Google Scholar
• Regev O., Ezrahi S., Aserin A., Garti N., Wachtel E., Kaler E. W., Khan A., Talmon Y. A study of the microstructure of a four-component nonionic microemulsion by Cryo-TEM, NMR, SAXS, and SANS. Langmuir 1996; 12: 668–674
   Web of Science ®Google Scholar
• Rhee Y.-S., Choi J.-G., Park E.-S., Chi S.-C. Transdermal delivery of ketoprofen using microemulsions. Int. J. Pharmaceut. 2001; 228: 161–170
   PubMed Web of Science ®Google Scholar
• Schmalfuss U., Neubert R., Wohlrab W. Modification of drug penetration into human skin using microemulsions. J. Control. Rel. 1997; 46: 279–285
   Web of Science ®Google Scholar
• Schwarz J. S., Weisspapir M. R., Shani A., Amselem S. Enhanced anti-inflammatory activity of diclofenac in jojoba oil submicron emulsion cream. J. Appl. Cosmetol. 1996; 14: 19–24
   Google Scholar
• Shani A. The struggles of jojoba. CHEMTECH 1995; 25: 49–54
   Google Scholar
• Shevachman M., Shani A., Garti N. Formation and Investigation of microemulsions based on jojoba oil and nonionic surfactants. JAOCS 2004; 81: 1143–1152
   Web of Science ®Google Scholar
• Sintov A. C., Shapiro L. New microemulsion vehicle facilitates percutaneous penetration in vitro and cutaneous drug bioavailability in vivo. J. Control Rel. 2004; 95: 173–183
   PubMed Web of Science ®Google Scholar
• Spiclin P., Gasperlin M., Kmetec V. Stability of ascorbyl palmitate in topical microemulsions. 2001; 222: 27–279
   Google Scholar
• Takahashi K., Sakano H., Yoshida M., Numata N., Mizuno N. Characterization of the influence of polyol fatty acid esters on the permeation of diclofenac through rat skin. J. Control. Rel. 2001; 73: 351–358
   PubMed Web of Science ®Google Scholar
• Teubner M., Strey R. Origin of the scattering peak in microemulsions. J. Chem. Phys. 1987; 87: 3195–3200
   Web of Science ®Google Scholar
• Trotta M., Pattarino F., Gasco M. R. Influence of counter ions on the skin permeation of methotrexate from water-oil microemulsions. Pharm. Acta Helv. 1996; 71: 135–140
   PubMedGoogle Scholar
• Walters K. A. Penetration enhancers and their use in transdermal therapeutic systems. Transdermal drug delivery, developmental issues and research initiatives, J. Hadgraft, R. H. Guy. Marcel Dekker, New York and BaselSwitzerland 1989; 197–246
   Google Scholar
• Wisniak J. Chemistry and technology of jojoba oil: State of the art. Proceedings of the 6th International Conference on Jojoba and Its Uses, J. Wisniak, J. Zabick. Ben-Gurion University of the Negev, Beer-ShevaIsrael 1985; 311–321
   Google Scholar