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Research Articles

Comparative binder efficiency modeling of dry granulation binders using roller compaction

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Pages 574-583 | Received 06 Jun 2016, Accepted 11 Dec 2016, Published online: 05 Jan 2017

References

  • Singh R, Ierapetritou M, Ramachandran R. An engineering study on the enhanced control and operation of continuous manufacturing of pharmaceutical tablets via roller compaction. Int J Pharm 2012;438:307–26.
  • FDA. 2016. Available from: http://www.fda.gov/downloads/Drugs/…/Guidances/ucm073507.pdf [last accessed on 02/15/2016].
  • Teng Y, Qiu Z, Wen H. Systematical approach of formulation and process development using roller compaction. Eur J Pharm Biopharm 2009;73:219–29.
  • Nachaegari N, Bansal AK. Coprocessed excipients for solid dosage forms. Pharm Technol 2004;52–64.
  • FMC-Biopolymers. 2016. Available from: http://www.fmcbiopolymer.com/Portals/Pharm/Content/Docs/Avicel%20DG%20Brochure%2012-4-09.pdf [last accessed on 02/11/2016].
  • Ali S, Langley N. Dry granulation simplifies tableting process. PFQ Pharm Formulat Qual 2010;12(2).
  • Kleinebudde P. Roll compaction/dry granulation: pharmaceutical applications. Eur J Pharm Biopharm 2004;58:317–26.
  • Gerteis. 2016. Available from: http://www.gerteis.com/_files/data/Gerteis_Mini_Pactor_Web_en.pdf [last accessed on 02/24/2016].
  • USP38-NF33. 2016. Powder flow. United States Pharmacopoeia, USP-NF online <1174>, USP 38-NF33, pp. 1326-1330, [last accessed on 02/10/2016].
  • USP38-NF33. 2016. Bulk density and tapped density of powders. United States Pharamacopoeia, USP-NF online <616>. USP38-NF33, pp.-420.
  • USP38-NF33. 2016. Tablet friability. United States Pharamacopoeia, USP-NF online <1216>. USP38-NF33, pp. 1432.
  • USP38-NF33. 2016. Tablet breaking force. United States Pharamacopoeia, USP-NF online <1217>. USP38-NF33, pp. 1433.
  • USP38-NF33. 2016. Disintegration. United States Pharamacopoeia, USP-NF online <701>. USP38-NF33, pp.-483.
  • Martens H, Martens M. Modified Jack-knife estimation of parameters uncertainity in bilinear mo deling by partial least square regression (PLSR). Food Qual Prefer 2000;11:5–16.
  • Esbensen K, Schoenkopf T, Midtgaard D, Guyot D. Multivariate data analysis. Trondheim, Norway: CAMO ASA; 2012.
  • Kolter K, Flick D. Structure and dry binding activity of different polymers, including Kollidon® VA 64. Drug Dev Ind Pharm 2000;26:1159–65.
  • Haware RV, Shivagari R, Johnson PR, et al. Application of multivariate methods to evaluate the functionality of bovine- and vegetable-derived magnesium stearate. J Pharm Sci 2014;103:1466–77.
  • Haware RV, Kancharla JP, Udupa AK, et al. Physico-mechanical properties of coprocessed excipient MicroceLac® 100 by DM3 approach. Pharm Res 2015;32:3618–35.
  • Haware RV, Dave VS, Kakarala B, et al. Vegetable-derived magnesium stearate functionality evaluation by DM3 approach. Eur J Pharm Sci 2016;89:115–24.
  • Gereg GW, Cappola ML. Roller compaction feasibility for new drug candidates: laboratory to production scale. Pharm Technol N Am 2002;(Suppl.)8:20–3.
  • Furhrer C. Lab Pharm Problem Technol 1977;269:759.
  • Karehill PG, Glazer M, Nyström C. Studies on direct compression of tablets. XXIII. The importance of surface roughness for the compactability of some directly compressible materials with different bonding and volume reduction properties. Int J Pharm 1990;64:35–43.
  • Inghelbrecht S, Remon JP. Roller compaction and tableting of microcrystalline cellulose/drug mixtures. Int J Pharm 1998;161:215–24.
  • Gupta A, Peck GE, Miller RW, Morris KR. Effect of the variation in the ambient moisture on the compaction behavior of powder undergoing roller-compaction and on the characteristics of tablets produced from the post-milled granules. J Pharm Sci 2005;94:2314–26.
  • Roberts RJ, Rowe RC. The effect of punch velocity on the compaction of a variety of materials. J Pharm Pharmacol 1985;37:377–84.
  • Malkowska S, Khan KA. Effect of re-conpression on the properties of tablets prepared by dry granulation. Drug Dev Ind Pharm 1983;9:331–47.
  • Riepma KA, Vromans H, Zuurman K, Lerk CF. The effect of dry granulation on the consolidation and compaction of crystalline lactose. Int J Pharm 1993;97:29–38.
  • Kochhar SK, Rubinstein MH, Barnes D. The effects of slugging and recompression on pharmaceutical excipients. Int J Pharm 1995;115:35–43.

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