Preparation and evaluation of posaconazole-loaded enteric microparticles in rats

References

• Courtney R, Pai S, Laughlin M, et al. Pharmacokinetics, safety, and tolerability of oral posaconazole administered in single and multiple doses in healthy adults. Antimicrob Agents Chemother 2003;47:2788–95.
   PubMed Web of Science ®Google Scholar
• Nomeir AA, Pramanik BN, Heimark L, et al. Posaconazole (Noxafil, SCH 56592), a new azole antifungal drug, was a discovery based on the isolation and mass spectral characterization of a circulating metabolite of an earlier lead (SCH 51048). J Mass Spectrom 2008;43:509–17.
   PubMed Web of Science ®Google Scholar
• Oakley KL, Moore CB, Denning DW. In vitro activity of SCH-56592 and comparison with activities of amphotericin B and itraconazole against Aspergillus spp. Antimicrob Agents Chemother 1997;41:1124–6.
   PubMed Web of Science ®Google Scholar
• Walravens J, Brouwers J, Spriet I, et al. Effect of pH and comedication on gastrointestinal absorption of posaconazole: monitoring of intraluminal and plasma drug concentrations. Clin Pharmacokinet 2011;50:725–34.
   PubMed Web of Science ®Google Scholar
• Varum FJO, Hatton GB, Basit AW. Food, physiology and drug delivery. Int J Pharm 2013;457:446–60.
   PubMed Web of Science ®Google Scholar
• Ozturk A, Ozturk SS, Palsson B, et al. Mechanism of release from pellets coated with an ethylcellulose-based film. J Control Release 1990;14:203–13.
   Web of Science ®Google Scholar
• Wu X, Eshun G, Zhou Y. Effect of interparticulate interaction on release kinetics of microsphere ensembles. J Pharm Sci 1998;87:586–93.
   PubMed Web of Science ®Google Scholar
• Davis SS. Microspheres and drug therapy: pharmaceutical, immunological, and medical aspects. USA and Canada: Elsevier Publishing Company; 1984.
   Google Scholar
• Vodak DT, Morgen M. Design and development of HPMCAS-based spray-dried dispersions, amorphous solid dispersions. New York: Springer; 2014.
   Google Scholar
• Obara S, Tanno FK, Sarode A. Properties and applications of hypromellose acetate succinate (HPMCAS) for solubility enhancement using melt extrusion. In: Melt extrusion. New York: Springer; 2013.
   Google Scholar
• Curatolo W, Nightingale JA, Herbig SM. Utility of hydroxypropylmethylcellulose acetate succinate (HPMCAS) for initiation and maintenance of drug supersaturation in the GI milieu. Pharm Res 2009;26:1419–31.
   PubMed Web of Science ®Google Scholar
• Dobry DE, Settell DM, Baumann JM, et al. A model-based methodology for spray-drying process development. J Pharm Innov 2009;4:133–42.
   PubMed Web of Science ®Google Scholar
• Arifin DY, Lee LY, Wang CH. Mathematical modeling and simulation of drug release from microspheres: implications to drug delivery systems. Adv Drug Deliv Rev 2006;58:1274–325.
   PubMed Web of Science ®Google Scholar
• Zhu G, Mallery SR, Schwendeman SP. Stabilization of proteins encapsulated in injectable poly (lactide-co-glycolide). Nat Biotechnol 2000;18:52–7.
   PubMed Web of Science ®Google Scholar
• Kang J, Schwendeman SP. Pore closing and opening in biodegradable polymers and their effect on the controlled release of proteins. Mol Pharm 2007;4:104–18.
   PubMed Web of Science ®Google Scholar
• Klose D, Siepmann F, Willart JF, et al. Drug release from PLGA-based microparticles: effects of the “microparticle: bulk fluid” ratio. Int J Pharm 2010;383:123–31.
   PubMed Web of Science ®Google Scholar
• Klose D, Delplace C, Siepmann J. Unintended potential impact of perfect sink conditions on PLGA degradation in microparticles. Int J Pharm 2011;404:75–82.
   PubMed Web of Science ®Google Scholar
• Streubel A, Peppas NBR, Siepmann J. Bimodal drug release achieved with multi-layer matrix tablets: transport mechanisms and device design. J Control Release 2000;69:455–68.
   PubMed Web of Science ®Google Scholar
• Baldursdóttir SG, Kjøniksen AL, Karlsen J, et al. Riboflavin-photosensitized changes in aqueous solutions of alginate. Rheological studies. Biomacromolecules 2003;4:429–36.
   PubMed Web of Science ®Google Scholar
• Elias HG. An introduction to polymer science. Ann Chim Sci Matér 1999;24:402–3.
   Google Scholar
• Bohr A, Yang M, Baldursdóttir S, et al. Particle formation and characteristics of celecoxib-loaded poly(lactic-co-glycolic acid) microparticles prepared in different solvents using electrospraying. Polymer 2012;53:3220–9.
   Web of Science ®Google Scholar
• Son WK, Youk JH, Lee TS, Park WH. The effects of solution properties and polyelectrolyte on electrospinning of ultrafine poly(ethylene oxide) fibers. Polymer 2004;45:2959–66.
   Web of Science ®Google Scholar
• Antoniou E, Alexandridis P. Polymer conformation in mixed aqueous-polar organic solvents. Eur Polym J 2010;46:324–35.
   Web of Science ®Google Scholar
• Wang J, Wang BM, Schwendeman SP. Characterization of the initial burst release of a model peptide from poly(D,L-lactide-co-glycolide) microspheres. J Control Release 2002;82:289–307.
   PubMed Web of Science ®Google Scholar
• Schwartz JB, Simonelli AP, Higuchi WI. Drug release from wax matrices. I. Analysis of data with first-order kinetics and with the diffusion-controlled model. J Pharm Sci 1968;57:274–7.
   PubMed Web of Science ®Google Scholar
• Nomeir AA, Kumari P, Hilbert MJ, et al. Pharmacokinetics of SCH 56592, a new azole broad-spectrum antifungal agent, in mice, rats, rabbits, dogs, and cynomolgus monkeys. Antimicrob Agents Chemother 2000;44:727–31.
   PubMed Web of Science ®Google Scholar
• Hartman RPA, Brunner D, Camelot D, et al. Electrohydrodynamic atomization in the cone–jet mode physical modeling of the liquid cone and jet. J Aerosol Sci 1999;30:823–49.
   Web of Science ®Google Scholar
• Tran PH, Tran TT, Piao ZZ, et al. Physical properties and in vivo bioavailability in human volunteers of isradipine using controlled release matrix tablet containing self-emulsifying solid dispersion. Int J Pharm 2013;450:79–86.
   PubMed Web of Science ®Google Scholar
• Litvinov V. EPDM/PP thermoplastic vulcanizates as studied by proton NMR relaxation: phase composition, molecular mobility, network structure in the rubbery phase, and network heterogeneity. Macromolecules 2006;39:8727–41.
   Web of Science ®Google Scholar
• Antoniou E, Buitrago CF, Tsianou M, Alexandridis P. Solvent effects on polysaccharide conformation. Carbohydr Polym 2010;79:380–90.
   Web of Science ®Google Scholar
• Wan F, Wu JX, Bohr A, et al. Impact of PLGA molecular behavior in the feed solution on the drug release kinetics of spray dried microparticles. Polymer 2013;54:5920–7.
   Web of Science ®Google Scholar
• Fredenberg S, Wahlgren M, Reslow M, Axelsson A. The mechanisms of drug release in poly(lactic-co-glycolic acid)-based drug delivery systems – a review. Int J Pharm 2011;415:34–52.
   PubMed Web of Science ®Google Scholar