264
Views
11
CrossRef citations to date
0
Altmetric
Research Article

Co-crystallization for enhanced dissolution rate of bicalutamide: preparation and evaluation of rapidly disintegrating tablets

, , &
Pages 1215-1223 | Received 25 Sep 2018, Accepted 01 Dec 2018, Published online: 27 May 2019

References

  • Rajbhar P, Gautam SS, Prasad RK, et al. Co-crystals formation of clarithromycin with urea: An efficient approach to enhance the solubility and dissolution rate. AJADD. 2016;4:12–20.
  • Michael D, Feng L, Charles BD, et al. Micellar delivery of bicalutamide and embelin for treating prostate cancer. Pharm Res. 2009;26:2081–2092.
  • Meer T, Fule R, Khanna D, et al. Solubility modulation of bicalutamide using porous silica. J Pharm Investig. 2013;43:279–285.
  • Srikanth MV, Murali Mohan Babu GV, Sreenivasa Rao N, et al. Dissolution rate enhancement of poorly soluble bicalutamide using β-cyclodextrin inclusion complexation. Int J Pharm Pharm Sci. 2010;2:191–198.
  • Narkhede KB, Laware RB, Sharma YB, et al. Enhancement of solubility of bicalutamide using solid dispersion technique. Int J Pharm Sci. 2012;3:2739–2748.
  • Meer TS, Sawant KP, Amin PD. Liquid antisolvent precipitation process for solubility modulation of bicalutamide. Acta Pharm. 2011;61:435–445.
  • Patel RP, Bhavsar VA. Studies in development of bicalutamide nano formulations. Eur J Biomed Pharm Sci. 2016;3:281–287.
  • Pankaj P, Kailash B, Rao RT, et al. Micronization: an efficient tool for dissolution enhancement of dienogest. Int J Drug Dev Res. 2011;3:329–333.
  • Srikanth MV, Ram BJ, Rajan DS, et al. Dissolution rate enhancement of bicalutamide by adsorption process. Afr J Pharm Pharmacol. 2013;7:1357–1362.
  • El Maghraby GM, Elsergany RN. Fast disintegrating tablets of nisoldipine for intra-oral administration. Pharm Dev Technol. 2014;19:641–650.
  • El-Gizawy SA, Osman MA, Arafa MF, et al. Aerosil as a novel co-crystal co-former for improving the dissolution rate of hydrochlorothiazide. Int J Pharm. 2015;478:773–778.
  • Nalte YK, Arsul VA, Shep SG, et al. Solubility enhancement of nevirapine by co-crystallisation technique. J Pharm Res. 2015;9:556–561.
  • Budiman A, Nurlatifah E, Amin S. Enhancement of solubility and dissolution rate of glibenclamide by co crystal approach and solvent drop grinding method. Int J Curr Pharm Rev Res. 2016;7:248–250.
  • Tile MK, Pawar AY. Solubility and dissolution rate enhancement of olmesartan medoxomil by chitosan based co crystal approach. Int J Pharm Bio Sci. 2015;5:400–411.
  • Arafa MF, El-Gizawy SA, Osman MA, et al. Co-crystallization for enhanced dissolution rate of nateglinide: In vitro and in vivo evaluation. J Drug Deliv Sci Technol. 2017;38:9–17.
  • Arafa MF, El-Gizawy SA, Osman MA, et al. Xylitol as a potential co-crystal co-former for enhancing dissolution rate of felodipine: preparation and evaluation of sublingual tablets. Pharm Dev Technol. 2018;23:454–463.
  • Dengale SJ, Grohganz H, Rades T, et al. Recent advances in co-amorphous drug formulations. Adv Drug Deliv Rev. 2016;100:116–125.
  • Arafa MF, El-Gizawy SA, Osman MA, et al. Sucralose as co-crystal co-former for hydrochlorothiazide: development of oral disintegrating tablets. Drug DevInd Pharm. 2016;42:1225–1233.
  • Khan KA. The concept of dissolution efficiency. J Pharm Pharmacol. 1975;27:48–49.
  • Kour P, Kataria MK, Bilandi A. Dissolution rate enhancement of pioglitazone by solid dispersion technique. IAJPR. 2015;5:2664–2681.
  • United States Pharmacopiae National Formulary 24. Rockville (MD): United States Pharmacopial Convention; 2000.
  • Jain CP, Naruka PS. Formulation and evaluation of fast dissolving tablets of valsartan. Int J Pharm and Pharm Sci. 2009;1:219–226.
  • Patil A, Pore Y, Kuchekar B. Effect of l-Arginine on bicalutamide complexation with hydroxyl propyl-β-cyclodextrin. Dig J NanomaterBio. 2008;3:89–98.
  • Li C, Li C, Le Y, et al. Formation of bicalutamide nanodispersion for dissolution rate enhancement. Int J Pharm. 2011;404:257–263.
  • Vega DR, Polla G, Martinez A, et al. Conformational polymorphism in bicalutamide. Int J Pharm. 2007;328:112–118.
  • Le Y, Ji H, Chen JF, et al. Nanosized bicalutamide and its molecular structure in solvents. Int J Pharm. 2009;370:175–180.
  • Srikanth MV, Muralimohan babu GV, Sunil SA, et al. Studies on the effect of hydrophilic carriers in the dissolution rate enhancement of poorly soluble drug, bicalutamide. Res J Pharm Tech. 2010;3:1–4.
  • Basavoju S, Boström D, Velaga SP. Indomethacin-saccharin cocrystal: design, synthesis and preliminary pharmaceutical characterization. Pharm Res. 2008;25:530–541.
  • Goud NR, Gangavaram S, Suresh K, et al. Novel furosemide cocrystals and selection of high solubility drug forms. J Pharm Sci. 2012;101:664–680.
  • Shiraki K, Takata N, Takano R, et al. Dissolution improvement and the mechanism of the improvement from cocrystallization of poorly water-soluble compounds. Pharm Res. 2008;25:2581–2592.
  • U.S. Department of Health and Human Services Food and Drug Administration Center for Drug Evaluation and Research (CDER). Guidance for industry orally disintegrating tablets – cder data standards manual. Chemistry. 2008;12:1–3.
  • Mannur VS, Karki SS, Ramani KB. Formulation and characterization of ranitidine hydrochloride fast disintegrating tablets. Int J Chem Tech Res. 2010;2:1163–1169.
  • Mohite BP, Chafle SA, Somasundaram J, et al. Development and evaluation of ofloxacin orally disintegrating tablets. Braz J Pharm Sci. 2012;48:217–225.
  • Balata GF, Zidan AS, Abourehab MAS, et al. Rapid disintegrating tablets of simvastatin dispersions in polyoxyethylene–polypropylene block copolymer for maximized disintegration and dissolution. Drug Des Devel Ther. 2016;10:3211–3223.
  • Essa EA, Elmarakby AO, Donia AM, et al. Controlled precipitation for enhanced dissolution rate of flurbiprofen: development of rapidly disintegrating tablets. Drug Dev Ind Pharm. 2017;43:1430–1439.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.