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Research Article

Preparation, Relative Toxicity, Chemotherapeutic Activity, and Pharmacokinetics of Liposomal SJA-95: A New Polyene Macrolide Antibiotic

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Pages 279-292 | Published online: 09 Dec 2008

References

  • A. Adedoyin, C. E. Swenson, A. Hellmann, D. Radowska, G. Horwith, A. S. Janoff, and et al (2000). A pharmacokinetic study of amphotericin-B lipid complex injection (Abelcet) in patients with definite or probable systemic fungal infections. Antimicrob. Ag. Chemother. 44 (10):2900–2902.
  • T. M. Allen. (1997). Liposomes: opportunities in drug delivery. Drugs 54:8–14.
  • T. M. Allen, and C. Hanson. (1991). Pharmacokinetics of stealth versus conventional liposomes: effect of dose. Biochem. Biophys. Acta. 1068 (2):133–141.
  • L. Berestein. (1989). Liposomes in infectious diseases: present and future. Curr. Clin. Top. Infect. Dis. 10:241–253.
  • K. K. Chakraborty, and S. R. Naik. (2000). In situ liposomal preparation containing amphotericin B: related toxicity and tissue diposition studies. Pharm. Dev. Tech. 5:543–553.
  • K. K. Chakraborty, and S. R. Naik. (2001). Pharmacokinetic studies of in situ liposomal preparation containing amphotericin B complex with different chemically modified β-cyclodextrins. J. Lip. Res. 11 (1):1–14.
  • K. K. Chakraborty, and S. R. Naik. (2003). Therapeutic and hemolytic evaluation of in situ liposomal preparation containing amphotericin B complexed with different chemically modified β-cyclodextrins. J. Pharm. Pharmceut. Sci. 6 (2):231–237.
  • S. K. Desai, and S. R. Naik. (2008). Probable mechanism(s) of antifungal activity of SJA-95, a heptaene polyene antibiotic. Ind. J. Pharm. Sci. 270:165–169.
  • R. D. Diamond. (1988). Fungal surfaces: effects of interactions with phagocytic cells. Rev. Infect. Dis. 2:428–431.
  • M. A. Dietrich. (2004). New advances in fungal pharmacotherapy: voriconazole and caspofungin Inet Ce 221–146–04–069–H01. http://www.Inetce.com(pdf).
  • M. Gibaldi. (2005). Compartmental and noncompartmental pharmacokinetics. In: Biopharmaceutics and Clinical Pharmacokinetics, 4th ed. Hyderabad, India: Pharma Book Syndicate, pp 14–23.
  • J. Harindran, K. K. Chakraborty, and S. R. Naik. (1999). Preparation, relative toxicity, and therapeutic efficacy in mice and rats of liposomal HA–1–92 (a new oxohexaene polyene macrolide antibiotic). J. Pharm. Pharmacol. 51:771–776.
  • D. J. Hoban, G. G. Zhanel, and J. A. Karlowsky. (1999). In vitro susceptibilities of Candida and Cryptococcus neoformans from blood cultures and neutropenic patients. Antimicrob. Ag. Chemother. 43 (6):1463–1464.
  • V. L. Kan, J. E. Bennett, M. A. Amantea, M. C. Smolkis, E. McManus, and D. M. Grasela. (1991). Comparative safety, tolerance, and pharmacokinetics of amphotericin B lipid complex and amphotericin B deoxycholate in healthy male volunteers. J. Infect. Dis. 164:408–412.
  • V. E. Khutorsky. (1992). Structure of amphotericin B–cholesterol complex. Biochim. Biophys. Acta. 1108:123–127.
  • J. W. Lee, M. A. Amantea, P. A. Franchis, E. E. Navarro, J. Bacher, P. A. Pizzo, and et al (1994). Pharmacokinetics and safety of a unilamellar liposomal formulation of amphotericin B (Ambisome) in rabbits. Antimicrob. Ag. Chemother. 38 (4):713–718.
  • R. I. Leher. (1966). Antifungal effects of peroxidase systems. J. Bacteriol. 99:361–365.
  • J. T. Litchfield, and F. A. WilcoxonJr.. (1949). Simplified method of evaluating dose effects experiments. J. Pharmacol. Exp. Ther. 96:99–113.
  • S. de Marie, R. Janknegt, and I. A. J. M. Bakker-Woudenberg. (1994). Clinical use of liposomal and lipid-complexed amphotericin B. J. Antimicrob. Chem. 33:907–916.
  • B. McCormack, and B. Gregoriadis. (1996). Comparative Studies of the fate of free and liposome-entrapped hydroxypropyl-β-cyclodextrin/drug complexes after intravenous injection into rats: implications in drug delivery. Biochem. Biophys. Acta. 1291:237–244.
  • S. R. Naik, S. K. Desai, R. K. Nanda, and M. S. Narayanan. (2007). Fermentation, isolation, purification, and biological activity of SJA-95, a heptaene polyene macrolide antibiotic produced by Streptomyces sp. strain S-24. Arzneimittel-Forschung Drug Res. 57 (3):171–179.
  • L. E. Nicolle, C. Rotstein, A. M. Bourgault, G. St. Germain, and G. Garber. (1998). The Canadian Infections Invasive Fungal Registry. Invasive fungal infections in Canada from 1992 to 1994. Can. J. Infect. Dis. 9:347–352.
  • S. Perrett, M. Golding, and W. P. Willians. (1991). A simple method for the preparation of liposomes for pharmaceutical application: characterization of the liposomes. J. Pharm. Pharmacol. 43:154–161.
  • R. P. Rapp, P. O. Gubbuns, and M. E. Evans. (1997). Amphotericin B lipid complex. Ann. Pharmacother. 31:1174–1186.
  • K. Richardson, K. W. Brammer, M. S. Marriott, and P. F. Troke. (1985). Activity of UK-49, 858, a bis-triazole derivative, against experimental infections with Candida albicans and Trichophyton mentagrophytes. Antimicrob. Agents Chemother. 27:832–835.
  • J. H. Senior. (1987). Fate and behaviour of liposomes in vivo: a review of controlling factors. CRC Crit. Rev.Ther. Drug Car. Sys. 3:123–193.
  • K. L. Therese, R. Bagyalakshmi, H. N. Madhavan, and P. Deepa. (2006). In vitro susceptibility testing by agar dilution method to determine the minimum inhibitory concentrations of amphotericin B, fluconazole, and ketoconazole against ocular fungal isolates. Ind. J. Microbiol. 24 (4):273–279.
  • A. K. Uppadhyay, S. K. Jain, and V. K. Dixit. (1997). Long circulation liposomes: an overview. Ind. Drugs 34 (9):483–487.

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