References
- Allan HR, Robert FB. Purification and properties of trans-N-deoxyribosylase. J Biol Chem 1958; 238: 261–266
- Beach JW, Kim HO, Jeong LS. A highly stereoselective synthesis of anti-HIV 2′, 3′-dideoxy-and 2′, 3′-didehydro-2′3′-dideoxynucleosides. J Org Chem 1992; 57: 3887–3894
- Betbeder D, Hutchinson DW, Richards AO. The stereoselective enzymatic synthesis of 9-beta-D-2′-deoxyribofuranosyl 1-deazapurine. Nucleic Acids Res 1989; 17: 4217–22
- Cardinaud R. Nucleoside deoxyribosyltransferase from Lactobacillus helveticus. Meth Enzymol 1978; 51: 446–455
- Carson DA, Wasson DB. Synthesis of 2′,3′-dideoxynucleosides by enzymatic trans-glycosylation. Biochem Biophys Res Commun 1988; 155: 829–834
- Chen SH, Lin S, King I. Synthesis and comparative evaluation of two antiviral agents: β-L-Fd4C and β-D-fd4C. Bioorg Med Chem Lett 1998; 8: 3245–3250
- Chu, CK. 1995. Method for the preparation of 2′,3′-dideoxy and 2′,3′-dideoxy-didehydro nucleoside. USP 5,455,339. (USP in full).
- Hammond, J, Schinazi, R, Schlueter-Wirtz, S. Mellors, J. 1999. Novel mutations in HIV-1 reverse transcriptase selected for by 2′,3′-dideoxy-2′,3′-didehydro-5-fluorocytidine, a potent inhibitor of HIV-1. 6th Conference on Retroviruses and Opportunistic Infections; Chicago, 6: abstract 597 p.
- Lin TS, Yang JH, Gao YS. Synthesis of 2′,3′-unsaturated and 2′,3′-dideoxy analogs of 6-azapyrimidine nucleosides as potential anti-HIV agents. Nucleosides & Nucleotides 1990; 9: 97–108
- Okuyama K, Shibuya S, Hamamoto T, Noguchi T. Enzymatic synthesis of 2′-deoxyguanosine with nucleoside deoxyribosyltransferase-II. Biosci Biotechnol Biochem 2003; 65: 989–995
- Schinazi, RF, Liotta, DC. 1996. [5-carboxamide or 5-fluoro]-[2′,3′-unsaturated or 3′-modified]-pyrimidine nucleosides. WO9622778.
- Schinazi, R, Ma, L, Shi, J, Liotta, D, Faraj, A, Sommadossi, JP. 1998. Anti-HIV activity, biochemistry, and pharmacokinetics of β-D-2′,3′-didehydro-2′,3′-dideoxy-5-fluorocytidine (D-D4FC). 12th world AIDS conf; 1998 June 28–July 3, Geneva: abstract 557 p.
- Shi JX, Jeffrey M, Wirtz SS. Synthesis and biological evaluation of 2′,3′-didehydro-2′,3′-dideoxy-5-fluorocytidine(D4FC)analogues: discovery of carbocyclic nucleoside triphosphates with potent inhibitory activity against HIV-1 reverse transcriptase. J Med Chem 1999; 42: 859–867