Correlation between the viscoelastic properties of the gel layer of swollen HPMC matrix tablets and their in vitro drug release

References

• Yin X, Li H, Guo Z, et al. Quantification of swelling and erosion in the controlled release of a poorly water-soluble drug using synchrotron X-ray computed microtomography. AAPS J 2013;15:1025–1034.
   PubMed Web of Science ®Google Scholar
• Colombo P, Bettini R, Santi P, et al. Swellable matrices for controlled drug delivery: gel-layer behaviour, mechanisms and optimal performance. Pharm Sci Tech Today 2000;3:198–204.
   PubMedGoogle Scholar
• Choi DH, Kim KH, Park JS, et al. Evaluation of drug delivery profiles in geometric three-layered tablets with various mechanical properties, in vitro–in vivo drug release, and Raman imaging. J Control Release 2013;172:763–772.
   PubMed Web of Science ®Google Scholar
• Jamzad S, Fassihi R. Development of a controlled release low dose class II drug-Glipizide. Int J Pharm 2006;312:24–32.
   PubMed Web of Science ®Google Scholar
• Li L, Wang LL, Li JF, et al. Insights into the mechanisms of chitosan-anionic polymers-based matrix tablets for extended drug release. Int J Pharm 2014;476:253–265.
   PubMed Web of Science ®Google Scholar
• Roshdy MN, Schwartz JB, Schnaare RL. A novel method for measuring gel strength of controlled release hydrogel tablets using a cone/plate rheometer. Pharm Dev Technol 2001;6:107–116.
   PubMed Web of Science ®Google Scholar
• Bonferoni MC, Rossi S, Tamayo M, et al. On the employment of λ-carrageenan in a matrix system. I. Sensitivity to dissolution medium and comparison with Na carboxymethylcellulose and xanthan gum. J Control Release 1993;26:119–127.
   Web of Science ®Google Scholar
• Hardy IJ, Windberg-Baarup A, Neri C, et al. Modulation of drug release kinetics from hydroxypropyl methyl cellulose matrix tablets using polyvinyl pyrrolidone. Int J Pharm 2007;337:246–253.
   PubMed Web of Science ®Google Scholar
• Kumar SV, Sasmal D, Pal SC. Rheological characterization and drug release studies of gum exudates of Terminalia catappa Linn. AAPS PharmSciTech 2008;9:885–890.
   PubMed Web of Science ®Google Scholar
• Lapidus H, Lordi NG. Drug release from compressed hydrophilic matrices. J Pharm Sci 1968;57:1292–1301.
   PubMed Web of Science ®Google Scholar
• Reynolds TD, Dasbach TP. A study of polymer blending and polymer erosion of different viscosity grades of hypromellose for hydrophilic matrix tablets. Dow Technical Literature 1999.
   Google Scholar
• Cao QR, Choi YW, Cui JH, et al. Formulation, release characteristics and bioavailability of novel monolithic hydroxypropylmethylcellulose matrix tablets containing acetaminophen. J Control Release 2005;108:351–361.
   PubMed Web of Science ®Google Scholar
• Ebube NK, Jones AB. Sustained release of acetaminophen from a heterogeneous mixture of two hydrophilic non-ionic cellulose ether polymers. Int J Pharm 2004;272:19–27.
   PubMed Web of Science ®Google Scholar
• Joshi SC. Sol-gel behavior of hydroxypropyl methylcellulose (HPMC) in ionic media including drug release. Materials 2011;4:1861–1905.
   PubMed Web of Science ®Google Scholar
• Koffi AA, Agnely F, Ponchel G, et al. Modulation of the rheological and mucoadhesive properties of thermosensitive poloxamer-based hydrogels intended for the rectal administration of quinine. Eur J Pharm Sci 2006;27:328–335.
   PubMed Web of Science ®Google Scholar
• Pham AT, Lee PI. Probing the mechanisms of drug release from hydroxypropylmethyl cellulose matrices . Pharm Res 1994;11:1379–1384.
   PubMed Web of Science ®Google Scholar
• Siepmann J, Peppas NA. Modeling of drug release from delivery systems based on hydroxypropyl methylcellulose (HPMC). Adv Drug Deliv Rev 2012;64:163–174.
   Web of Science ®Google Scholar
• Samani SM, Montaseri H, Kazemi A. The effect of polymer blends on release profiles of diclofenac sodium from matrices. Eur J Pharm Biopharm 2003;55:351–355.
   PubMed Web of Science ®Google Scholar
• Velasco MV, Ford JL, Rowe P, et al. Influence of drug:hydroxypropylmethylcellulose ratio, drug and polymer particle size and compression force on the release of diclofenac sodium from HPMC tablets. J Control Release 1999;57:75–85.
   PubMed Web of Science ®Google Scholar
• De Brabander C, Vervaet C, Remon JP. Development and evaluation of sustained release mini-matrices prepared via hot melt extrusion. J Control Release 2003;89:235–247.
   PubMed Web of Science ®Google Scholar
• Gil EC, Colarte AI, Bataille B, et al. Development and optimization of a novel sustained-release dextran tablet formulation for propranolol hydrochloride. Int J Pharm 2006;317:32–39.
   PubMed Web of Science ®Google Scholar
• Hiremath PS, Saha RN. Oral matrix tablet formulations for concomitant controlled release of anti-tubercular drugs: design and in vitro evaluations. Int J Pharm 2008;362:118–125.
   PubMed Web of Science ®Google Scholar
• Missaghi S, Fegely KA, Rajabi-Siahboomi AR. Investigation of the effects of hydroalcoholic solutions on textural and rheological properties of various controlled release grades of hypromellose. AAPS PharmSciTech 2009;10:77–80.
   PubMed Web of Science ®Google Scholar
• Ribeiro L, Ferreira DC, Veiga FJB. In vitro controlled release of vinpocetine-cyclodextrin-tartaric acid multicomponent complexes from HPMC swellable tablets. J Control Release 2005;103:325–339.
   PubMed Web of Science ®Google Scholar
• Asare-Addo K, Kaialy W, Levina M, et al. The influence of agitation sequence and ionic strength on in vitro drug release from hypromellose (E4M and K4M) ER matrices – the use of the USP III apparatus. Colloids Surf B Biointerfaces 2013;104:54–60.
   PubMed Web of Science ®Google Scholar
• Rajabi-Siahboomi A, Bowtell R, Mansfield P, et al. Structure and behavior in hydrophilic matrix sustained release dosage forms: 4. Studies of water mobility and diffusion coefficients in the gel layer of HPMC tablets using NMR imaging. Pharm Res 1996;13:376–380.
   PubMed Web of Science ®Google Scholar
• Escudero JJ, Ferrero C, Jiménez-Castellanos MR. Compaction properties, drug release kinetics and fronts movement studies from matrices combining mixtures of swellable and inert polymers. II. Effect of HPMC with different degrees of methoxy/hydroxypropyl substitution. Int J Pharm 2010;387:56–64.
   PubMed Web of Science ®Google Scholar
• Ghori MU, Ginting G, Smith AM, et al. Simultaneous quantification of drug release and erosion from hypromellose hydrophilic matrices. Int J Pharm 2014;465:405–412.
   PubMedGoogle Scholar
• US FDA dissolution methods for quetiapine fumarate extended release and conventional tablets. Available from: http://www.accessdata.fda.gov/scripts/cder/dissolution/dsp_SearchResults_Dissolutions.cfm [last accessed 12 Nov 2015].
   Google Scholar
• Kočevar-Nared J, Kristl J, Šmid-Korbar J. Comparative rheological investigation of crude gastric mucin and natural gastric mucus. Biomaterials 1997;18:677–681.
   PubMed Web of Science ®Google Scholar
• Yoshimura AS, Prud'homme RK. Wall slip effects on dynamic oscillatory measurements. J Rheol 1988;32:575–584.
   Web of Science ®Google Scholar
• Hewlett KO, L'Hote-Gaston J, Radler M, et al. Direct measurement of the time-dependent mechanical response of HPMC and PEO compacts during swelling. Int J Pharm 2012;434:494–501.
   PubMed Web of Science ®Google Scholar
• Tukaram BN, Rajagopalan IV, Shartchandra PSI. The Effects of lactose, microcrystalline cellulose and dicalcium phosphate on swelling and erosion of compressed HPMC matrix tablets: texture analyzer. Iran J Pharm Res 2010;9:349–358.
   Web of Science ®Google Scholar
• Pygall SR, Kujawinski S, Timmins P, et al. Mechanisms of drug release in citrate buffered HPMC matrices. Int J Pharm 2009;370:110–120.
   PubMed Web of Science ®Google Scholar
• Mehta RY, Missaghi S, Tiwari SB, et al. Application of ethylcellulose coating to hydrophilic matrices: a strategy to modulate drug release profile and reduce drug release variability. AAPS PharmScitech 2014;15:1049–1059.
   PubMed Web of Science ®Google Scholar
• Baumgartner S, Kristl J, Peppas NA. Network structure of cellulose ethers used in pharmaceutical applications during swelling and at equilibrium. Pharm Res 2002;19:1084–1090.
   PubMed Web of Science ®Google Scholar
• Mamani PL, Ruiz-Caro R, Veiga MD. Matrix tablets: the effect of hydroxypropyl methylcellulose/anhydrous dibasic calcium phosphate ratio on the release rate of a water-soluble drug through the gastrointestinal tract I. In vitro tests. AAPS PharmSciTech 2012;13:1073–1083.
   PubMed Web of Science ®Google Scholar
• Asare-Addo K, Levina M, Rajabi-Siahboomi AR, et al. Study of dissolution hydrodynamic conditions versus drug release from hypromellose matrices: the influence of agitation sequence. Colloid Surf B 2010;81:452–460.
   PubMed Web of Science ®Google Scholar
• Cardoso FA, Fujii AL, Pileggi RG, et al. Parallel-plate rotational rheometry of cement paste: influence of the squeeze velocity during gap positioning. Cement Concrete Res 2015;75:66–74.
   Web of Science ®Google Scholar
• Kulinowski P, Woyna-Orlewicz K, Rappen G-M, et al. An understanding of modified release matrix tablets behavior during drug dissolution as the key for prediction of pharmaceutical product performance – case study of multimodal characterization of quetiapine fumarate tablets. Int J Pharm 2015;484:235–245.
   PubMed Web of Science ®Google Scholar
• Kulinowski P, Woyna-Orlewicz K, Obrał J, et al. Multimodal approach to characterization of hydrophilic matrices manufactured by wet and dry granulation or direct compression methods. Int J Pharm 2016;499:263–270.
   PubMedGoogle Scholar
• Rudraraju VS, Wyandt CM. Rheology of microcrystalline cellulose and sodiumcarboxymethyl cellulose hydrogels using a controlled stress rheometer: part II. Int J Pharm 2005;292:63–73.
   PubMed Web of Science ®Google Scholar
• Ford JL, Mitchell K, Rowe P, et al. Mathematical modelling of drug release from hydroxypropylmethylcellulose matrices: Effect of temperature. Int J Pharm 1991;71:95–104.
   Web of Science ®Google Scholar
• Sauri J, Millan D, Sune-Negre JM, et al. Quality by Design approach to understand the physicochemical phenomena involved in controlled release of captopril SR matrix tablets. Int J Pharm 2014;477:431–441.
   PubMed Web of Science ®Google Scholar
• Jones DS, Muldoon BCO, David Woolfson A, et al. Rheological destructuring of aqueous gels composed of cellulose ethers following storage in the presence of redox agents. J Appl Polym Sci 2005;98:852–859.
   Web of Science ®Google Scholar