Inhibition of the solid state transformation of carbamazepine in aqueous solution: impact of polymeric properties

References

• Ashland. 2016. Pharma product grades. [accessed 2017 Oct 30]. http://www.ashland.com/file_source/Ashland/Industries/Pharmaceutical/Links/PHA17-1002_Pharma_Product_Grades.pdf
   Google Scholar
• Barton AFM. 1990. Handbook of polymer-liquid interaction parameters and solubility parameters. New York: CRC Press.
   Google Scholar
• Cardew PT, Davey RJ. 1985. The kinetics of solvent mediated phase transformations. Proc R Soc London. A398:415–428.
   Web of Science ®Google Scholar
• Gift AD, Luner PE, Luedeman L, Taylor LS. 2008. Influence of polymeric excipients on crystal hydrate formation kinetics in aqueous slurries. J Pharm Sci. 97:5198–5211.
   PubMed Web of Science ®Google Scholar
• Gift AD, Luner PE, Luedeman L, Taylor LS. 2009. Manipulating hydrate formation during high shear wet granulation using polymeric excipients. J Pharm Sci. 98:4670–4683.
   PubMed Web of Science ®Google Scholar
• Gift AD, Southard LA, Riesberg AL. 2012. Influence of polymeric excipient properties on crystal hydrate formation kinetics of caffeine in aqueous slurries. J Pharm Sci. 101:1755–1762.
   PubMed Web of Science ®Google Scholar
• Ilevbare GA, Liu HY, Edgar KJ, Taylor LS. 2012. Inhibition of solution crystal growth of ritonavir by cellulose polymers - factors influencing polymer effectiveness. Crystengcomm. 14:6503–6514.
   Web of Science ®Google Scholar
• Jorgensen AC, Airaksinen S, Karjalainen M, Luukkonen P, Rantanen J, Yliruusi J. 2004. Role of excipients in hydrate formation kinetics of theophylline in wet masses studied by near-infrared spectroscopy. Eur J Pharm Sci. 23:99–104.
   PubMed Web of Science ®Google Scholar
• Katzhendler I, Azoury R, Friedman M. 1998. Crystalline properties of carbamazepine in sustained release hydrophilic matrix tablets based on hydroxypropyl methylcellulose. J Control Release. 54:69–85.
   PubMed Web of Science ®Google Scholar
• Keary CM. 2001. Characterization of METHOCEL cellulose ethers by aqueous SEC with multiple detectors. Carbohyd Polym. 45:293–303.
   Web of Science ®Google Scholar
• Kestur US, Taylor LS. 2010. Role of polymer chemistry in influencing crystal growth rates from amorphous felodipine. Crystengcomm. 12:2390–2397.
   Web of Science ®Google Scholar
• Kramarenko EY, Winkler RG, Khalatur PG, Kohkhlov AR, Reineker P. 1996. Molecular dynamics simulation study of adsorption of polymer chains with variable degree of rigidity. 1. Static properties. J Chem Phys. 104:4806–4813.
   Web of Science ®Google Scholar
• Kubota N. 2001. Effect of impurities on the growth kinetics of crystals. Cryst Res Technol. 36:749–769.
   Web of Science ®Google Scholar
• Luhtala S, Kinos E, Yliruusi J, Tanninen VP. 1992a. X-ray-powder diffraction study of carbamazepine crystals grown in surfactant solutions. Acta Pharm Nordica. 4:283–290.
   Google Scholar
• Luhtala S. 1992b. Effect of poloxamer 184 on crystal-growth and aqueous solubility of carbamazepine. Acta Pharm Nordica. 4:271–276.
   Google Scholar
• Luhtala S. 1992c. Effect of sodium lauryl sulfate and polysorbate-80 on crystal-growth and aqueous solubility of carbamazepine. Acta Pharm Nordica. 4:85–90.
   Google Scholar
• McMahon LE, Timmins P, Williams AC, York P. 1996. Characterization of dihydrates prepared from carbamazepine polymorphs. J Pharm Sci. 85:1064–1069.
   PubMed Web of Science ®Google Scholar
• Otsuka M, Ohfusa T, Matsuda Y. 2000. Effect of binders on polymorphic transformation kinetics of carbamazepine in aqueous solution. Colloid Surface B. 17:145–152.
   Web of Science ®Google Scholar
• Paisana M, Wahl M, Pinto J. 2015. Role of polymeric excipients in the stabilization of olanzapine when exposed to aqueous environments. Molecules. 20:22364–22382.
   PubMed Web of Science ®Google Scholar
• Patel DD, Anderson BD. 2015. Adsorption of polyvinylpyrrolidone and its impact on maintenance of aqueous supersaturation of indomethacin via crystal growth inhibition. J Pharm Sci. 104:2923–2933.
   PubMed Web of Science ®Google Scholar
• Qu H, Louhi-Kultanen M, Kallas J. 2007. Additive effects on the solvent-mediated anhydrate/hydrate phase transformation in a mixed solvent. Cryst Growth Des. 7:724–729.
   Web of Science ®Google Scholar
• Raina SA, Van Eerdenbrugh B, Alonzo DE, Mo HP, Zhang GGZ, Gao Y, Taylor LS. 2015. Trends in the precipitation and crystallization behavior of supersaturated aqueous solutions of poorly water-soluble drugs assessed using synchrotron radiation. J Pharm Sci. 104:1981–1992.
   PubMed Web of Science ®Google Scholar
• Rodriguez-Hornedo N, Murphy D. 2004. Surfactant-facilitated crystallization of dihydrate carbamazepine during dissolution of anhydrous polymorph. J Pharm Sci. 93:449–460.
   PubMed Web of Science ®Google Scholar
• Schram CJ, Taylor LS, Beaudoin SP. 2015. Influence of polymers on the crystal growth rate of felodipine: correlating adsorbed polymer surface coverage to solution crystal growth inhibition. Langmuir. 31:11279–11287.
   PubMed Web of Science ®Google Scholar
• Shefter E, Higuchi T. 1963. Dissolution behavior of crystalline solvated and nonsolvated forms of some pharmaceuticals. J Pharm Sci. 52:781–791.
   PubMed Web of Science ®Google Scholar
• Somasundaran P, Krishnakumar S. 1997. Adsorption of surfactants and polymers at the solid-liquid interface. Colloid Surface A. 123:491–513.
   Google Scholar
• Tian F, Saville DJ, Gordon KC, Strachan CJ, Zeitler JA, Sandler N, Rades T. 2007. The influence of various excipients on the conversion kinetics of carbamazepine polymorphs in aqueous suspension. J Pharm Pharmacol. 59:193–201.
   PubMed Web of Science ®Google Scholar
• Tian F, Zeitler JA, Strachan CJ, Saville DJ, Gordon KC, Rades T. 2006. Characterizing the conversion kinetics of carbamazepine polymorphs to the dihydrate in aqueous suspension using Raman spectroscopy. J Pharmaceut Biomed. 40:271–280.
   PubMed Web of Science ®Google Scholar
• Trasi NS, Taylor LS. 2012a. Effect of additives on crystal growth and nucleation of amorphous flutamide. Cryst Growth Des. 12:3221–3230.
   Web of Science ®Google Scholar
• Trasi NS, Taylor LS. 2012b. Effect of polymers on nucleation and crystal growth of amorphous acetaminophen. Crystengcomm. 14:5188–5197.
   Web of Science ®Google Scholar
• Wikstrom H, Carroll WJ, Taylor LS. 2008a. Manipulating theophylline monohydrate formation during high-shear wet granulation through improved understanding of the role of pharmaceutical excipients. Pharmaceut Pharm Res. 25:923–935.
   PubMed Web of Science ®Google Scholar
• Wikstrom H, Rantanen J, Gift AD, Taylor LS. 2008b. Toward an understanding of the factors influencing anhydrate-to-hydrate transformation kinetics in aqueous environments. Cryst Growth Des. 8:2684–2693.
   Web of Science ®Google Scholar
• Ziller KH, Rupprecht H. 1988. Control of crystal-growth in drug suspensions. 1. Design of a control unit and application to acetaminophen suspensions. Drug Dev Ind Pharm. 14:2341–2370.
   Web of Science ®Google Scholar
• Zimmermann A, Millqvist-Fureby A, Elema MR, Hansen T, Muellertz A, Hovgaard L. 2009. Adsorption of pharmaceutical excipients onto microcrystals of siramesine hydrochloride: effects on physicochemical properties. Eur J Pharm Biopharm. 71:109–116.
   PubMed Web of Science ®Google Scholar