Synthesis and anti-inflammatory activity of some selected aminothiophene analogs

References

• De Almeida EC, Menezes H. Anti-inflammatory activity of propolis extracts: A review. J Venom Anim Toxins 2002; 8: 191–212
   Google Scholar
• Heiba HI, Ghorab MM, El-Gawish MA. Biological and biochemical screening of some new amino acid thienopyrimidinone derivatives for potential radioprotective character. Phosphorus, Sulphur Silicon Relat Elem 1997; 131: 197–205
   Web of Science ®Google Scholar
• Pathak US, Gandhi NV, Singh S, Warde RP, Jain KS. Synthesis of some [1,2,4]triazolo[4,3-a]thieno[3,2-e]pyrimidin-5(4H)-ones. Indian J Chem Sec B 1992; 31: 223–229
   Google Scholar
• Sauter F. Ger. Offen, 2,210,503. 2-Mercapto-3,4-dihydrothieno[2,3-d]pyrimidin-4-ones Chem Abstr. 1972;77:164752n.
   Google Scholar
• Kinnard WJ, Carr CJ. A preliminary procedure for evaluation of central-nervous-system depressants. J Pharmacol Exptl Therap 1957; 121: 354–361
   PubMed Web of Science ®Google Scholar
• Tripathi S, Ahmad S, Barthwal JP, Tangri KK, Kishore K, Bhargava KP. Anticonvulsant and MAO inhibitory activity of substituted quinozolines. Indian J Exp Biol 1981; 19: 30–33
   Web of Science ®Google Scholar
• Doria G, Passarotti C, Arcari G, Buttinoni A. Belg. BE 893,835, Substituted thiazolo[3,2-a]pyrimidines Chem Abstr, 1983;99:70749u.
   Google Scholar
• Zhikhareva GP, Mastafanova LI, Evstratova MI, Polukhina LM, Pushkina TV, Pershin GN, Yakhontov LN. Synthesis and chemotherapeutic study of 2-styryl-4-(δ-diethylamino-α-methylbutylamino)quinazolines. Khim-Farm Zh 1982; 16: 199625t, 1982;16:183–188; Chem Abstr
   Google Scholar
• Zhikhareva GP, Pronina EV, Golovanova EA, Pershin GN, Novitskaya NA, Zykova TN, Guśkova TA, Yakhontov LN. Synthesis and chemotherapeutic study of substituted 2-styryl-4-amino-6-methoxyquinazolines. Khim-Farm Zh 1976; 85: 123848v, 1976;10:62; Chem Abstr
   Google Scholar
• Manhas MS, Amin SG, Sharma SD, Dayal B, Bose KA. Heterocyclic compounds. XI Potential Post-Coital Antifertility Agent (I). J Heterocyclic Chem 1979; 16: 371–376
   Web of Science ®Google Scholar
• Bosin TR, Campaigne EE. Biologically active benzo[b]thiophene derivatives. Adv Drug Res 1977; 11: 191–232
   PubMedGoogle Scholar
• Campaigne E, Homfeld E. Benzo[b]thiophene derivatives. XXV. Condensation and reductive Alkylation of 3-aminoalkylbenzo[b]thiophenes with formaldehyde (1). J Heterocyclic Chem 1979; 16: 1321–1324
   Web of Science ®Google Scholar
• Schmidt P, Eichenberger K, Schweizer E, Ger Offen 1969;497:1,908, Pyrimidines. Chem Abstr. 1970;72;31837u
   Google Scholar
• Eichenberger K, Schweizer E, Schmidt P, U. S. Patent. 2,627,766, December 14, 1971
   Google Scholar
• Medicinal Chemistry. Medicinal Chemistry3rd ed., A Burgered. Willey-Inter sciences, New York 1970; 72–544 and 719
   Google Scholar
• Brown DJ. Katritzky and Rees Comprehensive Heterocyclic Chemistry, AJ Boulton, A McKillop. Pergamon Press, Oxford 1983; 3: 57
   Google Scholar
• Charles H, Fred JA. Experimental and clinical use of fluorinated pyrimidines in cancer chemotherapy. Cancer Res 1963; 23: 1226–1243
   PubMed Web of Science ®Google Scholar
• De Clercq E. Chemotherapeutic approaches to the treatment of the acquired immune deficiency syndrome (AIDS). J Med Chem 1986; 29: 1561–1569
   PubMed Web of Science ®Google Scholar
• Baba M, Pauwels R, Herdewijn P, De Clercq E, Desmyter J, Vandeputte M. Both 2′,3′-dideoxythymidine and its 2′,3′-unsaturated derivatives (2′,3′-dideoxythymidinene) are potent and selective inhibitors of human immunodeficiency virus replication in vitro. Biochem Biophys Res Commun 1987; 142: 128–134
   PubMed Web of Science ®Google Scholar
• Kelley JL, Linn JA, Selway JWT. Synthesis and structure-activity relationship of 2-substituted-6-(dimethylamino)-9-(4-methybenzyl)-(4H)-purines with antirhinovirus activity. J Med Chem 1989; 32: 218–224
   PubMed Web of Science ®Google Scholar
• Peet NP, Sunder S, Barbuch RJ. Mechanistic observations in Gewald syntheses of 2-aminothiophenes. J Heterocylic Chem 1986; 23: 129–134
   Web of Science ®Google Scholar
• Siddiqui RA, English D, Harvey K, Cui Y, Martin MI, Wentland J, Akard L, Jansen J, Thompson J, Garcia JGN. Phorbol ester-induced priming of superoxide generation by phosphatidic acid-stimulated neutrophils and granule-free neutrophil cytoplasts. J Leukocytes Biol 1995; 58: 189–195
   PubMed Web of Science ®Google Scholar
• Bagchi D, Bagchi M, Stohs SJ. In vitro effects of a smokeless tobacco extract in the production of reactive oxygen species by human oral epidermal cells and rat hepatic mitochondria and microsomes and peritoneal macrophages. Biosci Biotech Biochem 1995; 59: 822
   PubMed Web of Science ®Google Scholar