References
- Levitzki A, Gazit A. Science 1995; 276: 1782–1788
- Gibbs JB, Oliff A. Cell 1994; 79: 193–198
- Clark GJ, Der CJ. Ras prota-oncogene activation in human malignancy. Cellular markers, CT Garnett, S Sell, 1995; 17–52
- Lowry DR, Willumsen BM. Annu Rev Biochem 1993; 62: 851–891
- Bernards R. Biochim Biophys Acta 1995; 1242: 43–59
- Largacspada DA, Branan CI, Jenkins NA, Copeland NG. Nat Genet 1996; 12: 137–143
- Gibbs JB. Semin Cancer Biol 1992; 3: 383–390
- Spaargaren M, Bischoff JR, McCornick F. Gene Exp 1995; 4: 345–356
- Manne V, Ricca CS, Brown JG, Tuomari AV, Yan N. Drug Dev Res 1995; 34: 121–137
- Willumsen BM, Norris K, Papageorge AG, Hubbert NL, Lowrey DR. EMBO J 1984; 3: 2581–2585
- Casey PJ, Solski PA, Der C, Bus JE. Proc Natl Acad Sci USA 1989; 86: 8323–8327
- Zhang FL, Casey PJ. Annu Rev Biochem 1996; 65: 241–269
- Leonard DM. J Med Chem 1997; 40: 2971–2990
- Fu HW, Casey PJ. Recent Prog Horm Res 1999; 54: 315–343
- Long SB, Casey PJ, Beese LS. Nature 2002; 419: 645–650
- Hightower KE, Huang C, Casey PJ, Fierke CA. Biochemistry 1998; 37: 15555–15562
- Rozema DB, Poulter CD. Biochemistry 1999; 38: 13138–13146
- Tschantz WR, Furfine ES, Casey PJ. J Biol Chem 1997; 272: 9989–9993
- Adjei A. J Natl Cancer Inst. 1062–1074, 932001a
- Cox D. Drugs 2001; 61: 723–732
- Hill TH, Hunt JT, Ding CZ, Batorsky R, Bednarz M, Bhide R, Cho Y, Chong S, Cho S, Gullo-Brown J, Guo P, Kim SH, Lee FY, Leftheris K, Miller A, Mitt T, Patel M, Penhallow BA, Ricca C, Rose WC, Schmidt R, Slusarchyk WA, Vite G, Perrin D, Kruczynski L. Crit Rev Oncol Hematol 2000; 33: 7–23
- Hahn SM, Bernhard E, McKenna WG. Semi Oncol 2001; 28: 86–93
- Karp JE, Kauffman SH, Adjei AA, Lancet JE, Wright JJ. Curr Opin Oncol 2001a; 13: 470–476
- Katz ME, McCormick F. Curr Opin Genet Dev 1997; 7: 75–79
- Boettner B, Van Aelst L. Genes Dev 2002; 16: 2033–2038
- Olson MF, Marais R. Semin Immunol 2000; 12: 63–73
- Hamad NE, Elconin JE, Karnoub AE, Bai W, Rich NJ, Abraham NT, Der CJ, Counter CM. Genes Dev 2002; 16: 2045–2057
- Bos JL. Cancer Res 1989; 49: 4682–4689
- Takai Y, Sasaki T, Matozaki T. Physiol Rev 2001; 81: 153–208
- Purcell WT, Donehower RC. Curr Oncol Rep 2002; 4: 29–36
- Falugi C, Trombino S, Granote P, Margaritota S, Russo P. Curr Cancer Drug Targets 2003; 3: 109–118
- Sebti SM, Hamilton AD. Oncogene 2000; 19: 6584–6593
- Crespo NC, Ohkanda J, Yen TJ, Hamilton AD, Sebti SM. J Biol Chem 2001; 276: 16161–16167
- Crespo NC, Delarve F, Ohkanda J, Carrico D, Hamilton AD, Sebti SM. Cell Death Differ 2002; 9: 702–709
- Ashar HR, James L, Gray K, Carr D, Black S, Armstrong L, Bishop WR, Kirschmeier P. J Biol Chem 2000; 275: 30451–30457
- Ashar HR, James L, Gray K, Carr D, McGuirk M, Maxwell E, Black S, Armstrong L, Doll RJ, Taveras AG, Bishop WR, Kirschmeier P. Exp Cell Res 2001; 262: 17–27
- Sebti SM, Hamilton AD. Drug Discov Today 1998; 3: 26–33
- Williams TM. Expert Opin Ther Patents 1999; 9: 1263–1280
- Rowinsky EK, Patnaik A. Emerg Drugs 2000; 5: 161–199
- Taveras G, Kirschneier P, Baum CM. Curr Top Med Chem 2003; 3: 1103–1114
- Kohl N, Omer C, Conner M, Anthony N, Davide J, Desolms S, Giuliani E, Gomez R, Graham S, Hamilton K, Handt L, Hartman G, Koblan K, Kral K, Miller P, Mosser S, O'Neil T, Rands T, Schabler M, Gibbs J, Oliff A. Nature Med 1995; 1: 792–797
- Lerner LC, Qian Y, Blaskowich MA, Ossum RD, Vogt A. J Biol Chem 1995; 270: 26802–26806
- Stephens TC, Wardleworth MJ, Matuziak MZ, Ashton SE, Hancox UJ, Bate M, Ferguson R, Boyle T. Proc Am Assoc Cancer Res 2003; 44: R4870
- Williams TM, Giccarone TM, MacTough SC, Bock RL, Conner MW, Davide JP, Hamilton K, Koblan KS, Kohl NE, Kral AM, Mosser SD, Omer CA, Pompliano DE, Rands E, Schaber MD, Shah D, Wilson FR, Gibbs JB, Graham SL, Hartman GD, OLiff AI, Smith RL. J Med Chem 1996; 39: 1345–1348
- Anthony NJ, Gomez RP, Schaber MD, Mosser SD, Hamilton KA, O'Neill TJ, Koblan KS, Graham SL, Hartman GD, Shah D, Rands E, Kohl NE, Gibbs JB, Oliff AI. J Med Chem 1999; 42: 3356–3368
- Williams TM, Bergman JM, Braschear K, Breslin MJ, Dinsmore CJ, Hutchinson JH, MacTough SC, Stump CA, Wei DD, Zartmen CB, Bogusky MJ, Culberson JC, Buser-Doepner C, Davide J, Greenberg IB, Hamilton KA, Koblan KS, Kohl NE, Liu D, Lobell RB, Mosser SD, O'Neill TJ, Rands E, Schabler MD, Wilson F, Senderak E, Motzel SL, Gibbs JB, Graham SL, Heimbook DC, Hartman GD, Oliff AI, Huff JR. J Med Chem 1999a; 42: 3779–3784
- Dinsmore CJ, Bogusky MJ, Culberson JC, Bergman JM, Homnick CF, Zartman CB, Mosser SD, Schaber MD, Robinson RG, Koblan KS, Huber HE, Graham SL, Hartman GD, Huff JR, Williams TM. J Am Chem Soc 2001; 123: 2107–2108
- Bell M, Gallicchio SN, Abrams M, Beese LS, Bishore DC, Bhimnathwala H, Bogusky MJ, Buser CA, Culberson JC, Divide J, Ellis-Hutchings M, Fernandes C, Gibbs JB, Graham SL, Hartman GD, Heimbrook DC, Homnick CF, Huber HE, Huff JR, Kassahun K, Koblan KS, Kohl NE, Lobell RB, Lynch JJ, Robinson R, Rodrigues AD, Taylor JS, Walsh ES, Williams TM, Zartmen CB. J Med Chem 2002; 45: 2388–2409
- Hunt JT, Lee VJ, Leftheris K, Seizinger B, Carboni J, Mabus J, Ricca C, Yan N, Manne V. J Med Chem 1996; 39: 353–358
- Ding CZ, Batorsky R, Bhide R, Chao HJ, Cho Y, Chong S, Gullu-Brown J, Guo P, Kim SH, Lee F, Leftheris K, Miller A, Mitt T, Patel M, Penhallow BA, Ricca C, Rose WC, Schmidt R, Slusarchyk WA, Vite G, Yan N, Manne V, Hunt JT. J Med Chem 1999; 42: 5241–5253
- Njoroge FG, Taveras AG, Kelly J, Remiszewiski S, Mallams AK, Wolin R, Afonso A, Cooper AB, Rane DF, Liu YT, Wong J, Vibhulban B, Pinto P, Deskus J, Alvarez CS, Del Rosario J, Connoly M, Wang J, Desai J, Rossman RR, Venet M, End D, Anggibaud P. Curr Top Med Chem 2003; 3: 1095–1102
- End DW, Smets G, Todd AV, Applegate TL, Fuery CJ, Angibaud P, Venet M, Sanz G, Poignet H, Skrzat S, Devine A, Wouters W, Bowden C. Cancer Res 2001; 61: 131–137
- Esteva MI, Kettler K, Maidana C, Fichera L, Ruiz AM, Bontempi EJ, Anderson B, Dahse H-M, Haebel P, Ortmann R, Klebe G, Schlitzer M. J Med Chem 2005; 48: 7186–7191
- Huckeo O, Gelb MH, Verlinde CLMJ, Buckner FS. J Med Chem 2005; 48: 5415–5421
- Huang C-Y, Stauffer TM, Strickland CL, Reader JC, Huang H, Li G, Cooper AB, Doll RJ, Ganguly AK, Baldwin JJ, Rokosz LL. Bioorg Med Chem Lett 2006; 16: 507–511
- Li Q, Li T, Woods KW, Gu WZ, Cohen J, Stoll VS, Galicia T, Hutchins C, Frost D, Rosenberg SH, Sham HL. Bioorg Med Chem Lett 2005; 15: 2918–2922
- Kettler K, Wiesner J, Sibler K, Haebel P, Ortmann R, Sattler I, Dahse H-M, Jomaa H, Klebe G, Schlitzer M. Eur J Med Chem 2005; 40: 93–101
- Guida WC, Hamilton AD, Crotty JW, Sebti SM. J Comput Aided Mol Des 2006; 19: 871–885
- Graham SL. Expert Opin Ther Patents 1995; 5: 1269–1285
- Hara M, Akasaka K, Akinaga S, Okabe M, Nakano H. Proc Natl Acad Sci USA 1993; 90: 2281–2285
- Gibbs JB, Pompliano DL, Mosser SD, Rands E, Lingham RB. J Biol Chem 1993; 268: 7617–7620
- Kohl NE, Mosser SD, dsolms SJ, Giuliani EA, Pomliano DL. Science 1993; 260: 1934–1937
- James GL, Goldstein JL, Brown MS, Rawson TE, Sommers TC. Science 1993; 260: 1937–1942
- Dalton MB, Fantle KS, Beehtold HE, DeMaio L, Evans RM. Cancer Res 1995; 55: 3295–3304
- James GL, Goldstein JL, Pathak RK, Anderson RJW, Brown MS. J Biol Chem 1994; 269: 14182–14190
- Vogt A, Qian Y, Blaskowich MA, Fossum RD, Hamilton AD. J Biol Chem 1995; 270: 660–664
- Lerner EC, Qian Y, Blaskowich MA, Fossum RD, Vogt A, Sun J, Cox AD, Der CJ, Hamilton AD, Sebti SM. J Biol Chem 1995; 270: 26802–26806
- Nagasu T, Yoshimatsu K, Rowel C, Lewis MD, Garcin AM. Cancer Res 1995; 55: 5310–5314
- Cox D, Garcia AM, Westwick JK, Kowalczyk JJ, Lewis MD. J Biol Chem 1994; 269: 19203–19206
- Prendergast GC, Davide JP, deSolms SJ, Giulani EA, Graham SL. Mol Cell Biol 1994; 14: 4193–4202
- Sun J, Qian Y, Hamilton AD, Sebti SM. Cancer Res 1995; 55: 4243–4247
- Pai JJ-K, Bishop WR, Catino J, Kirschemeier P, Whyte D. Proc Am Assoc Cancer Res 1996; 37: 503–510
- Yan N, Ricca C, Fletcher J, Glover T, Scizinger BR. Cancer Res 1995; 55: 3569–3575
- Sepp-Lorenzino L, Ma Z, Rands E, Kohl NE, Gibbs JB. Cancer Res 1995; 55: 5302–5309
- Smith MR, DeGudiebus SJ, Staccay DW. Nature 1986; 320: 540–543
- Staccy DW, Roudebush M, Day R, Mosser SD, Gibbs JB. Oncogene 1991; 6: 2297–2304
- Ito T, Kawata S, Tamura S, Igura T, Nagase T. Jpn J Cancer Res 1996; 87: 113–116
- Sinn E, Muller W, Pattengale P, Tepler I, Wallace R. Cell 1987; 49: 465–475
- Hancock JF, Kadwalleder K, Patterson H, Marshall CJ. EMBO J 1991; 10: 4033–4039
- Cox D, Hisaka MM, Buss JE, Der CJ. Mol Cell Biol 1992; 12: 2606–2615
- James GL, Brown MS, Cobb MH, Goldstein JH. J Biol Chem 1994; 269: 27705–27714
- Prevost GP, Pradines A, Viossat I, Brezak MC, Miquek K, Lonchampt MO, Kaspryzk P, Favre G, Pignol B, Le Breton C, Dong J, Morgan B. Int J Cancer 1999; 83: 283–287
- Prevost GP, Pradines A, Brezak MC, Lonchampt MO, Viossat I, Ader I, Toulas C, Kaspryzk P, Gordon T, Favre G, Morgan B. Int J Cancer 2001; 91: 718–722
- Adjei A, Davis JN, Bruzek LM, Erlichman C, Kauffman SH. Clin Cancer Res 2001; 7: 1438–1445
- Shi B, Yaremko B, Hajian G, Terracina G, Bishop WR, Liu M, Nielson LL. Cancer Chemother Pharmacol 2000; 46: 387–393
- Mangues R, Corral T, Kohl NE, Symanns WF, Lu S, Malumbres M, Gibbs JB, Oliff A. Cancer Res 1998; 58: 1253–1259
- Liu M, Bryant MS, Chen J, Lee S, Yaremko B, Lipari P, Malkowiski M, Ferrari E, Nielson L, Prioli N, Dell J, Sinha D, Syed J, Korfmacher WA, Nomier AA, Lin CC, Wang L, Taveras AG, Doll RJ, Njoroge FG, Mallams AK, Remiszewiski S, Catino JJ, Girijavallabhan VM, Bishop WR. Cancer Res 1998; 58: 4947–4956
- Dinsmore CJ, Bell IM. Curr Top Med Chem 2003; 3: 1075–1093
- Crul M, de Klerk GJ, Swart M, van't Veer LJ, de Jong D, Boerrigter L, Palmer PA, Bol CJ, Tan H, de Gast GC, Beijnen JH, Schellens JH. J Clin Oncol 2002; 20: 2726–2735
- Kantarjian HM, Cortes JE, Rowe JM, Kurzrock R. Semin Hematol 2002; 39: 36–38
- Lobell RB, Liu D, Buser CA, Davide JP, DePuy E, Hamilton K, Koblan KS, Lee Y, Mosser S, Motzel SL, Abruzzesse JL, Fuchs CS, Rowinsky EK, Rubin EH, Sharma S, Deustch PJ, Mazina KE, Morrison BW, Wildonger L, Yao SL, Kohl NE. Mol Cancer Ther 2002; 1: 747–758
- Adjei A, Davis JN, Erlichman C, Svigen PA, Kaufman SH. Clin Cancer Res 2000; 6: 2318–2325
- , Johnston HRD, Hickish T, Houston S, Ellis PA, Howes AJ, Thibault A. Presented at the 38th Annual meeting of the American Society of Clinical Oncology 2002. Abstract 138.
- Karp JE, Lancet JE, Kauffman SH, End DW, Wright JJ, Bol K, Horak I, Tidwell ML, Liesweld J, Kottke TJ, Ange D, Buddharaju L, Gojo I, Highsmith WE, Belly RT, Hohl RJ, Rybak ME, Thibault A, Rossenbat J. Blood 2001; 97: 3361–3369
- Cortes J, Albitar M, Thomas D, Giles F, Kurzrock R, Thibault A, Rackoff W, Koller C, O'Brien S, Garcia-Manero G, Talpaz M, Kantarjian H. Blood 2003; 101: 1692–1697
- , Lersch C, van Custem E, Amado R, Ehninger G, Heike M, Kerr D, Rothenberg ML, Baum CM, Zakneon SL. Presented at the 37th Annual meeting of the American Society of Clinical Oncology 2001. Abstract 608.
- Britten CD, Rowinsky EK, Soignet S, Patnaik A, Yao SL, Deutsch P, Lee Y, Lobell RB, Mazina KE, McCreery H, Pezulli S, Spriggs DA. Clin Cancer Res 2001; 7: 3894–3903
- Haluska P, Dy GK, Adjei AA. Eur J Cancer 2002; 38: 1685–1700
- Moasser MM, Sepp-Lorenzino L, Kohl NE, Oliff A, Su DS, Danishefsky SJ, Rosen N. Proc Natl Acad Sci USA 1998; 95: 1369–1374
- Sun J, Blaskowich MA, Knowles D, Qian Y, Ohka J, Bailey RD, Hamilton AD, Sebti SM. Cancer Res 1999; 59: 4919–4926
- Hoover RR, Mahon FX, Melo JV, Daley GQ. Blood 2002; 100: 1068–1071
- Nakajima A, Tauchi T, Sumi M, Bishop WR, Ohyashik K. Mol Cancer Ther 2003; 2: 219–224
- Hahn SM, Bernhard EJ, Regine W, Mohiuddin M, Haller DG, Stevenson JP, Smith D, Pramanik B, Tepper J, DeLaney TF, Kiel KD, Morrison B, Deutsh P, Muschel RJ, McKenna WG. Clin Cancer Res 2002; 8: 1065–1072
- Adjei A, Croghan GA, Erlichman C, Marks RS, Reid JM, Sloan JA, Pitot HC, Alberts SR, Goldberg RM, Hanson LJ, Bruzek LM, Atherton P, Thibault A, Palmer PA, Kauffman SH. Clin Cancer Res 2003; 9: 2520–2526
- Widemann BC, Salzer WL, Arceci RJ, Blaney SM, Fox E, End D, Gillespie A, Whitcomb P, Palumbo JS, Pitney A, Jayaprakash N, Zannikos P, Balis FM. J Clin Oncol 2006; 24(3)507–516
- Sparano JA, Moulder S, Kazi A, Vahdat L, Li T, Pellegrino C, Munster P, Malafa M, Lee D, Hoschander S, Hopkins U, Hershman D, Wright JJ, Sebti SM. J Clin Oncol 2006; 24(19)3013–3018
- Corey LS, William TW, Rosalinda S, Lyan W, Richard B, Zhen W, Jeffry S, Hung VL, Lorena SB, Patricia CW. Biochemistry 1998; 37: 16601–16611
- Pete D, Ursula K, Robert C, David W, Robert P, Jens B. Biochemistry 1998; 37: 7907–7912
- Tammy CT, Corey LS, Mark DD. Biochemistry 2003; 42: 3716–3724
- Markus B, Andreas M, Pia W, Isbel S, Martin S. J Med Chem 2001; 44: 3317–3324
- Alessandro P, Luigi V, Giulio V. J Med Chem 2002; 45: 1460–1465
- Brian SH, Todd JZ, Jrffery DE, Steven MF, Richard AG. J Chem Inf Model 2005; 45: 1047–1052
- Perola E, Xu K, Kollmeyer TM, Kauffmann SH, Prendergast FG, Pang YP. J Med Chem 2000; 43: 401–408
- Puntambekar D, Giridhar R, Yadav MR. Bioorg Med Chem Lett 2006; 167: 1821–1827
- Puntambekar DS, Giridhar R, Yadav MR. Eu Med Chem 2006, In Press
- Xie A, Sivprakasan P, Doerkson R. Bioorg Med Chem 2006, Jul 10: In Press
- Gonzalez MP, Caballero J, Tundidor-Camba A, Helguera AM, Fernandez M. Bioorg Med Chem 2006; 14(1)200–213
- Rokosz LL, Huang CY, Reader JC, Stauffer TM, Southwick EC, Li G, Chelsky D, Baldwin JJ. Comb Chem High Throughput Screen 2006; 9(7)545–548