Advanced search
Publication Cover
Journal of Enzyme Inhibition and Medicinal Chemistry Volume 32, 2017 - Issue 1
Submit an article Journal homepage
1,273
Views
4
CrossRef citations to date
0
Altmetric
Original Article

Syntheses and evaluation of multicaulin and miltirone-like compounds as antituberculosis agents

Serdar BurmaoğluDepartment of Chemistry, Faculty of Science, Ataturk University, Erzurum, Turkey; ;Tercan Vocational High School, Erzincan University, Erzincan, Turkey; Correspondence[email protected]
View further author information
,
Hatice SeçintiDepartment of Chemistry, Faculty of Science, Ataturk University, Erzurum, Turkey; View further author information
,
Erkan MozioğluChemistry Group Laboratories, TÜBİTAK, UME, Gebze-Kocaeli, TurkeyView further author information
,
Ahmet C. GörenChemistry Group Laboratories, TÜBİTAK, UME, Gebze-Kocaeli, TurkeyView further author information
,
Ramazan AltundaşDepartment of Chemistry, Faculty of Science, Ataturk University, Erzurum, Turkey; View further author information
&
Hasan SeçenDepartment of Chemistry, Faculty of Science, Ataturk University, Erzurum, Turkey; View further author information
Pages 878-884 | Received 14 Mar 2017, Accepted 23 May 2017, Published online: 29 Jun 2017

References

  • Tiwari R, Moraski GC, Krchňák V, et al. Thiolates chemically induce redox activation of BTZ043 and related potent nitroaromatic anti-tuberculosis agents. J Am Chem Soc 2013;135:3539–49.
  • WHO Global Tuberculosis Report. (2016). Available from: http://who.int/tb/publications/global_report/en/ [last accessed 14 May 2017].
  • Addla D, Jallapally A, Gurram D, et al. Design, synthesis and evaluation of 1,2,3-triazoleadamantylacetamide hybrids as potent inhibitors of Mycobacterium tuberculosis. Bioorg Med Chem Lett 2014;24:1974–9.
  • Naik M, Ghorpade S, Jena LK, et al. Phenylindole and arylsulphonamide: novel scaffolds bactericidal against Mycobacterium tuberculosis. ACS Med Chem Lett 2014;5:1005–9.
  • Cappoen D, Jacobs J, Nguyen Van T, et al. Straightforward palladium-mediated synthesis and biological evaluation of benzo[j]phenanthridine-7,12-diones as anti-tuberculosis agents. Eur J Med Chem 2012;48:57–68.
  • Claes P, Cappoen D, Mbala BM, et al. Synthesis and antimycobacterial activity of analogues of the bioactive natural products sampangine and cleistopholine. Eur J Med Chem 2013;67:98–110.
  • Cappoen D, Claes P, Jacobs J, et al. 1,2,3,4,8,9,10,11-octahydrobenzo[j]phenanthridine-7,12-diones as new leads against Mycobacterium tuberculosis. J Med Chem 2014;57:2895–907.
  • Claes P, Cappoen D, Uythethofken C, et al. 2,4-Dialkyl-8,9,10,11-tetrahydrobenzo[g]pyrimido[4,5-c]isoquinoline-1,3,7,12(2H,4H)-tetraones as new leads against Mycobacterium tuberculosis. Eur J Med Chem 2014;77:409–21.
  • Dias DA, Urban S, Roessner U. A historical overview of natural products in drug discovery. Metabolites 2012;2:303–36.
  • Strohl WR. The role of natural products in a modern drug discovery program. Drug Discov Today 2000;5:39–41.
  • Ulubelen A. Cardioactive and antibacterial terpenoids from some Salvia species. Phytochemistry 2003;64:395–9.
  • Somer NU, Sarikaya B, Erac B, et al. Chemical composition and antimicrobial activity of essential oils from the aerial parts of Salvia pinnata L. Rec Nat Prod 2015;9:614–8.
  • Ulubelen A, Topcu G, Johansson CB. Norditerpenoids and diterpenoids from Salvia multicaulis with antituberculous activity. J Nat Prod 1997;60:1275–80.
  • Wu YB, Ni ZY, Shi QW, et al. Constituents from Salvia species and their biological activities. Chem Rev 2012;112:5967–6026.
  • Hatipoglu S, Zorlu D, Dirmenci NT, et al. Determination of volatile organic compounds in fourty five Salvia species by thermal desorption-GC-MS technique. Rec Nat Prod 2016;10:659–700.
  • Wang X, Wei Y, Yuan S, et al. Potential anticancer activity of tanshinone IIA against human breast cancer. Int J Cancer 2005;116:799–807.
  • Chang HM, Chui KY, Tan FW, et al. Structure-activity relationship of miltirone, an active central benzodiazepine receptor ligand isolated from Salvia miltiorrhiza Bunge (Danshen). J Med Chem 1991;34:1675–92.
  • Seçinti H, Burmaoğlu S, Altundaş R, Seçen H. Total syntheses of multicaulins via oxidative photocyclization of stilbenes. J Nat Prod 2014;77:2134–7.
  • Sengupta SK, Biswas RN, Bhattacharyya BK. Friedel–Crafts reaction. IV. Synthesis of 7-isopropyl-3-oxo-6-methoxy-1,2,3,9,10,10a-hexahydrophenanthrene. J Indian Chem Soc 1959;36:659–68.
  • Holzgrabe U. Quantitative NMR spectroscopy in pharmaceutical applications. Prog Nucl Magn Reson Spectrosc 2010;57:229–40.
  • Malz F, Jancke H. Validation of quantitative NMR. J Pharm Biomed Anal 2005;38:813–23.
  • Saito T, Ihara T, Koike M, et al. New traceability scheme for the development of international system-traceable persistent organic pollutant reference materials by quantitative nuclear magnetic resonance. Accredit Qual Assur 2009;14:79–86.
  • Bostan MS, Senol M, Cig T, et al. Controlled release of 5-aminosalicylicacid from chitosan based pH and temperature sensitive hydrogels. Int J Biol Macromol 2013;52:177–83.
  • Burnell RH, Caron S. Approach to the synthesis of candelabrone and synthesis of 3,7-diketo-12-hydroxyabieta-8,11,13-triene. Can J Chem 1992;70:1446–54.
  • Smith MB. March’s advanced organic chemistry, 6th ed. New Jersey: Wiley; 2007.
  • Caronna T, Ferrario F, Servi S. Intermolecular and intramolecular phenol phenylation: regioselective synthesis of unsymmetrically substituted biphenyls and 9,10-dihydrophenanthrenes. Tetrahedron Lett 1979;20:657–60.
  • Sokmen A, Gulluce M, Akpulat HA, et al. The in vitro antimicrobial and antioxidant activities of the essential oils and methanol extracts of endemic Thymus spathulifolius. Food Control 2004;15:627–34.

Related research

People also read lists articles that other readers of this article have read.

Recommended articles lists articles that we recommend and is powered by our AI driven recommendation engine.

Cited by lists all citing articles based on Crossref citations.
Articles with the Crossref icon will open in a new tab.