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Miscellaneous

HIV-1 protease inhibitors in development

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Pages 387-395 | Published online: 24 Feb 2005

Bibliography

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  • ••The first demonstration of PI cross-resistance.
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  • ••A seminal paper introducing the concept ofPI genetic barrier.
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  • •A paper which highlights the potential pharmacological pressure by a PI even after therapeutical shift to another.
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  • ••A pivotal paper which relates the clinicaloutcome with the phenotypic resistance at baseline.
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  • •The first description of the new antiretroviral tipranavir.
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  • •An interesting paper described the emergence of specific mutations induced by BMS-232632.
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