Dissolution evaluation in vitro and bioavailability in vivo of self-microemulsifying drug delivery systems for pH-sensitive drug loratadine

References

• Amidon GL, Lennernas H, Shah VP, Crison JR. A theoretical basis for a biopharmaceutic drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability. Pharm Res, 1995;12:413–20
   PubMed Web of Science ®Google Scholar
• Arida AL, Al-Tabakha MM, Hamoury HA. Improving the high variable bioavailability of griseofulvin by SEDDS. Chem Pharm Bull, 2007;55:1713–19
   PubMed Web of Science ®Google Scholar
• Baird JA, Taylor LS. Evaluation and modeling of the eutectic composition of various drug-polyethylene glycol solid dispersions. Pharm Dev Technol, 2010;16:201–11
   PubMed Web of Science ®Google Scholar
• Banerji A, Long AA, Camargo CA. Diphenhydramine versus nonsedating antihistamines for acute allergic reactions: A literature review. Allergy Asthma Proc, 2007;28:418–26
   PubMed Web of Science ®Google Scholar
• Capek I. Degradation of kinetically-stable o/w emulsions. Adv Colloid Interface Sci, 2004;107:125–55
   PubMed Web of Science ®Google Scholar
• Constantinides PP, Scalart JP. Formulation and physical characterization of water-in-oil microemulsions containing long-versus medium-chain glycerides. Int J Pharm, 1997;158:57–68
   Web of Science ®Google Scholar
• Constantinides PP. Lipid microemulsions for improving drug dissolution and oral absorption: physical and biopharmaceutical aspects. Pharm Res, 1995;12:1561–72
   PubMed Web of Science ®Google Scholar
• Costa P, Lobo JMS. Modeling and comparison of dissolution profiles. Eur J Pharm Sci, 2001;13:123–33
   PubMed Web of Science ®Google Scholar
• Frizon F, Eloy JDO, Donaduzzi CM, Mitsui ML, Marchetti JM. Dissolution rate enhancement of loratadine in polyvinylpyrrolidone K-30 solid dispersions by solvent methods. Powder Technol, 2013;235:532–9
   Web of Science ®Google Scholar
• Gao P, Morozowich W. Development of supersaturatable self-emulsifying drug delivery system formulations for improving the oral absorption of poorly soluble drugs. Expert Opin Drug Deliv, 2006;3:97–110
   PubMedGoogle Scholar
• Gursoy RN, Benita S. Self-emulsifying drug delivery systems (SEDDS) for improved oral delivery of lipophilic drugs. Biomed Pharmacother, 2004;58:173–82
   PubMed Web of Science ®Google Scholar
• Hong J, Kim J, Song Y, Park J, Kim CK. A new self emulsifying formulation of itraconazole with improved dissolution and oral absorption. J Control Release, 2006;110:332–8
   PubMed Web of Science ®Google Scholar
• Jackson MJ. 1987. Drug transport across gastrointestinal epithelial. Physiology of the gastrointestinal tract. New York: Rave Press, pp. 1597–621
   Google Scholar
• Khan MZI, Rausl D, Zanoski R, Zidar S, Mikulcic JH, Krizmanic L, Eskinja M, Mildner B, Knezevic Z. Classification of loratadine based on the biopharmaceutics drug classification concept and possible in vitro–in vivo correlation. Biol Pharm Bull, 2004;27:1630–5
   PubMed Web of Science ®Google Scholar
• Lawrence MJ, Rees GD. Microemulsion-based media as novel drug delivery systems. Adv Drug Deliv Rev, 2000;45:89–121
   PubMed Web of Science ®Google Scholar
• Li J, Hu Y, Qin FH, Lin Y. Preparation and quality evaluation of loratadine self-emulsifying drug delivery system. Cent South Pharm, 2008;6: 414–16
   Google Scholar
• Lobenberg R, Amidon, GL. Modern bioavailability, bioequivalence and biopharmaceutics classification system new scientific approaches to international regulatory standards. Eur J Pharm Biopharm, 2000;50:3–12
   PubMed Web of Science ®Google Scholar
• Nacsa A, Berkesi O, Szabo-Revesz P, Aigner Z. Achievement of pH-independence of poorly-soluble, ionizable loratadine by inclusion complex formation with dimethyl-β-cyclodextrin. J Incl Phenom Macrocycl Chem, 2009;64:249–54
   Web of Science ®Google Scholar
• Papadopoulou V, Kosmidis K, Vlachou M, Mcheras P. On the use of the Weibull function for the discernment of drug release mechanisms. Int J Pharm, 2006;309:44–50
   PubMed Web of Science ®Google Scholar
• Patil P, Paradkar A. Porous polystyrene beads as carriers for self-emulsifying system containing loratadine. AAPS PharmSciTech, 2006;7:E1–7
   PubMed Web of Science ®Google Scholar
• Pedersen PV, Myrick JW. Versatile kinetic approach to analysis of dissolution data. J Pharm Sci, 1978;67:1450–5
   PubMed Web of Science ®Google Scholar
• Popovic G, Cakar M, Agbaba D. Acid–base equilibria and solubility of loratadine and desloratadine in water and micellar media. J Pharm Biomed Anal, 2009;49:42–7
   PubMed Web of Science ®Google Scholar
• Porter CJH, Pouton CW, Cuine JF, Charman WN. Enhancing intestinal drug solubilisation using lipid-based delivery systems. Adv Drug Deliv Rev, 2008;60:673–91
   PubMed Web of Science ®Google Scholar
• Pouton CW. Self-emulsifying drug delivery systems: Assessment of the efficiency of emulsification. Int J Pharm, 1985;27:335–48
   Web of Science ®Google Scholar
• Pouton CW. Lipid formulations for oral administration of drugs: Nonemulsifying, self-emulsifying and ‘self-microemulsifying’ drug delivery systems. Eur J Pharm Sci, 2000;11:S93–8
   PubMed Web of Science ®Google Scholar
• Reiss H. Entropy-induced dispersion of bulk liquids. J Colloid Interface Sci, 1975;53:61–70
   Web of Science ®Google Scholar
• Robinson JR. Introduction: Semi-solid formulations for oral drug delivery. Bull Tech Gattefosse, 1996;89:11–13
   Google Scholar
• Szabados-Nacsa A, Sipos P, Mandity T, Mandity I, Blazso G, Balogh A, Szabo-Revesz P, Aigner Z. Physico-chemical characterization and in vitro/in vivo evaluation of loratadine: dimethyl-β-cyclodextrin inclusion complexes. J Pharm Biomed Anal, 2011;55:294–300
   PubMed Web of Science ®Google Scholar
• Tang JL, Sun J, He ZG. Self-emulsifying drug delivery systems: Strategy for improving oral delivery of poorly soluble drugs. Curr Drug Ther, 2007;2:85–93
   Google Scholar
• Walsh GM. Second-generation antihistamines in asthma therapy: Is there a protective effect? Am J Respir Med, 2002;1:27–34
   PubMedGoogle Scholar
• Yamaoka K, Nakagawa T, Uno T. Application of akaike,s information criterion (AIC), in the evaluation of linear pharmacokinetic equations. J Pharmacokin Biopharm, 1978;6:165–75
   PubMedGoogle Scholar