Formulation of spray congealed microparticles with self-emulsifying ability for enhanced glibenclamide dissolution performance

References

• Albertini B, Passerini N, Di Sabatino M, Monti D, Burgalassi S, Chetoni P, Rodriguez L. Poloxamer 407 microspheres for orotransmucosal drug delivery. Part I: Formulation, manufacturing and characterization. Int J Pharm, 2010;399:71–9
   PubMed Web of Science ®Google Scholar
• Albertini B, Passerini N, Di Sabatino M, Vitali B, Brigidi P, Rodriguez L. Polymer-lipid based mucoadhesive microspheres prepared by spray-congealing for the vaginal delivery of econazole nitrate. Eur J Pharm Sci, 2009;36:591–601
   PubMed Web of Science ®Google Scholar
• Balakrishnan P, Lee BJ, Oh DH, Kim JO, Hong MJ, Jee JP, Kim JA, Yoo BK, Woo JS, Yong CS, Choi HG. Enhanced oral bioavailability of dexibuprofen by a novel solid self-emulsifying drug delivery system (SEDDS). Eur J Pharm Biophar, 2009;72:539–45
   PubMed Web of Science ®Google Scholar
• Blagden N, de Matas M, Gavan PT, York P. Crystal engineering of active pharmaceutical ingredients to improve solubility and dissolution rates. Adv Drug Del Rev, 2007;59:617–30
   PubMed Web of Science ®Google Scholar
• Brewster ME, Loftsson T. Cyclodextrins as pharmaceutical solubilizers. Adv Drug Del Rev, 2007;59:645–66
   PubMed Web of Science ®Google Scholar
• Franceschinis E, Voinovich D, Grassi M, Perissutti B, Filipovic-Grcicc J, Martinac A, Meriani-Merloa F. Self-emulsifying pellets prepared by wet granulation in high-shear mixer: Influence of formulation variables and preliminary study on the in vitro absorption. Int J Pharm, 2005;291:87–97
   PubMed Web of Science ®Google Scholar
• Gupta S, Kesarla R, Omri A. Formulation strategies to improve the bioavailability of poorly absorbed drugs with special emphasis on self-emulsifying systems. ISRN Pharmaceut, 2013;2013:1–16
   Google Scholar
• Hussain SIF, Badawy MA. Microenvironmental pH modulation in solid dosage forms. J Pharm Sci, 2007;96:948–59
   PubMed Web of Science ®Google Scholar
• Ito Y, Kusawake T, Ishida M, Tawa RI, Shibata N, Takada K. Oral solid gentamicin preparation using emulsifier and adsorbent. J Control Release, 2005;105:23–31
   PubMed Web of Science ®Google Scholar
• Jung MS, Kim JS, Kim MS, Alhalaweh A, Cho W, Hwang SJ, Velaga SP. Bioavailability of indomethacin-saccharin cocrystals. J Pharm Pharmacol, 2010;62:1560–68
   PubMed Web of Science ®Google Scholar
• Kawabata Y, Wada K, Nakatani M, Yamada S, Onoue S. Formulation design for poorly water-soluble drugs based on biopharmaceutics classification system: Basic approaches and practical applications. Int J Pharm, 2011;420:1–10
   PubMed Web of Science ®Google Scholar
• Kohli K, Chopra S, Dhar D, Arora S, Khar RK. Self-emulsifying drug delivery systems: An approach to enhance oral bioavailability. Drug Disc Today, 2010;15:958–65
   PubMed Web of Science ®Google Scholar
• Martena V, Censi R, Hoti E, Malaj L, Di Martino P. Preparation of glibenclamide nanocrystals by a simple laboratory scale ultra cryo-milling. J Nanopart Res, 2013;15:1712. DOI: 10.1007/s11051-013-1712-4
   Web of Science ®Google Scholar
• Milovic M, Djuris J, Djekic L, Vasiljevic D, Ibric S. Characterization and evaluation of solid self-microemulsifying drug delivery systems with porous carriers as system for improved carbamazepine release. Int J Pharm, 2012;436:58–65
   PubMed Web of Science ®Google Scholar
• Miyako Y, Khalef N, Matsuzaki K, Pinal R. Solubility enhancement of hydrophobic compounds by cosolvents: Role of solute hydrophobicity on the solubilization effect. Int J Pharm, 2010;393:48–54
   PubMed Web of Science ®Google Scholar
• Passerini N, Albertini B, Perissutti B, Rodriguez L. Evaluation of melt granulation and ultrasonic spray congealing as techniques to enhance the dissolution of praziquantel. Int J Pharm, 2006;318:92–102
   PubMed Web of Science ®Google Scholar
• Passerini N, Qi S, Albertini B, Grassi M, Rodriguez L, Craig DQM. Solid lipid microparticles produced by spray congealing: Influence of the atomizer on microparticle characteristics and mathematical modeling of the drug release. J Pharm Sci, 2010;99:916–31
   PubMed Web of Science ®Google Scholar
• Pouton CW, Porter CJ. Formulation of lipid-based delivery systems for oral administration: Materials, methods and strategies. Adv Drug Del Rev, 2008;60:625–37
   PubMed Web of Science ®Google Scholar
• Rehder S, Sakmann A, Rades T, Leopold CS. Thermal degradation of amorphous glibenclamide. Eur J Pharm Biopharm, 2012;80:203–8
   PubMed Web of Science ®Google Scholar
• Serajuddin AT. Salt formation to improve drug solubility. Adv Drug Del Rev, 2007;59:603–16
   PubMed Web of Science ®Google Scholar
• Shah AV, Serajuddin AT. Development of solid self-emulsifying drug delivery system (SEDDS) I: Use of poloxamer 188 as both solidifying and emulsifying agent for lipids. Pharm Res, 2012;29:2187–32
   Google Scholar
• Shanmugam S, Baskaran R, Balakrishnan PR, Thapa P, Yong CS, Yoo BK. Solid self-nanoemulsifying drug delivery system (S-SNEDDS) containing phosphatidylcholine for enhanced bioavailability of highly lipophilic bioactive carotenoid lutein. Eur J Pharm Biopharm, 2011;79:250–57
   PubMed Web of Science ®Google Scholar
• Shegokar R, Müller RH. Nanocrystals: Industrially feasible multifunctional formulation technology for poorly soluble actives. Int J Pharm, 2010;399:129–39
   PubMed Web of Science ®Google Scholar
• Singh SK, Srinivasan KK, Gowthamarajan K, Prakash D, Gaikwad NB, Singare DS. Influence of formulation parameters on dissolution rate enhancement of glyburide using liquisolid technique. Drug Dev Ind Pharm, 2012;2112:1–10
   Google Scholar
• Singh SK, Srinivasan KK, Gowthamarajan K, Singare DS, Prakash D, Gaikwad NB. Investigation of preparation parameters of nanosuspension by top-down media milling to improve the dissolution of poorly water-soluble glyburide. Eur J Pharm Biopharm, 2011;78:441–6
   PubMed Web of Science ®Google Scholar
• Singh SK, Verma PRP, Razdan B. Glibenclamide-loaded self-nanoemulsifying drug delivery system: Development and characterization. Drug Dev Ind Pharm, 2010;36:933–45
   PubMed Web of Science ®Google Scholar
• Tang B, Cheng G, Gu JC, Xu CH. Development of solid self-emulsifying drug delivery systems: Preparation techniques and dosage forms. Drug Disc Today, 2008;13:606–12
   PubMed Web of Science ®Google Scholar
• Tashtoush BM, Al-Qashi ZS, Najib NM. In vitro and in vivo evaluation of glibenclamide in solid dispersion systems. Drug Dev Ind Pharm, 2004;30:601–7
   PubMed Web of Science ®Google Scholar
• Vasconcelos T, Sarmento B, Costa P. Solid dispersions as strategy to improve oral bioavailability of poor water soluble drugs. Drug Disc Today, 2007;12:1068–75
   PubMed Web of Science ®Google Scholar
• Xiao Y, Wang S, Chen Y, Ping Q. Self-emulsifying bifendate pellets: Preparation, characterization and oral bioavailability in rats. Drug Dev Ind Pharm, 2013;39:724–32
   PubMed Web of Science ®Google Scholar
• Zoeller T, Dressman JRB, Klein S. Application of a ternary HP-beta-CD-complex approach to improve the dissolution performance of a poorly soluble weak acid under biorelevant conditions. Int J Pharm, 2012;430:176–83
   PubMed Web of Science ®Google Scholar