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Research Article

Development of reconstitutable suspensions containing diclofenac sodium-loaded microspheres for pediatric delivery

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Pages 317-328 | Received 25 May 2014, Accepted 02 Feb 2015, Published online: 08 Jul 2015

References

  • Al-Kahtani Ahmed A, Bhojya Naik HS, Sherigara BS. Synthesis and characterization of chitosan-based pH-sensitive semi-interpenetrating network microspheres for controlled release of diclofenac sodium. Carbohydr Res, 2009;344(5):699–706
  • Bolourtchian N, Karimi K, Aboofazeli R. Preparation and characterization of ibuprofen microspheres. J Microencapsulation, 2005;22(5):529–38
  • Castelli F, Messina C, Sarpietro MG, Pignatello R, Puglisi G. Flurbiprofen release from Eudragit RS and RL aqueous nanosus-pensions: A kinetic study by DSC and dialysis experiments. AAPS Pharm Sci Tech, 2002;3:1–8
  • Chuasuwan B, Binjesoh V, Polli JE, Zhang H, Amidon GL, Junginger HE, Midha KK, Shah VP, Stavchansky S, Dressman JB, Barends DM. Biowaiver monographs for immediate release solid oral dosage forms: Diclofenac sodium and diclofenac potassium. J Pharm Sci, 2009;98(4):1206–19
  • Cui F, Cun D, Tao A, Yang M, Shi K, Zhao M, Guan Y. Preparation and characterization of melittin-loaded poly (dl-lactic acid) or poly (dl-lactic-co-glycolic acid) microspheres made by double emulsion method. J Control Release, 2005;107:310–19
  • Deng XM, Li XH, Yuan ML, Xiong CD, Huang ZT, Jia WX, Zhang YH. Optimization of preparative conditions for poly-dl-lactide-polyethylene glycol microspheres with entrapped Vibrio cholera antigens. J Control Release, 1999;58(2):123–31
  • Devrim B, Bozkır A, Canefe K. Preparation and evaluation of PLGA microparticles as carrier for the pulmonary delivery of rhIL-2: I. Effects of some formulation parameters on microparticle characteristics. J Microencapsulation, 2011a;28(6):582–94
  • Devrim B, Bozkir A, Canefe K. Formulation and evaluation of reconstitutable suspensions containing ibuprofen-loaded Eudragit microspheres. Acta Pol Pharm, 2011b;68(4):593–9
  • Devrim B, Bozkır A. Preparation and evaluation of double-walled microparticles prepared with a modified water-in-oil-in-oil-in-water (w1/o/o/w3) method. J Microencapsulation, 2013;30(8):741–54
  • Donnelly RF, Pascuet E, Ma C, Vaillancourt R. Stability of diclofenac sodium oral suspensions packaged in amber polyvinyl chloride bottles. Can J Hosp Pharm, 2010;63(1):25–30
  • Elkheshen SA, Abd El-Gawad NA, Badawi AA. Factorial design and computer optimization of a reconstitutable suspension of erythromycin ethylsuccinate. Pharm Ind, 1997;59:439–43
  • El-Leithy ES, Shaker DS, Ghorab MK, Abdel-Rashid RS. Optimization and characterization of diclofenac sodium microspheres prepared by a modified coacervation method. Drug Discov Ther, 2010;4(3):208–16
  • Ferrero C, Massuelle D, Doelker E. Towards elucidation of the drug release mechanism from compressed hydrophilic matrices made of cellulose ethers. II. Evaluation of a possible swelling-controlled drug release mechanism using dimensionless analysis. J Control Release, 2010;141:223–33
  • Fini A, Cavallari C, Rabasco Alvarez AM, Rodriguez MG. Diclofenac salts, part 6: Release from lipid microspheres. J Pharm Sci, 2011;100(8):3482–94
  • Freitas S, Merkle HP, Gander B. Microencapsulation by solvent extraction/evaporation: Reviewing the state of the art of microspheres preparation process technology. J Control Release, 2005;102:313–32
  • Garcia-Ochoa F, Santos VE, Casas JA, Gomez E. 2000. Xanthan gum: Production, recovery, and properties. Biotechnol Adv, 2000;18:549–79
  • Gonzalez-Rodrıguez ML, Maestrelli F, Mura P, Rabasco AM. In vitro release of sodium diclofenac from a central core matrix tablet aimed for colonic drug delivery. Eur J Pharm Sci, 2003;20:125–31
  • Hickey T, Kreutzer D, Burgess DJ, Moussy F. Dexamethasone/PLGA microspheres for continuous delivery of an anti-inflammatory drug for implantable medical devices. Biomaterials, 2002;23:1649–56
  • Hua S, Yang H, Li Q, Zhang J, Wang A. pH-sensitive sodium alginate/calcined hydrotalcite hybrid beads for controlled release of diclofenac sodium. Drug Dev Ind Pharm, 2012;38(6):728–34
  • Jiao YY, Ubrich N, Hoffart V, Marchand-Arvier M, Vigneron C, Hoffman M, Maincent P. Preparation and characterization of heparin-loaded polymeric microparticles. Drug Dev Ind Pharm, 2002;28(8):1033–41
  • Kamila MM, Mondal N, Ghosh LK, Gupta BK. Multiunit floating drug delivery system of rosiglitazone maleate: Development, characterization, statistical optimization of drug release and in vivo evaluation. AAPS PharmSciTech, 2009;10(3):887–99
  • Katzbauer B. Properties and applications of xanthan gum. Polym Degradation Stab, 1998;59:81–4
  • Kishori LD, Nilima AT, Paraag SG. Formulation and development of tinidazole microspheres for colon targeted drug delivery system. J Pharm Res, 2013;5:158–60
  • Labouta HI, El Khordaguı LK, Molokhıa AM, Ghaly GM. Multivariate modeling of encapsulation and release of an ionizable drug from polymer microspheres. J Pharm Sci, 2009;98(12):4603–15
  • Lai F, Sinico C, Ennas G, Marongiu F, Marongiu G, Fadda AM. Diclofenac nanosuspensions: Influence of preparation procedure and crystal form on drug dissolution behaviour. Int J Pharm, 2009;373(1–2):124–32
  • Lee J, Park TG, Choi H. Effect of formulation and processing variables on the characteristics of microspheres for water-soluble drugs prepared by w/o/o double emulsion solvent diffusion method. Int J Pharm, 2000;196:75–83
  • Leonardi D, Salomón CJ, Lamas MC, Olivieri AC. Development of novelfor mulations for Chagas’ disease: Optimization of benznidazole chitosan microparticles based on artificial neural networks. Int J Pharm, 2009;367:140–7
  • Lewis L, Boni RL, Adeyeye CM. The physical and chemical stability of suspensions of sustained-release diclofenac microspheres. J Microencapsulation, 1998;15(5):555–67
  • Mahboubian A, Hashemein SK, Moghadam S, Atyabi F, Dinarvand R. Preparation and in-vitro evaluation of controlled release PLGA microparticles containing triptoreline. Iran J Pharm Res, 2010;9(4):369–78
  • Mao S, Xu J, Cai C, Germershaus O, Schaper A, Kissel T. Effect of wow process parameters on morphology and burst release of FITC-dextran loaded PLGA microspheres. Int J Pharm, 2007;334:137–48
  • Mateovic-Rojnik T, Frlan R, Bogataj M, Bukovec P, Mrhar A. Effect of preparation temperature in solvent evaporation process on Eudragit RS microsphere properties. Chem Pharm Bull, 2005;53:143–6
  • Moffat AC, Osselton DM, Widdop B. 2004. Clark’s analysis of drugs and poisons. London: Pharmaceutical Press
  • Momoh MA, Kenechukwu FC, Adedokun MO, Odo CE, Attama AA. Pharmacodynamics of diclofenac from novel Eudragit entrapped microspheres. Drug Deliv, 2014;21(3):193–203
  • Nafea EH, El-Massik MA, El-Khordagui LK, Marei MK, Khalafallah NM. Alendronate PLGA microspheres with high loading efficiency for dental applications. J Microencapsulation, 2007;24(6):525–38
  • Nath B, Kantanath L, Kumar P. Preparation and in vitro dissolution profile of zidovudine loaded microspheres made of Eudragit RS 100, RL 100 and their combinations. Acta Pol Pharm, 2011;68(3):409–15
  • Nayak AK, Pal D. Development of pH-sensitive tamarind seed polysaccharide–alginate composite beads for controlled diclofenac sodium delivery using response surface methodology. Int J Biol Macromol, 2011;49(4):784–93
  • Ntawukulilyayo JD, De Smedt SC, Demeester J, Remon JP. Stabilisation of suspensions using sucrose esters and low substituted n-octenylsuccinate starch–xanthan gum associations. Int J Pharm, 1996;128:73–9
  • Omari DM, Sallam A, Abd-Elbary A, El-Samaligy M. Lactic acid-induced modifications in films of Eudragit RL and RS aqueous dispersions. Int J Pharm, 2004;274:85–96
  • Perugini P, Genta I, Conti B, Modena T, Pavanetto F. Long-term release of clodronate from biodegradable microspheres. AAPS PharmSciTech, 2001;2:E10
  • Piao H, Kamiya N, Watanabe J, Yokoyama H, Hirata A, Fujii T, Shimizu I, Ito S, Goto M. Oral delivery of diclofenac sodium using a novel solid-in-oil suspension. Int J Pharm, 2006;313(1–2):159–62
  • Pongjanyakul T, Puttipipatkhachorn S. Polymer-magnesium aluminum silicate composite dispersions for improved physical stability of acetaminophen suspensions. AAPS Pharm Sci Tech, 2009;10(2):346–54
  • Provenza N, Calpena AC, Mallandrich M, Halbaut L, Clares B. Design and physicochemical stability studies of paediatric oral formulations of sildenafil. Int J Pharm, 2014;460(1–2):234–9
  • Ramasamy T, Ruttala HB, Shanmugam S, Umadevi SK. Eudragit-coated aceclofenac-loaded pectin microspheres in chronopharmacological treatment of rheumatoid arthritis. Drug Deliv, 2013;20(2):65–77
  • Sahoo SK, Panyam J, Prabha S, Labhasetwar V. Residual polyvinyl alcohol associated with poly (d,l-lactide-co-glycolide) nanoparticles affects their physical properties and cellular uptake. J Control Release, 2002;82:105–14
  • Shinde UA, Shete JN, Nair HA, Singh KH. Eudragit RL100 based microspheres for ocular administration of azelastine hydrochloride. J Microencapsulation, 2012;29(6):511–19
  • Sipos P, Szucs M, Szabó A, Eros I, Szabó-Révész P. An assessment of the interactions between diclofenac sodium and ammonio methacrylate copolymer using thermal analysis and Raman spectroscopy. J Pharm Biomed Anal, 2008;46(2):288–94
  • Song X, Song S-K, Zhao P, Wei L-M, Jiao H-S. β-Methasone-containing biodegradable poly(lactide-coglycolide) acid microspheres for intraarticular injection: Effect of formulation parameters on characteristics and in vitro release. Pharm Dev Technol, 2013;18(5):1220–9
  • Swarbrick J. 2007. Encyclopedia of pharmaceutical technology. New York: Informa Heathcare
  • Tiwary AK, Panpalia GM. Influence of crystal habit on trimethoprim suspension formulation. Pharm Res, 1999;16(2):261–5
  • Tudja P, Khan MZ, Mestrović E, Horvat M, Golja P. Thermal behaviour of diclofenac sodium: Decomposition and melting characteristics. Chem Pharm Bull, 2001;49(10):1245–50
  • Vladisavljevi’c GT, Schubert H. Influence of process parameters on droplet size distribution in SPG membrane emulsification and stability of prepared emulsion droplets. J Membr Sci, 2003;225:15–23
  • Wang Q, Xie X, Zhang X, Zhang J, Wang A. Preparation and swelling properties of pH-sensitive composite hydrogel beads based on chitosan-g-poly (acrylic acid)/vermiculite and sodium alginate for diclofenac controlled release. Int J Biol Macromol, 2010;46(3):356–62
  • Weidenauer U, Bodmer D, Kissel T. Microencapsulation of hydrophilic drug substances using biodegradable polyesters. Part I: Evaluation of different techniques for the encapsulation of pamidronate di-sodium salt. J Microencapsulation, 2003;20:509–24
  • Yang Y-Y, Chung T-S, Ng NP. Morphology, drug distribution, and in vitro release profiles of biodegradable polymeric microspheres containing protein fabricated by double-emulsion solvent extraction/evaporation method. Biomaterials, 2001;22:231–41

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