Effects of Oleic Acid on the Corneal Permeability of Compounds and Evaluation of its Ocular Irritation of Rabbit Eyes

References

• Rawas-Qalaji M, Williams C. Advances in ocular drug delivery. Curr Eye Res 2012;37:345–356
   PubMed Web of Science ®Google Scholar
• Eljarrat-Binstock E, Pe’er J, Domb A. New techniques for drug delivery to the posterior eye segment. Pharm Res 2010;27:530–543
   PubMed Web of Science ®Google Scholar
• Xu X, Yu N, Bai Z, Xun Y, Jin D, Li Z, Cui H. Effect of menthol on ocular drug delivery. Graefes Arch Clin Exp Ophthalmol 2011;249:1503–1510
   PubMedGoogle Scholar
• Qi HP, Wei SQ, Gao XC, Yu NN, Hu WZ, Bi S, Cui H. Ursodeoxycholic acid prevents selenite-induced oxidative stress and alleviates cataract formation: in vitro and in vivo studies. Mol Vis 2012;18:151–160
   PubMed Web of Science ®Google Scholar
• Achouri D, Alhanout K, Piccerelle P, Andrieu V. Recent advances in ocular drug delivery. Drug Dev Ind Pharm 2013;39:1599–1617
   PubMed Web of Science ®Google Scholar
• Lee SS, Hughes PM, Robinson M. Recent advances in drug delivery systems for treating ocular complications of systemic diseases. Curr Opin Ophthalmol 2009;20:511–519
   PubMed Web of Science ®Google Scholar
• Liu R, Liu Z, Zhang C, Zhang B. Gelucire44/14 as a novel absorption enhancer for drugs with different hydrophilicities: in vitro and in vivo improvement on transcorneal permeation. J Pharm Sci 2011;100:3186–3195
   PubMed Web of Science ®Google Scholar
• Kaur IP, Smitha R. Penetration enhancers and ocular bioadhesives: two new avenues for ophthalmic drug delivery. Drug Dev Ind Pharm 2002;28:353–369
   PubMed Web of Science ®Google Scholar
• Majumdar S, Hippalgaonkar K, Repka M. Effect of chitosan, benzalkonium chloride and ethylenediaminetetraacetic acid on permeation of acyclovir across isolated rabbit cornea. Int J Pharm 2008;348:175–178
   PubMed Web of Science ®Google Scholar
• Moreira TS, de Sousa VP, Pierre M. Influence of oleic acid on the rheology and in vitro release of lumiracoxib from poloxamer gels. J Pharm Pharm Sci 2010;13:286–302
   PubMed Web of Science ®Google Scholar
• da Silva ER, de Freitas ZM, deGitirana LB, Ricci-Júnior E. Improving the topical delivery of zinc phthalocyanine using oleic acid as a penetration enhancer: in vitro permeation and retention. Drug Dev Ind Pharm 2011;37:569–575
   PubMed Web of Science ®Google Scholar
• Ochalek M, Podhaisky H, Ruettinger HH, Neubert RH, Wohlrab J. SC lipid model membranes designed for studying impact of ceramide species on drug diffusion and permeation, part III: influence of penetration enhancer on diffusion and permeation of model drugs. Int J Pharm 2012;436:206–213
   PubMedGoogle Scholar
• Sztriha L, Betz A. Oleic acid reversibly opens the blood–brain barrier. Brain Res 1991;550:257–262
   PubMed Web of Science ®Google Scholar
• Dhiman MK, Dhiman A, Sawant K. Transbuccal delivery of 5-fluorouracil: permeation enhancement and pharmacokinetic study. AAPS PharmSciTech 2009;10:258–265
   PubMed Web of Science ®Google Scholar
• Prasanthi D, Lakshmi P. Effect of chemical enhancers in transdermal permeation of alfuzosin hydrochloride. ISRN Pharm 2012;2012:965280
   PubMedGoogle Scholar
• Engelbrecht TN, Schroeter A, Hauss T, Neubert R. Lipophilic penetration enhancers and their impact to the bilayer structure of stratum corneum lipid model membranes: neutron diffraction studies based on the example oleic acid. Biochim Biophys Acta 2011;1808:2798–2809
   PubMed Web of Science ®Google Scholar
• Bloemen M, Brullot W, Luong TT, Geukens N, Gils A, Verbiest T. Improved functionalization of oleic acid-coated iron oxide nanoparticles for biomedical applications. J Nanopart Res 2012;14:1100
   PubMed Web of Science ®Google Scholar
• Zhang T, Zheng Y, Peng Q, Cao X, Gong T, Zhang Z. A novel submicron emulsion system loaded with vincristine-oleic acid ion-pair complex with improved anticancer effect: in vitro and in vivo studies. Int J Nanomedicine 2013;8:1185–1196
   PubMed Web of Science ®Google Scholar
• Monti D, Chetoni P, Burgalassi S, Najarro M, Saettone M. Increased corneal hydration induced by potential ocular penetration enhancers: assessment bydifferential scanning calorimetry (DSC) and by desiccation. Int J Pharm 2002;232:139–147
   PubMed Web of Science ®Google Scholar
• Draize JH, Woodard G, Calvery H. Methods for the study of irritation and toxicity of substances applied topically to the skin and mucous membranes. J Pharmacol Exp Ther 1944;82:377–390
   Web of Science ®Google Scholar
• Salama NN, Eddington ND, Fasano A. Tight junction modulation and its relationship to drug delivery. Adv Drug Deliv Rev 2006;58:15–28
   PubMed Web of Science ®Google Scholar
• Sahoo SK, Dilnawaz F, Krishnakumar S. Nanotechnology in ocular drug delivery. Drug Discov Today 2008;13:144–151
   PubMed Web of Science ®Google Scholar
• Afouna MI, Khedr A, Abdel-Naim AB, Al-Marzoqi A. Influence of various concentrations of terpene-4-ol enhancer and carbopol-934 mucoadhesive upon the in vitro ocular transport and the in vivo intraocular pressure lowering effects of dorzolamide ophthalmic formulations using albino rabbits. J Pharm Sci 2010;99:119–127
   PubMed Web of Science ®Google Scholar
• Qi HP, Gao XC, Zhang LQ, Wei SQ, Bi S, Yang ZC, Cui H. In vitro evaluation of enhancing effect of borneol on transcorneal permeation of compounds with different hydrophilicities and molecular sizes. Eur J Pharmacol 2013;705:20–25
   PubMed Web of Science ®Google Scholar
• Jiang SJ, Zhou X. Examination of the mechanism of oleic acid-induced percutaneous penetration enhancement: an ultrastructural study. Biol Pharm Bull 2003;26:66–68
   PubMed Web of Science ®Google Scholar
• Jiang SJ, Hwang SM, Choi EH, Elias PM, Ahn SK, Lee S. Structural and function effects of oleic acid and iontophoresis on hairless mouse stratum corneum. J Invest Dermatol 2000;114:64–70
   PubMedGoogle Scholar
• Cui CY, Lu WL, Xiao L, Zhang SQ, Huang YB, Li SL, et al. Sublingual delivery of insulin: effects of enhancers on the mucosal lipid fluidity and protein conformation, transport, and in vivo hypoglycemic activity. Biol Pharm Bull 2005;28:2279–2288
   PubMed Web of Science ®Google Scholar
• Zhao H, Lu H, Gong T, Zhang Z. Nanoemulsion loaded with lycobetaine-oleic acid ionic complex physicochemical characteristics, in vitro, in vivo evaluation, and antitumor activity. Inter J Nanomedcine 2013;8:1959–1973
   PubMed Web of Science ®Google Scholar
• Ma L, Kuang K, Smith RW, Rittenband D, Iserovich P, Diecke FPJ, Fischbarg J. Modulation of tight junction properties relevant to fluid transport across rabbit corneal endothelium. Exp Eye Res 2007;84:790–798
   PubMed Web of Science ®Google Scholar
• Fischbarg J, Warshavsky CR, Lim J. Pathways for hydraulically and osmotically-induced water flows across epithelia. Nature 1977;266:71–74
   PubMed Web of Science ®Google Scholar
• Ambati J, Canakis C, Miller JW, Gragoudas E, Edwards A, Weissgold DJ, et al. Diffusion of high molecular weight compounds though sclera. Invest Ophthalmol Vis Sci 2000;41:1181–1185
   PubMed Web of Science ®Google Scholar