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Research Article

Characterising the surface adhesive behavior of tablet tooling components by atomic force microscopy

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Pages 875-885 | Received 11 May 2010, Accepted 02 Dec 2010, Published online: 20 Jan 2011

References

  • Chow K, Tong HH, Lum S, Chow AH. (2008). Engineering of pharmaceutical materials: an industrial perspective. J Pharm Sci, 97:2855–2877.
  • Hickey AJ, Mansour HM, Telko MJ, Xu Z, Smyth HD, Mulder T et al. (2007). Physical characterization of component particles included in dry powder inhalers. I. Strategy review and static characteristics. J Pharm Sci, 96:1282–1301.
  • Roberts CJ. (2005). What can we learn from atomic force microscopy adhesion measurements with single drug particles? Eur J Pharm Sci, 24:153–157.
  • Booth SW, Newton JM. (1987). Experimental investigation of adhesion between powders and surfaces. J Pharm Pharmacol, 39:679–684.
  • King H. (2007). The Practical Guide to Tableting. Victoria, Canada: Trafford Publishing.
  • Toyoshima K, Yasumura M, Ohnishi N, Ueda Y. (1988). Quantitative evolution of tablet sticking by surface roughness measurement. Int J Pharm, 46:211–215.
  • Aljaberi A, Chatterji A, Shah NH, Sandhu HK. (2009). Functional performance of silicified microcrystalline cellulose versus microcrystalline cellulose: a case study. Drug Dev Ind Pharm, 35:1066–1071.
  • Anuar MS, Briscoe BJ. (2009). The elastic relaxation of starch tablets during ejection. Powder Technol, 195:96–104.
  • Lam KK, Newton JM. (1991). Investigation of applied compression on the adhesion of powders to a substrate surface. Powder Technol, 65:167–175.
  • Podczeck F. (1999). Investigations into the reduction of powder adhesion to stainless steel surfaces by surface modification to aid capsule filling. Int J Pharm, 178:93–100.
  • Wang JJ, Li T, Bateman SD, Erck R, Morris KR. (2003). Modeling of adhesion in tablet compression–I. Atomic force microscopy and molecular simulation. J Pharm Sci, 92:798–814.
  • Wang J, Wen H, Desai D. (2010). Lubrication in tablet formulations. Eur J Pharm Biopharm, In press, doi:10.1016/j.ejpb.2010.01.007.
  • Shibata Y, Fujii M, Noda S, Kokudai M, Okada H, Kondoh M et al. (2006). Fluidity and tableting characteristics of a powder solid dispersion of the low melting drugs ketoprofen and ibuprofen with crospovidone. Drug Dev Ind Pharm, 32:449–456.
  • Roberts M, Ford JL, MacLeod GS, Fell JT, Smith GW, Rowe PH. (2003). Effects of surface roughness and chrome plating of punch tips on the sticking tendencies of model ibuprofen formulations. J Pharm Pharmacol, 55:1223–1228.
  • Sabir A, Evans B, Jain S. (2001). Formulation and process optimization to eliminate picking from market image tablets. Int J Pharm, 215:123–135.
  • Wu C-Y, Hancock BC, Mills A, Bentham AC, Best SM, Elliot JA. (2008). Numerical and experimental investigation of capping mechanisms during pharmaceutical tablet compaction. Powder Technol, 181:121–129.
  • Schumann S, Searle GD. (1992). The effects of chromium nitride ION bombardment treatment of tablet tooling on tablet adherence. Drug Dev Ind Pharm, 18:1037–1061.
  • Mitrove A, Augsburger LL. (1980). Adhesion of tablets in a rotary tablet press I. Instrumentation and preliminary study of variables affecting adhesion. Drug Dev Ind Pharm 6:331–377.
  • Bunker M, Davies M, Roberts C. (2005). Towards screening of inhalation formulations: measuring interactions with atomic force microscopy. Expert Opin Drug Deliv, 2:613–624.
  • Begat P, Morton DA, Staniforth JN, Price R. (2004). The cohesive-adhesive balances in dry powder inhaler formulations I: Direct quantification by atomic force microscopy. Pharm Res, 21:1591–1597.
  • Eve JK, Patel N, Luk SY, Ebbens SJ, Roberts CJ. (2002). A study of single drug particle adhesion interactions using atomic force microscopy. Int J Pharm, 238:17–27.
  • Hooton JC, German CS, Allen S, Davies MC, Roberts CJ, Tendler SJ et al. (2004). An atomic force microscopy study of the effect of nanoscale contact geometry and surface chemistry on the adhesion of pharmaceutical particles. Pharm Res, 21:953–961.
  • Hooton JC, Jones MD, Harris H, Shur J, Price R. (2008). The influence of crystal habit on the prediction of dry powder inhalation formulation performance using the cohesive-adhesive force balance approach. Drug Dev Ind Pharm, 34:974–983.
  • Louey MD, Mulvaney P, Stewart PJ. (2001). Characterisation of adhesional properties of lactose carriers using atomic force microscopy. J Pharm Biomed Anal, 25:559–567.
  • Young PM, Price R, Lewis D, Edge S, Traini D. (2003). Under pressure: predicting pressurized metered dose inhaler interactions using the atomic force microscope. J Colloid Interface Sci, 262:298–302.
  • James J, Crean B, Davies M, Toon R, Jinks P, Roberts CJ. (2008). The surface characterisation and comparison of two potential sub-micron, sugar bulking excipients for use in low-dose, suspension formulations in metered dose inhalers. Int J Pharm, 361:209–221.
  • Zhang J, Ebbens S, Chen X, Jin Z, Luk S, Madden C et al. (2006). Determination of the surface free energy of crystalline and amorphous lactose by atomic force microscopy adhesion measurement. Pharm Res, 23:401–407.
  • Masterson VM, Cao X. (2008). Evaluating particle hardness of pharmaceutical solids using AFM nanoindentation. Int J Pharm, 362:163–171.
  • Perkins M, Ebbens SJ, Hayes S, Roberts CJ, Madden CE, Luk SY et al. (2007). Elastic modulus measurements from individual lactose particles using atomic force microscopy. Int J Pharm, 332:168–175.
  • Perkins MC, Bunker M, James J, Rigby-Singleton S, Ledru J, Madden-Smith C et al. (2009). Towards the understanding and prediction of material changes during micronisation using atomic force microscopy. Eur J Pharm Sci, 38:1–8.
  • Bunker MJ, Davies MC, Chen X, James MB, Roberts CJ. (2006). Single particle friction on blister packaging materials used in dry powder inhalers. Eur J Pharm Sci, 29:405–413.
  • Lee J. (2004). Intrinsic adhesion force of lubricants to steel surface. j Pharm Sci, 93:2310–2318.
  • Weber D, Pu Y, Clooney CL. (2008). Quantification of lubricant activity of magnesium stearate by atomic force microscopy. Drug Dev Ind Pharm, 22:1105–1120.
  • Beach ER, Tormoen GW, Drelich J, Han R. (2002). Pull-off force measurements between rough surfaces by atomic force microscopy. J Colloid Interface Sci, 247:84–99.
  • Cooper K, Ohler N, Gupta A, Beaudoin S. (2000). Analysis of Contact Interactions between a Rough Deformable Colloid and a Smooth Substrate. J Colloid Interface Sci, 222:63–74.
  • Götzinger M, Peukert W. (2003). Dispersive forces of particle–surface interactions: direct AFM measurements and modelling. Powder Technology, 130:102–109.
  • Li Q, Rudolph V, Peukert W. (2005). London-van der Waals adhesiveness of rough particles. Powder Technology, 161:248–255.
  • Jones R, Pollock HM, Cleaver JAS, Hodges CS. (2002). Adhesion forces between glass and silicon surfaces in air studied by AFM: Effects of relative humidity, particle size, roughness, and surface treatment. Langmuir, 18:8045–8055.
  • Podczeck F, Newton JM, James MB. (1997). Variations in the adhesion force between a drug and carrier particles as a result of changes in the relative humidity of the air. Int J Pharm, 149:151–160.
  • Xiao X, Qian L. (2000). Investigation humidity dependent capillary force. Langmuir, 16:8153–8158.
  • Bunker MJ, Davies MC, James MB, Roberts CJ. (2007). Direct observation of single particle electrostatic charging by atomic force microscopy. Pharm Res, 24:1165–1169.
  • Butt HJ, Kappl M. (2009). Normal capillary forces. Adv Colloid Interface Sci, 146:48–60.
  • Young PM, Price R, Tobyn MJ, Buttrum M, Dey F. (2003). Investigation into the effect of humidity on drug-drug interactions using the atomic force microscope. J Pharm Sci, 92:815–822.
  • Young PM, Price R, Tobyn MJ, Buttrum M, Dey F. (2004). The influence of relative humidity on the cohesion properties of micronized drugs used in inhalation therapy. J Pharm Sci, 93:753–761.
  • Bérard V, Lesniewska E, Andrès C, Pertuy D, Laroche C, Pourcelot Y. (2002). Dry powder inhaler: influence of humidity on topology and adhesion studied by AFM. Int J Pharm, 232:213–224.
  • Bérard V, Lesniewska E, Andrès C, Pertuy D, Laroche C, Pourcelot Y. (2002). Affinity scale between a carrier and a drug in DPI studied by atomic force microscopy. Int J Pharm, 247:127–137.
  • He M, Blum AS, Aston DE, Buenviaje C, Overney RM, Luginbuhl R. (2001). Critical phenomena of water bridges in nanoasperity contacts. J Chem Phys, 114:1355–1360.
  • Xu L, Lio A, Hu J, Ogletree DF, Salmeron M. (1998). Wetting and capillary phenomena of water on mica. J Phys Chem B, 102:540–548.
  • Islam N, Stewart P, Larson I, Hartley P. (2005). Surface roughness contribution to the adhesion force distribution of salmeterol xinafoate on lactose carriers by atomic force microscopy. J Pharm Sci, 94:1500–1511.
  • Traini D, Young PM, Jones M, Edge S, Price R. (2006). Comparative study of erythritol and lactose monohydrate as carriers for inhalation: atomic force microscopy and in vitro correlation. Eur J Pharm Sci, 27:243–251.
  • Young PM, Cocconi D, Colombo P, Bettini R, Price R, Steele DF et al. (2002). Characterization of a surface modified dry powder inhalation carrier prepared by “particle smoothing”. J Pharm Pharmacol, 54:1339–1344.
  • Rabinovich YI, Adler JJ, Ata A, Singh RK, Moudgil BM. (2000). Adhesion between Nanoscale Rough Surfaces. J Colloid Interface Sci, 232:10–16.
  • Rabinovich YI, Adler JJ, Ata A, Singh RK, Moudgil BM. (2000). Adhesion between Nanoscale Rough Surfaces. J Colloid Interface Sci, 232:17–24.
  • Rumpf H. (1990). Particle Technology. London/New York: Chapman & Hall.
  • Israelachvili JN (1992). Intermolecular and Surface Forces. London: Academic Press.
  • Hutter JL, Bechhoefer J. (1993). Calibration of atomic-force microscope tips. Rev Sci Instrum, 64:1868–1873.
  • Blanchard R. (2009). Personal communication, discussion on the practical application of coated tablet punch faces in industry. IHolland Ltd, Nottingham, UK.
  • Wang J, Qian J, Gao H. (2009). Effects of capillary condensation in adhesion between rough surfaces. Langmuir, 25:11727–11731.
  • Pakarinen OH, Foster AS, Paajanen M, Kalinainen T, Katainen J, Makkonen I, Lahtinen J, Nieminen RM. (2005). Towards an accurate description of the capillary force in nanoparticle-surface interactions. Modelling Simul Mater Sci Eng, 13:1175–1186.

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