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Research Article

Design and development of nanoemulsion drug delivery system of amlodipine besilate for improvement of oral bioavailability

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Pages 907-916 | Received 18 Aug 2010, Accepted 17 Dec 2010, Published online: 14 Mar 2011

References

  • Lawrence MJ, Rees GD. (2000). Microemulsion-based media as novel drug delivery systems. Adv Drug Deliv Rev, 45:89–121.
  • Mustafa G, Iqbal Z, Bansal T, Talegaonkar S. (2009). Preparation and characterization of ultrafine oil in water nano-reservoir systems for improved oral delivery of atorvastatin. Current Nanosci, 5:428–440.
  • Jain NK. (2004). Progress in controlled and novel drug delivery system. New Delhi, India: CBS Publisher and Distributor.
  • Kawakami K, Yoshikawa T, Moroto Y, Kanaoka E, Takahashi K, Nishihara Y, Masuda K. (2007). Microemulsion formulation for enhanced absorption of poorly soluble drugs II. In -vivo study. J Cont Rel, 81:75–82.
  • Shafiq S, Shakeel F, Talegaonkar S, Ahmad FJ, Khar RK, Ali M. (2007). Development and bioavailability assessment of ramipril nanoemulsion formulation. Eur J Pharm Biopharm, 66:227–243.
  • Humphreys A, Boersig C. (2003). Cholesterol drugs dominate. Med Ad News, 22:42–57.
  • Robertson R.M, Robertson D, Hardman JG, Limbird LE, Molinoff PE, Ruddon RW, Gilman AG. (2006). Goodman and Gilman’s: The Pharmacological Basis of Therapeutics, New York: McGraw Hill.
  • McDaid DM, Deasy PB. (1996). Formulation development of a transdermal drug delivery system for amlodipine base. Int J Pharm, 133:71–83.
  • Martindale (2002). The Complete Drug Reference, New York, Pharmaceutical Press.
  • Shafiq S, Shakeel F. (2010). Stability and self-nanoemulsification efficiency of ramipril nanoemulsion containing labrasol and plurol oleique. Clinical Res Reg Affairs., 27:7–12.
  • Shafiq-un-Nabi S, Shakeel F, Talegaonkar S, Ali J, Baboota S, Ahuja A et al. (2007). Formulation development and optimization using nanoemulsion technique: a technical note. AAPS Pharm Sci Tech, 8:E28.
  • Hong JY, Kim JK, Song YK, Park JS, Kim CK. (2006). A new self-emulsifying formulation of itraconazole with improved dissolution and oral absorption. j Control Release, 110:332–338.
  • Vyas SP, Khar RK. (2002). Controlled drug delivery: Concepts and advances. New Delhi, India: Vallabh Prakashan.
  • Kumar M, Misra A, Mishra AK, Mishra P, Pathak K. (2008). Mucoadhesive nanoemulsion-based intranasal drug delivery system of olanzapine for brain targeting. j Drug Target, 16:806–814.
  • Kumar M, Misra A, Babbar AK, Mishra AK, Mishra P, Pathak K. (2008). Intranasal nanoemulsion based brain targeting drug delivery system of risperidone. Int J Pharm, 358:285–291.
  • Kumar M, Pathak K, Misra A. (2008). Formulation and characterization of nanoemulsion based drug delivery of risperidone. Drug Dev Ind Pharm, 35:387–395.
  • Singh SK, Verma PR, Razdan B. (2010). Glibenclamide-loaded self-nanoemulsifying drug delivery system: development and characterization. Drug Dev Ind Pharm, 36:933–945.
  • Roland I, Piel G, Delattre L, Evrard B. (2003). Systematic characterization of oil-in-water emulsions for formulation design. Int J Pharm, 263:85–94.
  • Aulton ME. (2008). Pharmaceutics: The design and manufacture of medicines, New York: Elsevier.
  • Snehalatha M, Venugopal K, Saha RN, Babbar AK, Sharma RK. (2008). Etoposide loaded PLGA and PCL nanoparticles II: biodistribution and pharmacokinetics after radiolabeling with Tc-99m. Drug Deliv, 15:277–287.
  • Craig DQM, Barker SA, Banning D, Booth SW. (1995). An investigation into the mechanisms of self-emulsification using particle size analysis and low frequency dielectric spectroscopy. Int J Pharm, 114:103–110.
  • Peltola S, Saarinen-Savolainen P, Kiesvaara J, Suhonen TM, Urtti A. (2003). Microemulsions for topical delivery of estradiol. Int J Pharm, 254:99–107.
  • El-Laithy HM. (2003). Preparation and physicochemical characterization of dioctyl sodium sulfosuccinate (aerosol OT) microemulsion for oral drug delivery. aaps Pharmscitech, 4:E11.
  • Gao Z, Choi H, Shin H, Park K, Lim S, Hwang K, Kim C. (1998). Physicochemical characterization and evaluation of a microemulsion system for oral delivery of cyclosporine A. Int J Pharm, 161:75–86.
  • Shakeel F, Faisal MS. (2010). Nanoemulsion: a promising tool for solubility and dissolution enhancement of celecoxib. Pharm Dev Technol, 15:53–56.
  • Singh KK, Vingkar SK. (2008). Formulation, antimalarial activity and biodistribution of oral lipid nanoemulsion of primaquine. Int J Pharm, 347:136–143.
  • Aburahma MH, El-Laithy HM, Hamza YS. (2010). Oral bioavailability enhancement of vinpocetine using self-microemulsifying drug delivery system containing long chain triglycerides: Preparation and in vitro/in vivo evaluation. Clinical Res Reg Affairs, 27:97–107.
  • Vyas TK, Shahiwala A, Amiji MM. (2008). Improved oral bioavailability and brain transport of Saquinavir upon administration in novel nanoemulsion formulations. Int J Pharm, 347:93–101.
  • Ghosh PK, Majithiya RJ, Umrethia ML, Murthy RS. (2006). Design and development of microemulsion drug delivery system of acyclovir for improvement of oral bioavailability. aaps Pharmscitech, 7:77.
  • Araya H, Tomita M, Hayashi M. (2005). The novel formulation design of O/W microemulsion for improving the gastrointestinal absorption of poorly water soluble compounds. Int J Pharm, 305:61–74.

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